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5 in total

1. Design, synthesis, docking, and biological evaluation of novel diazide-containing isoxazole- and pyrazole-based histone deacetylase probes.

Authors: Raghupathi Neelarapu; Denise L Holzle; Subash Velaparthi; He Bai; Michael Brunsteiner; Sylvie Y Blond; Pavel A Petukhov
Journal: J Med Chem Date: 2011-06-02 Impact factor: 7.446

2. Beyond picomolar affinities: quantitative aspects of noncovalent and covalent binding of drugs to proteins.

Authors: Adam J T Smith; Xiyun Zhang; Andrew G Leach; K N Houk
Journal: J Med Chem Date: 2009-01-22 Impact factor: 7.446

3. Binding ensemble profiling with photoaffinity labeling (BEProFL) approach: mapping the binding poses of HDAC8 inhibitors.

Authors: Bai He; Subash Velaparthi; Gilles Pieffet; Chris Pennington; Aruna Mahesh; Denise L Holzle; Michael Brunsteiner; Richard van Breemen; Sylvie Y Blond; Pavel A Petukhov
Journal: J Med Chem Date: 2009-11-26 Impact factor: 7.446

4. Novel hybrid molecule overcomes the limited response of solid tumours to HDAC inhibitors via suppressing JAK1-STAT3-BCL2 signalling.

Authors: Zhi Huang; Wei Zhou; Yongtao Li; Mei Cao; Tianqi Wang; Yakun Ma; Qingxiang Guo; Xin Wang; Chao Zhang; Chenglan Zhang; Wenzhi Shen; Yanhua Liu; Yanan Chen; Jianyu Zheng; Shengyong Yang; Yan Fan; Rong Xiang
Journal: Theranostics Date: 2018-10-05 Impact factor: 11.556

5. In search of constrained FTY720 and phytosphingosine analogs as dual acting anticancer agents targeting metabolic and epigenetic pathways.

Authors: Jean-Baptiste Garsi; Lorenzo Sernissi; Vito Vece; Stephen Hanessian; Alison N McCracken; Grigor Simitian; Aimee L Edinger
Journal: Eur J Med Chem Date: 2018-09-21 Impact factor: 6.514

5 in total