Literature DB >> 17875108

Compatibility and stability of tramadol and dexamethasone in solution and its use in terminally ill patients.

S Negro1, A Salama, Y Sánchez, M L Azuara, E Barcia.   

Abstract

BACKGROUND: Delivery of drug admixtures by continuous subcutaneous infusion is common practice in palliative medicine, but analytical confirmation of their compatibility and stability is not always available.
OBJECTIVE: To study the compatibility and stability of tramadol hydrochloride and dexamethasone sodium phosphate combined in solution and to report on its use in terminally ill patients.
METHOD: Twelve different solutions containing tramadol hydrochloride (8.33-33.33 mg/mL) and dexamethasone sodium phosphate (0.33-3.33 mg/mL) were prepared in saline and stored in polypropylene syringes for 5 days (25 degrees C). Analysis was performed on days 1, 3 and 5 days with simultaneous determination by HPLC. pH was measured at 0 and 5 days. Clinical performance was assessed retrospectively in six terminal-ill oncology patients.
RESULTS: Maximum losses of 7% and 6% were observed for tramadol and dexamethasone. Pain was completely controlled in four patients. Local tolerance resulted in haematoma in three patients, which resolved by switching to a butterfly insertion site.
CONCLUSION: Tramadol hydrochloride (100-400 mg/day) and dexamethasone sodium phosphate (4-40 mg/day) are stable for at least 5 days when combined in saline and stored at 25 degrees C. These results are only valid for the type of syringes and the specific commercial preparations tested.

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Year:  2007        PMID: 17875108     DOI: 10.1111/j.1365-2710.2007.00839.x

Source DB:  PubMed          Journal:  J Clin Pharm Ther        ISSN: 0269-4727            Impact factor:   2.512


  5 in total

1.  Stability of tramadol with three 5-HT3 receptor antagonists in polyolefin bags for patient-controlled delivery systems.

Authors:  Fu-Chao Chen; Jun Zhu; Bin Li; Fang-Jun Yuan; Lin-Hai Wang
Journal:  Drug Des Devel Ther       Date:  2016-06-03       Impact factor: 4.162

2.  Simultaneous Determination of Dexamethasone, Ondansetron, Granisetron, Tropisetron, and Azasetron in Infusion Samples by HPLC with DAD Detection.

Authors:  Fu-Chao Chen; Lin-Hai Wang; Jun Guo; Xiao-Ya Shi; Bao-Xia Fang
Journal:  J Anal Methods Chem       Date:  2017-01-11       Impact factor: 2.193

3.  Stability of azasetron-dexamethasone mixture for chemotherapy-induced nausea and vomiting administration.

Authors:  Bao-Xia Fang; Fu-Chao Chen; Dan Zhu; Jun Guo; Lin-Hai Wang
Journal:  Oncotarget       Date:  2017-10-31

Review 4.  The current evidence base for the feasibility of 48-hour continuous subcutaneous infusions (CSCIs): A systematically-structured review.

Authors:  James Baker; Andrew Dickman; Stephen Mason; John Ellershaw
Journal:  PLoS One       Date:  2018-03-14       Impact factor: 3.240

5.  Long-Term Stability of Tramadol and Ketamine Solutions for Patient-Controlled Analgesia Delivery.

Authors:  Junfeng Gu; Wengang Qin; Fuchao Chen; Zhongyuan Xia
Journal:  Med Sci Monit       Date:  2015-08-26
  5 in total

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