| Literature DB >> 17869509 |
Michael F Parker1, Joanne J Bronson, Donna M Barten, Jason A Corsa, Wengsheng Du, Kevin M Felsenstein, Valerie L Guss, Darcy Izzarelli, Alice Loo, Kate E McElhone, Larry R Marcin, Ramesh Padmanabha, Roger Pak, Craig T Polson, Jeremy H Toyn, Sam Varma, Jian Wang, Victoria Wong, Ming Zheng, Susan B Roberts.
Abstract
A series of amino-caprolactam sulfonamides were developed from a screening hit. Compounds with good in vitro and in vivo gamma-secretase activity are reported.Entities:
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Year: 2007 PMID: 17869509 DOI: 10.1016/j.bmcl.2007.08.047
Source DB: PubMed Journal: Bioorg Med Chem Lett ISSN: 0960-894X Impact factor: 2.823