Literature DB >> 17944472

Tethering small molecules to a phage display library: discovery of a selective bivalent inhibitor of protein kinase A.

Scott C Meyer1, Carolyn D Shomin, Thomas Gaj, Indraneel Ghosh.   

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Year:  2007        PMID： 17944472     DOI： 10.1021/ja076197d

Source DB:  PubMed          Journal:  J Am Chem Soc        ISSN： 0002-7863            Impact factor:   15.419


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  23 in total

1.  Targeting diverse signaling interaction sites allows the rapid generation of bivalent kinase inhibitors.

Authors:  Zachary B Hill; B Gayani K Perera; Simeon S Andrews; Dustin J Maly
Journal:  ACS Chem Biol       Date:  2011-12-22       Impact factor: 5.100

2.  Selection of cyclic-peptide inhibitors targeting Aurora kinase A: problems and solutions.

Authors:  Carolyn D Shomin; Elizabeth Restituyo; Kurt J Cox; Indraneel Ghosh
Journal:  Bioorg Med Chem       Date:  2011-09-29       Impact factor: 3.641

Review 3.  Progress in phage display: evolution of the technique and its application.

Authors:  Tomaz Bratkovic
Journal:  Cell Mol Life Sci       Date:  2010-03       Impact factor: 9.261

Review 4.  Targeting kinase signaling pathways with constrained peptide scaffolds.

Authors:  Laura E Hanold; Melody D Fulton; Eileen J Kennedy
Journal:  Pharmacol Ther       Date:  2017-02-07       Impact factor: 12.310

5.  Synthetic pathway for production of five-carbon alcohols from isopentenyl diphosphate.

Authors:  Howard H Chou; Jay D Keasling
Journal:  Appl Environ Microbiol       Date:  2012-08-31       Impact factor: 4.792

Review 6.  Bivalent inhibitors of protein kinases.

Authors:  Carrie M Gower; Matthew E K Chang; Dustin J Maly
Journal:  Crit Rev Biochem Mol Biol       Date:  2014-02-25       Impact factor: 8.250

7.  Iterative in situ click chemistry assembles a branched capture agent and allosteric inhibitor for Akt1.

Authors:  Steven W Millward; Ryan K Henning; Gabriel A Kwong; Suresh Pitram; Heather D Agnew; Kaycie M Deyle; Arundhati Nag; Jason Hein; Su Seong Lee; Jaehong Lim; Jessica A Pfeilsticker; K Barry Sharpless; James R Heath
Journal:  J Am Chem Soc       Date:  2011-10-24       Impact factor: 15.419

8.  Genetically encoded fragment-based discovery of glycopeptide ligands for carbohydrate-binding proteins.

Authors:  Simon Ng; Edith Lin; Pavel I Kitov; Katrina F Tjhung; Oksana O Gerlits; Lu Deng; Brian Kasper; Amika Sood; Beth M Paschal; Ping Zhang; Chang-Chun Ling; John S Klassen; Christopher J Noren; Lara K Mahal; Robert J Woods; Leighton Coates; Ratmir Derda
Journal:  J Am Chem Soc       Date:  2015-04-16       Impact factor: 15.419

9.  Protein-Protein Interactions as New Targets for Ion Channel Drug Discovery.

Authors:  Svetla Stoilova-McPhie; Syed Ali; Fernanda Laezza
Journal:  Austin J Pharmacol Ther       Date:  2013-12-31

10.  An efficient strategy to enhance binding affinity and specificity of a known isozyme inhibitor.

Authors:  Joo-Eun Jee; Jaehong Lim; Yong Siang Ong; Jessica Oon; Liqian Gao; Hak Soo Choi; Su Seong Lee
Journal:  Org Biomol Chem       Date:  2016-07-12       Impact factor: 3.876
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