Literature DB >> 18431653

Effect of drug lipophilicity and ionization on permeability across the buccal mucosa: a technical note.

Amit Kokate1, Xiaoling Li, Bhaskara Jasti.   

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Year:  2008        PMID： 18431653      PMCID： PMC2976956          DOI： 10.1208/s12249-008-9071-7

Source DB:  PubMed          Journal:  AAPS PharmSciTech        ISSN： 1530-9932            Impact factor:   3.246


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  16 in total

1.  The composite solubility versus pH profile and its role in intestinal absorption prediction.

Authors:  Barry A Hendriksen; Manuel V Sanchez Felix; Michael B Bolger
Journal:  AAPS PharmSci       Date:  2003

2.  Estimation of intradermal disposition kinetics of drugs: II. Factors determining penetration of drugs from viable skin to muscular layer.

Authors:  Kazutaka Higaki; Masahide Asai; Takayuki Suyama; Kazuki Nakayama; Ken-ichi Ogawara; Toshikiro Kimura
Journal:  Int J Pharm       Date:  2002-06-04       Impact factor: 5.875

Review 3.  Drug permeation in biomembranes: in vitro and in silico prediction and influence of physicochemical properties.

Authors:  Annika Mälkiä; Lasse Murtomäki; Arto Urtti; Kyösti Kontturi
Journal:  Eur J Pharm Sci       Date:  2004-09       Impact factor: 4.384

4.  ADME evaluation in drug discovery. 5. Correlation of Caco-2 permeation with simple molecular properties.

Authors:  T J Hou; W Zhang; K Xia; X B Qiao; X J Xu
Journal:  J Chem Inf Comput Sci       Date:  2004 Sep-Oct

5.  Effect of thermodynamic activities of the unionized and ionized species on drug flux across buccal mucosa.

Authors:  Amit Kokate; Xiaoling Li; Parminder Singh; Bhaskara R Jasti
Journal:  J Pharm Sci       Date:  2008-10       Impact factor: 3.534

6.  Corneal penetration behavior of beta-blocking agents I: Physiochemical factors.

Authors:  R D Schoenwald; H S Huang
Journal:  J Pharm Sci       Date:  1983-11       Impact factor: 3.534

7.  pH, pK(a) and dermal delivery.

Authors:  J Hadgraft; C Valenta
Journal:  Int J Pharm       Date:  2000-05-10       Impact factor: 5.875

8.  Transbuccal delivery of acyclovir: I. In vitro determination of routes of buccal transport.

Authors:  A H Shojaei; B Berner; L Xiaoling
Journal:  Pharm Res       Date:  1998-08       Impact factor: 4.200

Review 9.  Cellular and molecular basis of barrier function in oral epithelium.

Authors:  P W Wertz; C A Squier
Journal:  Crit Rev Ther Drug Carrier Syst       Date:  1991       Impact factor: 4.889

10.  Lipid content and water permeability of skin and oral mucosa.

Authors:  C A Squier; P Cox; P W Wertz
Journal:  J Invest Dermatol       Date:  1991-01       Impact factor: 8.551
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Journal:  J Med Chem       Date:  2019-01-03       Impact factor: 7.446

3.  Mucoadhesive Electrospun Patch Delivery of Lidocaine to the Oral Mucosa and Investigation of Spatial Distribution in a Tissue Using MALDI-Mass Spectrometry Imaging.

Authors:  Katharina H Clitherow; Craig Murdoch; Sebastian Guy Spain; Anna Mette Handler; Helen E Colley; Mai Bay Stie; Hanne Mørck Nielsen; Christian Janfelt; Paul V Hatton; Jette Jacobsen
Journal:  Mol Pharm       Date:  2019-08-15       Impact factor: 4.939

4.  Development and Evaluation of a Physiologically Based Pharmacokinetic Drug-Disease Model of Propranolol for Suggesting Model Informed Dosing in Liver Cirrhosis Patients.

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Journal:  Drug Des Devel Ther       Date:  2021-03-17       Impact factor: 4.162

5.  Perspectives of Positively Charged Nanocrystals of Tedizolid Phosphate as a Topical Ocular Application in Rabbits.

Authors:  Abdullah Alshememry; Musaed Alkholief; Mohd Abul Kalam; Mohammad Raish; Raisuddin Ali; Sulaiman S Alhudaithi; Muzaffar Iqbal; Aws Alshamsan
Journal:  Molecules       Date:  2022-07-20       Impact factor: 4.927
  5 in total

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