Literature DB >> 18680443

Clinical pharmacology of lubiprostone, a chloride channel activator in defecation disorders.

Regina Ginzburg1, Emily M Ambizas.   

Abstract

BACKGROUND: Lubiprostone, a prostaglandin E1 derivative, was approved in January 2006 for the treatment of chronic idiopathic constipation (CIC) in adults and in April 2008 for the treatment of irritable bowel syndrome with constipation (IBS-C) in adult women.
OBJECTIVE: To review the pharmacology, efficacy and safety of lubiprostone and recommend its place in therapy for CIC and IBS-C.
METHODS: We conducted a literature search using PubMed/Medline (1966-April 2008) using the keywords lubiprostone, chronic constipation, and irritable bowel syndrome. Data provided by the manufacturer and the FDA were also reviewed.
CONCLUSION: Available literature for lubiprostone is mostly available in abstract data making it difficult to evaluate the clinical evidence. Although this medication shows promise, more information is needed to determine its place in therapy.

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Year:  2008        PMID: 18680443     DOI: 10.1517/17425255.4.8.1091

Source DB:  PubMed          Journal:  Expert Opin Drug Metab Toxicol        ISSN: 1742-5255            Impact factor:   4.481


  7 in total

1.  Ligand-controlled regiodivergent palladium-catalyzed decarboxylative allylation reaction to access α,α-difluoroketones.

Authors:  Ming-Hsiu Yang; Douglas L Orsi; Ryan A Altman
Journal:  Angew Chem Int Ed Engl       Date:  2015-01-07       Impact factor: 15.336

2.  Cu(II)-Catalyzed Unsymmetrical Dioxidation of gem-Difluoroalkenes to Generate α,α-Difluorinated-α-phenoxyketones.

Authors:  Suvajit Koley; Kaylee T Cayton; Gisela A González-Montiel; M Ramu Yadav; Douglas L Orsi; Andrew J Intelli; Paul Ha-Yeon Cheong; Ryan A Altman
Journal:  J Org Chem       Date:  2022-08-01       Impact factor: 4.198

Review 3.  Lubiprostone: in constipation-predominant irritable bowel syndrome.

Authors:  Natalie J Carter; Lesley J Scott
Journal:  Drugs       Date:  2009-06-18       Impact factor: 9.546

Review 4.  Constipation-predominant irritable bowel syndrome: a review of current and emerging drug therapies.

Authors:  Khaled A Jadallah; Susan M Kullab; David S Sanders
Journal:  World J Gastroenterol       Date:  2014-07-21       Impact factor: 5.742

5.  A comparison of linaclotide and lubiprostone dosing regimens on ion transport responses in human colonic mucosa.

Authors:  Sang Bum Kang; Ronald R Marchelletta; Harrison Penrose; Michael J Docherty; Declan F McCole
Journal:  Pharmacol Res Perspect       Date:  2015-03-13

Review 6.  Novel pharmacological therapies for management of chronic constipation.

Authors:  Marina A Gonzalez-Martinez; Nayeli X Ortiz-Olvera; Jorge Mendez-Navarro
Journal:  J Clin Gastroenterol       Date:  2014-01       Impact factor: 3.062

7.  Lubiprostone stimulates duodenal bicarbonate secretion in rats.

Authors:  Misa Mizumori; Yasutada Akiba; Jonathan D Kaunitz
Journal:  Dig Dis Sci       Date:  2009-08-06       Impact factor: 3.199

  7 in total

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