Literature DB >> 18614925

Efavirenz in human breast milk, mothers', and newborns' plasma.

Serge Schneider1, Alexandra Peltier, Alain Gras, Vic Arendt, Christine Karasi-Omes, Anastasie Mujawamariwa, Patrick C Ndimubanzi, Gilles Ndayisaba, Robert Wennig.   

Abstract

BACKGROUND AND METHODS: Highly active antiretroviral therapy with efavirenz (EFV) has been prescribed to HIV-positive pregnant women in Rwanda (HIV status 1 and CD4 cell count > 350 cells/mm) during the last trimester of pregnancy and for 6 months after delivery. The EFV concentrations in maternal plasma, breast milk and in newborns' plasma of 13 women and their children between 6 weeks and 6 months post partum are reported.
RESULTS: Results show a mean EFV plasma concentration of 6.55 mg/L in maternal plasma, 3.51 mg/L in skim milk, and 0.85 mg/L in infant plasma. Significant linear correlations between maternal plasma and skim milk (r = 0.8666, P < 0.0001) and between skim milk and infant plasma (r = 0.6646, P < 0.02) were found, but no significant correlation was observed between maternal and infant plasma concentrations (P > 0.05).
CONCLUSIONS: After 6 months of breast-feeding, no child out of the 13 had been infected with HIV and all had good psychomotor and growth development. Our results suggest that EFV may be an alternative to nevirapine (NVP) during the third trimester of pregnancy and during the breast-feeding period. Further studies on larger groups of newborns will be necessary to get a better understanding of possible prophylactic protection of the newborns by highly active antiretroviral therapy with EFV given to the mothers.

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Year:  2008        PMID: 18614925     DOI: 10.1097/QAI.0b013e31817bbc21

Source DB:  PubMed          Journal:  J Acquir Immune Defic Syndr        ISSN: 1525-4135            Impact factor:   3.731


  19 in total

1.  Stavudine concentrations in women receiving postpartum antiretroviral treatment and their breastfeeding infants.

Authors:  Jessica M Fogel; Taha E Taha; Jin Sun; Donald R Hoover; Teresa L Parsons; Johnstone J Kumwenda; Lynne M Mofenson; Mary Glenn Fowler; Craig W Hendrix; Newton I Kumwenda; Susan H Eshleman; Mark Mirochnick
Journal:  J Acquir Immune Defic Syndr       Date:  2012-08-15       Impact factor: 3.731

2.  High Rates of Baseline Drug Resistance and Virologic Failure Among ART-naive HIV-infected Children in Mali.

Authors:  Claudia S Crowell; Almoustapha I Maiga; Mariam Sylla; Babafemi Taiwo; Niaboula Kone; Assaf P Oron; Robert L Murphy; Anne-Geneviève Marcelin; Ban Traore; Djeneba B Fofana; Gilles Peytavin; Ellen G Chadwick
Journal:  Pediatr Infect Dis J       Date:  2017-11       Impact factor: 2.129

3.  The Expanding Class of Non-Nucleoside Reverse Transcriptase Inhibitors for the Treatment of HIV-1 Infection.

Authors:  Jason J Schafer; Saranyu Ravi; Evelyn V Rowland; Germin Shenoda; Nicholas Leon
Journal:  P T       Date:  2011-06

4.  Lactation-associated postpartum weight changes among HIV-infected women in Zambia.

Authors:  Pamela M Murnane; Stephen M Arpadi; Moses Sinkala; Chipepo Kankasa; Mwiya Mwiya; Prisca Kasonde; Donald M Thea; Grace M Aldrovandi; Louise Kuhn
Journal:  Int J Epidemiol       Date:  2010-05-19       Impact factor: 7.196

5.  HIV diagnostic challenges in breast-fed infants of mothers on antiretroviral therapy.

Authors:  Renate Strehlau; Maria Paximadis; Faeezah Patel; Megan Burke; Karl-Gunter Technau; Stephanie Shiau; Elaine J Abrams; Gayle G Sherman; Gillian Hunt; Johanna Ledwaba; Ahmad H Mazanderani; Caroline T Tiemessen; Louise Kuhn
Journal:  AIDS       Date:  2019-09-01       Impact factor: 4.177

6.  Nelfinavir and its active metabolite, hydroxy-t-butylamidenelfinavir (M8), are transferred in small quantities to breast milk and do not reach biologically significant concentrations in breast-feeding infants whose mothers are taking nelfinavir.

Authors:  Paul J Weidle; Clement Zeh; Amy Martin; Richard Lando; Frank Angira; Joseph Osoga; Paul Ogindo; Sonali Girde; Timothy D Minniear; Timothy K Thomas
Journal:  Antimicrob Agents Chemother       Date:  2011-08-29       Impact factor: 5.191

Review 7.  Pharmacotherapy of pediatric HIV infection.

Authors:  Natella Rakhmanina; B Ryan Phelps
Journal:  Pediatr Clin North Am       Date:  2012-08-22       Impact factor: 3.278

Review 8.  Efavirenz in the therapy of HIV infection.

Authors:  Natella Y Rakhmanina; John N van den Anker
Journal:  Expert Opin Drug Metab Toxicol       Date:  2010-01       Impact factor: 4.481

9.  Antiretroviral pharmacokinetics in mothers and breastfeeding infants from 6 to 24 weeks post-partum: results of the BAN Study.

Authors:  Amanda H Corbett; Dumbani Kayira; Nicole R White; Nicole L Davis; Athena P Kourtis; Charles Chasela; Francis Martinson; Grace Phiri; Bonaface Musisi; Deborah Kamwendo; Michael G Hudgens; Mina C Hosseinipour; Julie Ae Nelson; Sascha R Ellington; Denise J Jamieson; Charles van der Horst; Angela Kashuba
Journal:  Antivir Ther       Date:  2014-01-24

10.  Antiretroviral concentrations in breast-feeding infants of mothers receiving highly active antiretroviral therapy.

Authors:  Mark Mirochnick; Timothy Thomas; Edmund Capparelli; Clement Zeh; Diane Holland; Rose Masaba; Prisca Odhiambo; Mary Glenn Fowler; Paul J Weidle; Michael C Thigpen
Journal:  Antimicrob Agents Chemother       Date:  2008-12-29       Impact factor: 5.191

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