Literature DB >> 17609247

A novel estrogen-free oral contraceptive pill for women: multicentre, double-blind, randomized controlled trial of mifepristone and progestogen-only pill (levonorgestrel).

F Lakha1, P C Ho, Z M Van der Spuy, K Dada, R Elton, A F Glasier, H O D Critchley, A R W Williams, D T Baird.   

Abstract

BACKGROUND: The acceptability and continuation rate of oral contraceptive steroids are limited by unpredictable bleeding and the fear of long-term risks such as breast cancer. By inhibiting ovulation and by altering the receptivity of the endometrium, antagonists of progesterone, such as mifepristone, could be developed as estrogen-free novel contraceptives.
METHODS: Multicentre, double-blind, randomized controlled trial comparing frequency of amenorrhoea (primary outcome), bleeding patterns, side effects and efficacy in women taking daily 5 mg mifepristone (n = 73) or 0.03 mg levonorgestrel (progestogen-only pill; POP, n = 23) for 24 weeks.
RESULTS: More women were amenorrhoeic while taking mifepristone than POP (49 versus 0% P < 0.001), and fewer women bled or spotted for >5 days per month (4 versus 39% P < 0.001). Forty-eight percent of women who took mifepristone for 6 months had cystic glandular dilatation of the endometrium but none showed hyperplasia or atypia. There were no pregnancies in 356 months of exposure in women who used only mifepristone for contraception. Two pregnancies occurred in women taking mifepristone who were also using condoms for dual protection.
CONCLUSIONS: Daily mifepristone (5 mg) is an effective oral contraceptive pill which has a better pattern of menstrual bleeding than an existing POP (levonorgestrel).

Entities:  

Mesh:

Substances:

Year:  2007        PMID: 17609247     DOI: 10.1093/humrep/dem177

Source DB:  PubMed          Journal:  Hum Reprod        ISSN: 0268-1161            Impact factor:   6.918


  7 in total

Review 1.  Role of nuclear progesterone receptor isoforms in uterine pathophysiology.

Authors:  Bansari Patel; Sonia Elguero; Suruchi Thakore; Wissam Dahoud; Mohamed Bedaiwy; Sam Mesiano
Journal:  Hum Reprod Update       Date:  2014-11-18       Impact factor: 15.610

2.  Distinguishing features of endometrial pathology after exposure to the progesterone receptor modulator mifepristone.

Authors:  Julietta Fiscella; Thomas Bonfiglio; Paul Winters; Steven H Eisinger; Kevin Fiscella
Journal:  Hum Pathol       Date:  2011-02-11       Impact factor: 3.466

3.  Effects of a novel estrogen-free, progesterone receptor modulator contraceptive vaginal ring on inhibition of ovulation, bleeding patterns and endometrium in normal women.

Authors:  Vivian Brache; Regine Sitruk-Ware; Alistair Williams; Diana Blithe; Horacio Croxatto; Narender Kumar; Sushma Kumar; Yun-Yen Tsong; Irving Sivin; Anita Nath; Heather Sussman; Leila Cochon; Maria Jose Miranda; Verónica Reyes; Anibal Faundes; Daniel Mishell
Journal:  Contraception       Date:  2011-12-15       Impact factor: 3.375

4.  The progesterone-receptor modulator, ulipristal acetate, drastically lowers breast cell proliferation.

Authors:  Carolyn L Westhoff; Hua Guo; Zhong Wang; Hanina Hibshoosh; Margaret Polaneczky; Malcolm C Pike; Richard Ha
Journal:  Breast Cancer Res Treat       Date:  2022-01-11       Impact factor: 4.624

Review 5.  Vaginal ring delivery of selective progesterone receptor modulators for contraception.

Authors:  Jeffrey T Jensen
Journal:  Contraception       Date:  2012-10-04       Impact factor: 3.375

Review 6.  Menstruation: science and society.

Authors:  Hilary O D Critchley; Elnur Babayev; Serdar E Bulun; Sandy Clark; Iolanda Garcia-Grau; Peter K Gregersen; Aoife Kilcoyne; Ji-Yong Julie Kim; Missy Lavender; Erica E Marsh; Kristen A Matteson; Jacqueline A Maybin; Christine N Metz; Inmaculada Moreno; Kami Silk; Marni Sommer; Carlos Simon; Ridhi Tariyal; Hugh S Taylor; Günter P Wagner; Linda G Griffith
Journal:  Am J Obstet Gynecol       Date:  2020-07-21       Impact factor: 10.693

Review 7.  90 YEARS OF PROGESTERONE: Selective progesterone receptor modulators in gynaecological therapies.

Authors:  H O D Critchley; R R Chodankar
Journal:  J Mol Endocrinol       Date:  2020-07       Impact factor: 5.098

  7 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.