Literature DB >> 18414865

Phase I clinical and pharmacokinetic study of oxaliplatin, irinotecan and capecitabine.

Smitha S Krishnamurthi1, Joanna M Brell, Charles L Hoppel, Merrill J Egorin, Karen C Weaver, Xiaolin Li, Stephen T Ingalls, Eleanor G Zuhowski, Mark D Schluchter, Afshin Dowlati, Matthew M Cooney, Joseph Gibbons, Beth A Overmoyer, S Percy Ivy, Scot C Remick.   

Abstract

PURPOSE: To determine the maximum tolerated dose (MTD) and dose-limiting toxicity (DLT) of the combination of weekly oxaliplatin x 4, weekly irinotecan x 4 and capecitabine Monday through Friday for 4 weeks of every 6 week cycle in patients with solid tumors; to determine the pharmacokinetic profile of these agents in this combination; to observe patients for clinical anti-tumor response.
METHODS: Twenty-two patients with metastatic solid tumors received oxaliplatin 60 mg/m(2) weekly x 4, irinotecan beginning at a dose of 40 mg/m(2) weekly x 4, and capecitabine Monday through Friday for 4 weeks of every 6 week cycle, initially at 1,000 mg twice daily (bid).
RESULTS: The MTD was oxaliplatin 60 mg/m(2) weekly x 4, irinotecan 50 mg/m(2) weekly x 4 and capecitabine 450 mg bid Monday through Friday for 4 weeks of every 6 week cycle. One of six patients at this dose level developed DLT of nausea, vomiting, and diarrhea. Among patients treated with a constant capecitabine dose of 450 mg bid, there was a higher mean AUC of 5-FU in women than in men (mean +/- SD: 892 +/- 287 nM h vs. 537 +/- 182 nM h; Mann-Whitney two-tailed, P = 0.02). There was one complete response in a patient with gastric cancer.
CONCLUSION: The novel schedule of weekly oxaliplatin, weekly irinotecan, and capecitabine Monday through Friday, all administered for 4 weeks of every 6 week cycle, evaluated in this phase I trial is well-tolerated and demonstrated activity in a patient with gastric cancer.

Entities:  

Mesh:

Substances:

Year:  2008        PMID: 18414865      PMCID: PMC4788493          DOI: 10.1007/s00280-008-0754-2

Source DB:  PubMed          Journal:  Cancer Chemother Pharmacol        ISSN: 0344-5704            Impact factor:   3.333


  39 in total

1.  Preliminary studies of a novel oral fluoropyrimidine carbamate: capecitabine.

Authors:  D R Budman; N J Meropol; B Reigner; P J Creaven; S M Lichtman; E Berghorn; J Behr; R J Gordon; B Osterwalder; T Griffin
Journal:  J Clin Oncol       Date:  1998-05       Impact factor: 44.544

2.  Phase I and pharmacokinetic study of oral irinotecan given once daily for 5 days every 3 weeks in combination with capecitabine in patients with solid tumors.

Authors:  Otto Soepenberg; Herlinde Dumez; Jaap Verweij; Dorothee Semiond; Maja J A deJonge; Ferry A L M Eskens; Judith ter Steeg; Johan Selleslach; Sylvie Assadourian; Ger-Jan Sanderink; Alex Sparreboom; A T van Oosterom
Journal:  J Clin Oncol       Date:  2005-02-01       Impact factor: 44.544

Review 3.  Clinical pharmacokinetics and metabolism of irinotecan (CPT-11).

Authors:  R H Mathijssen; R J van Alphen; J Verweij; W J Loos; K Nooter; G Stoter; A Sparreboom
Journal:  Clin Cancer Res       Date:  2001-08       Impact factor: 12.531

4.  Oxaliplatin as single agent in previously untreated colorectal carcinoma patients: a phase II multicentric study.

Authors:  E Díaz-Rubio; J Sastre; A Zaniboni; R Labianca; H Cortés-Funes; F de Braud; C Boni; M Benavides; G Dallavalle; M Homerin
Journal:  Ann Oncol       Date:  1998-01       Impact factor: 32.976

5.  Cellular interactions of 5-fluorouracil and the camptothecin analogue CPT-11 (irinotecan) in a human colorectal carcinoma cell line.

Authors:  S Guichard; I Hennebelle; R Bugat; P Canal
Journal:  Biochem Pharmacol       Date:  1998-03-01       Impact factor: 5.858

6.  Efficacy of intravenous continuous infusion of fluorouracil compared with bolus administration in advanced colorectal cancer.

Authors:  P Piedbois; P Rougier; M Buyse; J Pignon; L Ryan; R Hansen; B Zee; B Weinerman; J Pater; C Leichman; J Macdonald; J Benedetti; J Lokich; J Fryer; G Brufman; R Isacson; A Laplanche; E Levy
Journal:  J Clin Oncol       Date:  1998-01       Impact factor: 44.544

7.  Efficient nucleotide excision repair of cisplatin, oxaliplatin, and Bis-aceto-ammine-dichloro-cyclohexylamine-platinum(IV) (JM216) platinum intrastrand DNA diadducts.

Authors:  J T Reardon; A Vaisman; S G Chaney; A Sancar
Journal:  Cancer Res       Date:  1999-08-15       Impact factor: 12.701

8.  Biweekly intensified ambulatory chronomodulated chemotherapy with oxaliplatin, fluorouracil, and leucovorin in patients with metastatic colorectal cancer.

Authors:  F Bertheault-Cvitkovic; A Jami; M Ithzaki; P D Brummer; S Brienza; R Adam; F Kunstlinger; H Bismuth; J L Misset; F Lévi
Journal:  J Clin Oncol       Date:  1996-11       Impact factor: 44.544

9.  Women experience greater toxicity with fluorouracil-based chemotherapy for colorectal cancer.

Authors:  Jeff A Sloan; Richard M Goldberg; Daniel J Sargent; Delfino Vargas-Chanes; Suresh Nair; Steven S Cha; Paul J Novotny; Michael A Poon; Michael J O'Connell; Charles L Loprinzi
Journal:  J Clin Oncol       Date:  2002-03-15       Impact factor: 44.544

10.  Phase I study of weekly oxaliplatin plus irinotecan in previously treated patients with metastatic colorectal cancer.

Authors:  N Kemeny; W Tong; M Gonen; J Stockman; C Di Lauro; J Teitcher; P White; C Price; L Saltz; S Sharma; M A Graham
Journal:  Ann Oncol       Date:  2002-09       Impact factor: 32.976

View more
  3 in total

1.  A Phase Ib pharmacokinetic study of the anti-angiogenic agent CKD-732 used in combination with capecitabine and oxaliplatin (XELOX) in metastatic colorectal cancer patients who progressed on irinotecan-based chemotherapy.

Authors:  Sang Joon Shin; Joong Bae Ahn; Kyung Soo Park; Yoon Jung Lee; Yong Sang Hong; Tae Won Kim; Hye Ryun Kim; Sun Young Rha; Jae Kyung Roh; Dal-Hyun Kim; Chin Kim; Hyun Cheol Chung
Journal:  Invest New Drugs       Date:  2010-12-29       Impact factor: 3.850

2.  Phase I Clinical Trials in Patients ≥80.

Authors:  Himabindu Gaddipati; Pingfu Fu; Afshin Dowlati
Journal:  J Geriatr Oncol       Date:  2011-04-01       Impact factor: 3.599

3.  A multi-center phase II study of oxaliplatin, irinotecan, and capecitabine in advanced gastric/gastroesophageal junction carcinoma.

Authors:  Joanna M Brell; Smitha S Krishnamurthi; Milind Javle; Joel Saltzman; Ira Wollner; Robert Pelley; Afshin Dowlati; Belagodu N Kantharaj; Mark D Schluchter; Linda Rath; S Percy Ivy; Scot C Remick
Journal:  Cancer Chemother Pharmacol       Date:  2008-08-01       Impact factor: 3.333

  3 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.