Literature DB >> 17482813

ERbeta ligands. Part 6: 6H-Chromeno[4,3-b]quinolines as a new series of estrogen receptor beta-selective ligands.

An T Vu1, Alison N Campbell, Heather A Harris, Rayomand J Unwalla, Eric S Manas, Richard E Mewshaw.   

Abstract

A new class of estrogen receptor beta (ERbeta) ligands based on the 6H-chromeno[4,3-b]quinoline scaffold has been prepared. Several C7-substituted analogues displayed high affinity and modest selectivity for ERbeta.

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Year:  2007        PMID： 17482813     DOI： 10.1016/j.bmcl.2007.04.068

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  8 in total

1.  Analogs of N'-hydroxy-N-(4H,5H-naphtho[1,2-d]thiazol-2-yl)methanimidamide inhibit Mycobacterium tuberculosis methionine aminopeptidases.

Authors:  Shridhar Bhat; Omonike Olaleye; Kirsten J Meyer; Wanliang Shi; Ying Zhang; Jun O Liu
Journal:  Bioorg Med Chem       Date:  2012-05-17       Impact factor: 3.641

2.  Bibenzyl- and stilbene-core compounds with non-polar linker atom substituents as selective ligands for estrogen receptor beta.

Authors:  Michael Waibel; Meri De Angelis; Fabio Stossi; Karen J Kieser; Kathryn E Carlson; Benita S Katzenellenbogen; John A Katzenellenbogen
Journal:  Eur J Med Chem       Date:  2009-02-20       Impact factor: 6.514

3.  A one-pot three-component reaction involving 2-aminochromone in aqueous micellar medium: a green synthesis of hexahydrochromeno[2,3-b]quinolinedione.

Authors:  Jaydip Ghosh; Pritam Biswas; Michael G B Drew; Chandrakanta Bandyopadhyay
Journal:  Mol Divers       Date:  2015-03-11       Impact factor: 2.943

4.  Synthesis of chromeno[3,4-B]quinoline derivatives by heterogeneous [Cu(II)BHPPDAH] catalyst without being immobilized on any support under mild conditions using PEG 300 as green solvent.

Authors:  Hashem Sharghi; Reza Khalifeh; Zahra Rashidi
Journal:  Mol Divers       Date:  2013-08-22       Impact factor: 2.943

5.  Green Protocol for the Novel Synthesis of Thiochromeno[4,3-b]pyridine and Chromeno[4,3-b]pyridine Derivatives Utilizing a High-Pressure System.

Authors:  Haider Behbehani; Kamal M Dawood; Fatemah A Aryan; Hamada Mohamed Ibrahim
Journal:  ACS Omega       Date:  2021-11-30

6.  One-pot three-component tandem annulation of 4-hydroxycoumarine with aldehyde and aromatic amines using graphene oxide as an efficient catalyst.

Authors:  Rabindranath Singha; Aminul Islam; Pranab Ghosh
Journal:  Sci Rep       Date:  2021-10-06       Impact factor: 4.379

Review 7.  Advancements in the synthesis of fused tetracyclic quinoline derivatives.

Authors:  Ramadan A Mekheimer; Mariam A Al-Sheikh; Hanadi Y Medrasi; Kamal U Sadek
Journal:  RSC Adv       Date:  2020-05-27       Impact factor: 4.036

8.  Intramolecular Povarov Reactions for the Synthesis of Chromenopyridine Fused 2-Pyridone Polyheterocycles Binding to α-Synuclein and Amyloid-β Fibrils.

Authors:  Dan E Adolfsson; Mohit Tyagi; Pardeep Singh; Adrian Deuschmann; Jörgen Ådén; Anna L Gharibyan; Sanduni Wasana Jayaweera; Anders E G Lindgren; Anders Olofsson; Fredrik Almqvist
Journal:  J Org Chem       Date:  2020-10-25       Impact factor: 4.354
  8 in total

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