Literature DB >> 17896040

Solid-phase based synthesis of jasplakinolide analogs by intramolecular azide-alkyne cycloadditions.

Tai-Shan Hu1, René Tannert, Hans-Dieter Arndt, Herbert Waldmann.   

Abstract

The synthesis of a focused library of jasplakinolide analogs with a 1,2,3-triazole in place of an E-configured double bond is described, featuring the Cu(I) catalyzed azide-alkyne cycloaddition reaction as an efficient macrocyclization tool.

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Year:  2007        PMID： 17896040     DOI： 10.1039/b710650e

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  4 in total

1.  Synthesis of chondramide A analogues with modified β-tyrosine and their biological evaluation.

Authors:  Alexander Zhdanko; Anke Schmauder; Christopher I Ma; L David Sibley; David Sept; Florenz Sasse; Martin E Maier
Journal:  Chemistry       Date:  2011-10-20       Impact factor: 5.236

2.  Synthesis and biological evaluation of new jasplakinolide (jaspamide) analogs.

Authors:  Arun K Ghosh; Zachary L Dawson; Deuk Kyu Moon; Ruoli Bai; Ernest Hamel
Journal:  Bioorg Med Chem Lett       Date:  2010-07-11       Impact factor: 2.823

3.  Cyclodepsipeptides from marine sponges: natural agents for drug research.

Authors:  Gowri Shankar Bagavananthem Andavan; Rosa Lemmens-Gruber
Journal:  Mar Drugs       Date:  2010-03-22       Impact factor: 5.118

Review 4.  Macrocyclic drugs and synthetic methodologies toward macrocycles.

Authors:  Xufen Yu; Dianqing Sun
Journal:  Molecules       Date:  2013-05-24       Impact factor: 4.411
  4 in total

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