Literature DB >> 17986638

Insulin secretion and clearance after subacute estradiol administration in postmenopausal women.

Rachael E Van Pelt1, Robert S Schwartz, Wendy M Kohrt.   

Abstract

CONTEXT: Data from large clinical trials of postmenopausal women suggest that the incidence of diabetes is reduced in women randomized to estrogen-based hormone therapy when compared with placebo. Whether this is due to an effect of estrogen on insulin or glucose metabolism remains unclear.
OBJECTIVE: Our objective was to test the hypothesis that estradiol (E(2)) increases insulin secretion and clearance.
DESIGN: Serum insulin and C-peptide (CPEP) responses to hyperglycemia (250 mg/dl) plus iv L-arginine were measured on 2 separate days, with (EST) and without [control (CON)] subacute (24 h) transdermal E(2) administration. STUDY PARTICIPANTS: There were 11 postmenopausal women (mean +/- sd; 55 +/- 4 yr) included in this study. MAIN OUTCOMES: Insulin secretion and clearance were estimated from the CPEP area under the curve and the molar ratio of CPEP to insulin area under the curve, respectively. Mean glucose disposal rate (GDR) was estimated from the rate of glucose infusion during the final 30 min of the hyperglycemic clamp.
RESULTS: There were no differences in insulin secretion or clearance between the EST and CON days. Fasting glucose was lower on the EST compared with the CON (93 +/- 6 vs. 98 +/- 8 mg/dl), but mean GDR was not different. However, when one outlier was excluded from analysis, GDR was increased after EST compared with CON. Furthermore, a strong inverse association was observed between years since menopause and E(2)-mediated changes in GDR (r = -0.794; P = 0.004).
CONCLUSIONS: Contrary to our hypothesis, 24-h transdermal E(2) administration did not alter insulin secretion or clearance in postmenopausal women. However, a longer time since menopause was associated with a reduced effect of E(2) to increase glucose uptake.

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Year:  2007        PMID: 17986638      PMCID: PMC2243232          DOI: 10.1210/jc.2007-1657

Source DB:  PubMed          Journal:  J Clin Endocrinol Metab        ISSN: 0021-972X            Impact factor:   5.958


  40 in total

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2.  Estrogen causes dynamic alterations in endothelial estrogen receptor expression.

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4.  Effects of oral and transdermal 17beta-estradiol with cyclical oral norethindrone acetate on insulin sensitivity, secretion, and elimination in postmenopausal women.

Authors:  C P Spencer; I F Godsland; A J Cooper; D Ross; M I Whitehead; J C Stevenson
Journal:  Metabolism       Date:  2000-06       Impact factor: 8.694

5.  Long-term effects of oral estradiol and dydrogesterone on carbohydrate metabolism in postmenopausal women.

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6.  Effects of peroral and transdermal oestrogen replacement therapy on glucose and insulin metabolism.

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8.  Effect of postmenopausal oestradiol and dydrogesterone therapy on lipoproteins and insulin sensitivity, secretion and elimination in hysterectomised women.

Authors:  N A Manassiev; I F Godsland; D Crook; A J Proudler; M I Whitehead; J C Stevenson
Journal:  Maturitas       Date:  2002-07-25       Impact factor: 4.342

9.  Evidence that oestrogen receptor-alpha plays an important role in the regulation of glucose homeostasis in mice: insulin sensitivity in the liver.

Authors:  G Bryzgalova; H Gao; B Ahren; J R Zierath; D Galuska; T L Steiler; K Dahlman-Wright; S Nilsson; J-A Gustafsson; S Efendic; A Khan
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10.  Efficacy and safety of oral and transdermal hormonal replacement treatment containing levonorgestrel.

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  7 in total

Review 1.  Regulation of Body Composition and Bioenergetics by Estrogens.

Authors:  Rachael E Van Pelt; Kathleen M Gavin; Wendy M Kohrt
Journal:  Endocrinol Metab Clin North Am       Date:  2015-06-20       Impact factor: 4.741

2.  Acute estradiol treatment reduces skeletal muscle protein breakdown markers in early- but not late-postmenopausal women.

Authors:  Young-Min Park; Amy C Keller; Shauna S Runchey; Benjamin F Miller; Wendy M Kohrt; Rachael E Van Pelt; Chounghun Kang; Catherine M Jankowski; Kerrie L Moreau
Journal:  Steroids       Date:  2019-03-27       Impact factor: 2.668

3.  Timing of Estradiol Treatment After Menopause May Determine Benefit or Harm to Insulin Action.

Authors:  R I Pereira; B A Casey; T A Swibas; C B Erickson; P Wolfe; R E Van Pelt
Journal:  J Clin Endocrinol Metab       Date:  2015-10-01       Impact factor: 5.958

Review 4.  Menopausal Hormone Therapy and Type 2 Diabetes Prevention: Evidence, Mechanisms, and Clinical Implications.

Authors:  Franck Mauvais-Jarvis; JoAnn E Manson; John C Stevenson; Vivian A Fonseca
Journal:  Endocr Rev       Date:  2017-06-01       Impact factor: 19.871

Review 5.  Body composition and cardiometabolic health across the menopause transition.

Authors:  Kara L Marlatt; Dori R Pitynski-Miller; Kathleen M Gavin; Kerrie L Moreau; Edward L Melanson; Nanette Santoro; Wendy M Kohrt
Journal:  Obesity (Silver Spring)       Date:  2022-01       Impact factor: 5.002

6.  Estradiol-mediated improvements in adipose tissue insulin sensitivity are related to the balance of adipose tissue estrogen receptor α and β in postmenopausal women.

Authors:  Young-Min Park; Rocio I Pereira; Christopher B Erickson; Tracy A Swibas; Kimberly A Cox-York; Rachael E Van Pelt
Journal:  PLoS One       Date:  2017-05-04       Impact factor: 3.240

7.  Time since menopause and skeletal muscle estrogen receptors, PGC-1α, and AMPK.

Authors:  Young-Min Park; Rocio I Pereira; Christopher B Erickson; Tracy A Swibas; Chounghun Kang; Rachael E Van Pelt
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  7 in total

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