Literature DB >> 18238889

The use of trough ribavirin concentration to predict sustained virological response and haematological toxicity in HIV/HCV-co-infected patients treated with ribavirin and pegylated interferon.

D Aguilar Marucco1, D Gonzalez de Requena, S Bonora, C Tettoni, M Bonasso, T De Blasi, A D'Avolio, M Sciandra, M Siccardi, L Baietto, L Trentini, A Sinicco, G Cariti, G Di Perri.   

Abstract

OBJECTIVES: To study the association between trough ribavirin concentration (C(trough)) with sustained virological response (SVR) and haemoglobin (Hb) decrease in HIV/hepatitis C virus (HCV)-co-infected (HIV+/HCV+) patients treated with anti-HCV therapy.
METHODS: HIV+/HCV+ patients treated with ribavirin and pegylated interferon were prospectively evaluated. Qualitative and quantitative HCV-RNA, Hb levels and ribavirin C(trough) were measured at baseline and weeks 2, 4, 12, 24, 36 and 48 during therapy. HCV-RNA was also measured at 24 weeks after the end of therapy. Efficacy analysis was performed on patients with a definitive virological outcome (SVR, relapser and non-responder), whereas for toxicity analysis, dropouts were considered until the last available observation.
RESULTS: Fifty-two patients (54.7% with genotype 1 or 4) were included. Overall, no correlation between ribavirin C(trough) and early virological response (EVR) nor SVR was found. However, in patients with genotype 1 or 4, ribavirin C(trough) was independently associated with EVR (P = 0.036) and SVR (P = 0.046). A ribavirin C(trough) cut-off of 1600 ng/mL was found to be associated with both EVR (chi(2) = 5.69, P = 0.028) and SVR (chi(2)=4.2, P = 0.04). Higher ribavirin C(trough) correlated with Hb decrease (R = -0.361, P = 0.009) and was independently associated with an Hb decrease of >4 g/dL (P = 0.009). Receiver operating characteristic (ROC) analysis indicated that a ribavirin C(trough) of >2300 ng/mL was associated with an Hb decrease of >4 g/dL (chi(2) = 8.08, P = 0.01).
CONCLUSIONS: Our study confirmed a relationship between ribavirin exposure and both efficacy and toxicity. Moreover, we found ribavirin C(trough) cut-offs for both SVR in genotypes 1 and 4 and overall haematological toxicity. These findings deserve further clinical evaluation.

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Year:  2008        PMID: 18238889     DOI: 10.1093/jac/dkn013

Source DB:  PubMed          Journal:  J Antimicrob Chemother        ISSN: 0305-7453            Impact factor:   5.790


  10 in total

Review 1.  A pharmacological profile of ribavirin and monitoring of its plasma concentration in chronic hepatitis C infection.

Authors:  Girish S Naik; Manoj G Tyagi
Journal:  J Clin Exp Hepatol       Date:  2012-04-12

2.  Telaprevir and ribavirin interaction: higher ribavirin levels are not only due to renal dysfunction during triple therapy.

Authors:  Alicia Gutierrez-Valencia; Rosa Ruiz-Valderas; Omar J Ben-Marzouk-Hidalgo; Almudena Torres-Cornejo; Nuria Espinosa; Juan R Castillo-Ferrando; Pompeyo Viciana; Luis F Lopez-Cortes
Journal:  Antimicrob Agents Chemother       Date:  2015-03-23       Impact factor: 5.191

3.  Cell type mediated resistance of vesicular stomatitis virus and Sendai virus to ribavirin.

Authors:  Nirav R Shah; Amanda Sunderland; Valery Z Grdzelishvili
Journal:  PLoS One       Date:  2010-06-22       Impact factor: 3.240

4.  Plasma ribavirin trough concentrations at week 4 predict hepatitis C virus (HCV) relapse in HIV-HCV-coinfected patients treated for chronic hepatitis C.

Authors:  Judit Morello; Vincent Soriano; Pablo Barreiro; José Medrano; Antonio Madejón; Gema González-Pardo; Inmaculada Jiménez-Nácher; Juan González-Lahoz; Sonia Rodríguez-Novoa
Journal:  Antimicrob Agents Chemother       Date:  2010-01-25       Impact factor: 5.191

5.  Lower ribavirin biodisponibility in patients with HIV-HCV coinfection in comparison with HCV monoinfected patients.

Authors:  Giorgiana Hatu; François Bailly; Emmanuel Pourcelot; Pierre Pradat; Patrick Miailhes; Marianne Maynard; François Parant; Pierre Chiarello; Jean-Michel Livrozet; Fabien Zoulim; Marie-Claude Gagnieu
Journal:  BMC Infect Dis       Date:  2014-03-20       Impact factor: 3.090

6.  Liver decompensation predicts ribavirin overexposure in hepatitis C virus patients treated with direct-acting antivirals.

Authors:  Viola Guardigni; Lorenzo Badia; Matteo Conti; Matteo Rinaldi; Rita Mancini; Pierluigi Viale; Gabriella Verucchi
Journal:  World J Hepatol       Date:  2017-12-08

Review 7.  Antimicrobial therapeutic drug monitoring in critically ill adult patients: a Position Paper.

Authors:  Mohd H Abdul-Aziz; Jan-Willem C Alffenaar; Matteo Bassetti; Hendrik Bracht; George Dimopoulos; Deborah Marriott; Michael N Neely; Jose-Artur Paiva; Federico Pea; Fredrik Sjovall; Jean F Timsit; Andrew A Udy; Sebastian G Wicha; Markus Zeitlinger; Jan J De Waele; Jason A Roberts
Journal:  Intensive Care Med       Date:  2020-05-07       Impact factor: 17.440

8.  Improved HPLC method for the determination of ribavirin concentration in red blood cells and its application in patients with COVID-19.

Authors:  Liang Liu; Sixun Guo; Chunli Che; Quanming Su; Deqiu Zhu; Xin Hai
Journal:  Biomed Chromatogr       Date:  2022-03-31       Impact factor: 1.911

Review 9.  Treatment outcomes of treatment-naïve Hepatitis C patients co-infected with HIV: a systematic review and meta-analysis of observational cohorts.

Authors:  Anna Davies; Kasha P Singh; Zara Shubber; Philipp Ducros; Edward J Mills; Graham Cooke; Nathan Ford
Journal:  PLoS One       Date:  2013-02-05       Impact factor: 3.240

10.  Ribavirin Concentrations Do Not Predict Sustained Virological Response in HIV/HCV-Coinfected Patients Treated with Ribavirin and Pegylated Interferon in the Swiss HIV Cohort Study.

Authors:  Helen Kovari; Stefan Russmann; Bruno Ledergerber; Daniel Müller; Margalida Rotger; Pablo Velli; Matthias Cavassini; Juan Ambrosioni; Andrea Bregenzer; Marcel Stöckle; Enos Bernasconi; Andri Rauch; Roberto F Speck
Journal:  PLoS One       Date:  2015-07-28       Impact factor: 3.240

  10 in total

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