Literature DB >> 18441323

Cholesterol lowering is more important than pleiotropic effects of statins for endothelial function in patients with dysglycaemia and coronary artery disease.

Magnus Settergren1, Felix Böhm, Lars Rydén, John Pernow.   

Abstract

AIMS: The importance of pleiotropic effects of statins on endothelial function and inflammatory markers was investigated in patients with dysglycaemia and coronary artery disease (CAD). METHODS AND
RESULTS: Thirty-nine patients were randomized to simvastatin 80 mg daily (S80; n = 20) or ezetimibe 10 mg and simvastatin 10 mg daily (E10/S10; n = 19) for 6 weeks, aiming at similar cholesterol reduction. Endothelial function, evaluated by brachial artery flow-mediated vasodilatation (FMD) and the effect of endothelin receptor blockade, serum lipids, and inflammatory markers were evaluated at baseline and follow-up. At follow-up, low-density lipoprotein cholesterol decreased from 3.1 (2.8-3.4) (median and quartiles) to 1.5 mmol/L (1.4-1.7) and from 3.0 (2.5-3.4) to 1.3 mmol/L (1.1-1.8), in the S80 and E10/S10 groups, respectively. In the entire study group, FMD increased from 4.3% (3.4-6.1) at baseline to 5.5% (3.4-6.6) at follow-up, while C-reactive protein decreased from 3.1 (1.7-7.6) to 2.3 mg/L (0.9-6.5). The changes in FMD and C-reactive protein from baseline to follow-up were not significantly different between patients on S80 and E10/S10 groups. Endothelin blockade enhanced endothelium-dependent vasodilatation both at baseline and follow-up.
CONCLUSION: Lipid lowering is more important than pleiotropic effects of statins for improvement in endothelial function and inflammatory markers in patients with dysglycaemia and CAD.

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Year:  2008        PMID: 18441323     DOI: 10.1093/eurheartj/ehn166

Source DB:  PubMed          Journal:  Eur Heart J        ISSN: 0195-668X            Impact factor:   29.983


  17 in total

1.  Effect of treatment with pravastatin or ezetimibe on endothelial function in patients with moderate hypercholesterolemia.

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2.  The endothelin receptor antagonist bosentan improves peripheral endothelial function in patients with type 2 diabetes mellitus and microalbuminuria: a randomised trial.

Authors:  A Rafnsson; F Böhm; M Settergren; A Gonon; K Brismar; J Pernow
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3.  [Achievement of blood lipid target levels with Ezetimibe/Simvastatin in patients with atherosclerosis and/or diabetes mellitus--an Austrian observational study].

Authors:  Jörg Slany
Journal:  Wien Med Wochenschr       Date:  2009

4.  Association between chronic caregiving stress and impaired endothelial function in the elderly.

Authors:  Brent T Mausbach; Susan K Roepke; Michael G Ziegler; Milos Milic; Roland von Känel; Joel E Dimsdale; Paul J Mills; Thomas L Patterson; Matthew A Allison; Sonia Ancoli-Israel; Igor Grant
Journal:  J Am Coll Cardiol       Date:  2010-06-08       Impact factor: 24.094

5.  High-dose simvastatin exhibits enhanced lipid-lowering effects relative to simvastatin/ezetimibe combination therapy.

Authors:  Stuart G Snowden; Dmitry Grapov; Magnus Settergren; Fabio Luiz D'Alexandri; Jesper Z Haeggström; Oliver Fiehn; Tuulia Hyötyläinen; Theresa L Pedersen; John W Newman; Matej Orešič; John Pernow; Craig E Wheelock
Journal:  Circ Cardiovasc Genet       Date:  2014-12

6.  Comparison of Efficacy and Safety of Statin-Ezetimibe Combination Therapy with Statin Monotherapy in Patients with Diabetes: A Meta-Analysis of Randomized Controlled Studies.

Authors:  Kwang-Hee Shin; Hye Duck Choi
Journal:  Am J Cardiovasc Drugs       Date:  2021-12-20       Impact factor: 3.283

7.  Evidence for statin pleiotropy in humans: differential effects of statins and ezetimibe on rho-associated coiled-coil containing protein kinase activity, endothelial function, and inflammation.

Authors:  Ping-Yen Liu; Yen-Wen Liu; Li-Jen Lin; Jyh-Hong Chen; James K Liao
Journal:  Circulation       Date:  2008-12-15       Impact factor: 29.690

Review 8.  Renal endothelial dysfunction in diabetic nephropathy.

Authors:  Huifang Cheng; Raymond C Harris
Journal:  Cardiovasc Hematol Disord Drug Targets       Date:  2014

Review 9.  Impact of ezetimibe on atherosclerosis: is the jury still out?

Authors:  Firas J Al Badarin; Iftikhar J Kullo; Stephen L Kopecky; Randal J Thomas
Journal:  Mayo Clin Proc       Date:  2009-04       Impact factor: 7.616

Review 10.  Vascular inflammation and low-density lipoproteins: is cholesterol the link? A lesson from the clinical trials.

Authors:  Alberico Luigi Catapano; Angela Pirillo; Giuseppe Danilo Norata
Journal:  Br J Pharmacol       Date:  2017-05-05       Impact factor: 8.739

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