Literature DB >> 17695515

Antitumor activity of capecitabine and bevacizumab combination in a human estrogen receptor-negative breast adenocarcinoma xenograft model.

Brian Higgins1, Kenneth Kolinsky, Michael Linn, Violeta Adames, Yu-E Zhang, Carlos Moisa, Ute Dugan, David Heimbrook, Kathryn Packman.   

Abstract

BACKGROUND: Capecitabine and bevacizumab have each been shown to inhibit tumor growth. Their combination failed to improve survival in a phase III trial of metastatic breast cancer (MBC), although it should be noted patients had been heavily pretreated with anthracyclines and taxanes. Our aim was to evaluate whether combination treatment would increase tumor growth inhibition and survival in a breast cancer model.
MATERIALS AND METHODS: Mice bearing KPL-4 human estrogen receptor-negative breast adenocarcinoma xenografts were given capecitabine orally daily for 14 days at the maximum tolerated dose (MTD) or half MTD, alone or with 5 mg/kg intraperitoneal bevacizumab twice weekly.
RESULTS: Tumor growth inhibition (TGI) and increased life span (ILS) were superior in the combination groups versus monotherapy (p < 0.05). TGI and ILS were significantly improved in the high- versus low-dose capecitabine combination (p < 0.05).
CONCLUSION: Capecitabine in combination with bevacizumab provides a basis for pursuing the combination for first-line treatment of MBC.

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Year:  2007        PMID: 17695515

Source DB:  PubMed          Journal:  Anticancer Res        ISSN: 0250-7005            Impact factor:   2.480


  11 in total

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Journal:  Cell Mol Immunol       Date:  2014-03-10       Impact factor: 11.530

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Review 3.  Capecitabine monotherapy: review of studies in first-line HER-2-negative metastatic breast cancer.

Authors:  Joyce A O'Shaughnessy; Manfred Kaufmann; Friederike Siedentopf; Philippe Dalivoust; Marc Debled; Nicholas J Robert; Nadia Harbeck
Journal:  Oncologist       Date:  2012-03-14

4.  Optimizing chemotherapy dose and schedule by Norton-Simon mathematical modeling.

Authors:  Tiffany A Traina; Ute Dugan; Brian Higgins; Kenneth Kolinsky; Maria Theodoulou; Clifford A Hudis; Larry Norton
Journal:  Breast Dis       Date:  2010

5.  Activity of the kinesin spindle protein inhibitor ispinesib (SB-715992) in models of breast cancer.

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Journal:  Clin Cancer Res       Date:  2010-01-12       Impact factor: 12.531

6.  Preclinical validation of the small molecule drug quininib as a novel therapeutic for colorectal cancer.

Authors:  Adrian G Murphy; Rory Casey; Aoife Maguire; Miriam Tosetto; Clare T Butler; Emer Conroy; Alison L Reynolds; Kieran Sheahan; Diarmuid O'Donoghue; William M Gallagher; David Fennelly; Breandán N Kennedy; Jacintha O'Sullivan
Journal:  Sci Rep       Date:  2016-10-14       Impact factor: 4.379

7.  Bevacizumab in the treatment of HER2-negative breast cancer.

Authors:  Vito Lorusso
Journal:  Biologics       Date:  2008-12

8.  Preclinical profile of a potent gamma-secretase inhibitor targeting notch signaling with in vivo efficacy and pharmacodynamic properties.

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Journal:  Cancer Res       Date:  2009-09-22       Impact factor: 12.701

9.  Anti-tumor effect of bevacizumab on a xenograft model of feline mammary carcinoma.

Authors:  Masaki Michishita; Aya Ohtsuka; Rei Nakahira; Tsuyoshi Tajima; Takayuki Nakagawa; Nobuo Sasaki; Toshiro Arai; Kimimasa Takahashi
Journal:  J Vet Med Sci       Date:  2015-11-28       Impact factor: 1.267

10.  Numerical simulation of vascular tumour growth under antiangiogenic treatment: addressing the paradigm of single-agent bevacizumab therapy with the use of experimental data.

Authors:  Katerina D Argyri; Dimitra D Dionysiou; Fay D Misichroni; Georgios S Stamatakos
Journal:  Biol Direct       Date:  2016-03-22       Impact factor: 4.540

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