Literature DB >> 17403429

GPR30: a novel indicator of poor survival for endometrial carcinoma.

Harriet O Smith1, Kimberly K Leslie, Meenakshi Singh, Clifford R Qualls, Chetana M Revankar, Nancy E Joste, Eric R Prossnitz.   

Abstract

OBJECTIVE: This study was undertaken to evaluate the relationship between GPR30, classical steroidal receptor expression, and clinical outcome in patients with endometrial carcinoma. STUDY
DESIGN: Immunohistochemistry was used to investigate the expression of GPR30, estrogen, progesterone, epidermal growth factor receptors and Ki-67 in 47 consecutive consenting patients with endometrial carcinoma diagnosed between 1997 and 2001. Results were correlated with clinical and pathologic predictors of adverse outcome and survival.
RESULTS: GPR30 correlated positively with epidermal growth factor receptor (P = .005), but negatively with progesterone (P = .05) receptor expression. GPR30 overexpression occurred more frequently in tumors with deep myometrial invasion, high-grade, biologically aggressive histologic subtypes, and advanced stage. In patients with GPR30 overexpression, survival was significantly poorer (65.2% vs 100%, P = .005).
CONCLUSION: GPR30 represents an alternative estrogen-responsive receptor that is overexpressed in tumors where estrogen and progesterone receptors are downregulated, and in high-risk endometrial cancer patients with lower survival rates.

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Year:  2007        PMID: 17403429     DOI: 10.1016/j.ajog.2007.01.004

Source DB:  PubMed          Journal:  Am J Obstet Gynecol        ISSN: 0002-9378            Impact factor:   8.661


  109 in total

Review 1.  G protein-coupled receptors: novel targets for drug discovery in cancer.

Authors:  Rosamaria Lappano; Marcello Maggiolini
Journal:  Nat Rev Drug Discov       Date:  2011-01       Impact factor: 84.694

2.  Estrogenic transmembrane receptor of GPR30 mediates invasion and carcinogenesis by endometrial cancer cell line RL95-2.

Authors:  Yin-Yan He; Gui-Qiang Du; Bin Cai; Qin Yan; Long Zhou; Xiao-Yue Chen; Wen Lu; Yi-Xia Yang; Xiao-Ping Wan
Journal:  J Cancer Res Clin Oncol       Date:  2012-01-24       Impact factor: 4.553

Review 3.  Temporal and concentration-dependent effects of oestradiol on neural pathways mediating sexual receptivity.

Authors:  P Micevych; K Sinchak
Journal:  J Neuroendocrinol       Date:  2013-11       Impact factor: 3.627

4.  Female Sex Hormone Receptor Profiling in Uterine Adenosarcomas.

Authors:  Jenna Z Marcus; Merieme Klobocista; Rouzan G Karabakhtsian; Eric Prossnitz; Gary L Goldberg; Gloria S Huang
Journal:  Int J Gynecol Cancer       Date:  2018-03       Impact factor: 3.437

5.  The novel estrogen receptor GPER regulates the migration and invasion of ovarian cancer cells.

Authors:  Yan Yan; Huidi Liu; Haixia Wen; Xueli Jiang; Xuefeng Cao; Guangmei Zhang; Guoyi Liu
Journal:  Mol Cell Biochem       Date:  2013-04-12       Impact factor: 3.396

6.  GPR30 and estrogen receptor expression: new insights into hormone dependence of inflammatory breast cancer.

Authors:  Hugo Arias-Pulido; Melanie Royce; Yun Gong; Nancy Joste; Lesley Lomo; Sang-Joon Lee; Nabila Chaher; Claire Verschraegen; Juanita Lara; Eric R Prossnitz; Massimo Cristofanilli
Journal:  Breast Cancer Res Treat       Date:  2009-11-10       Impact factor: 4.872

7.  The G protein-coupled receptor GPR30 inhibits proliferation of estrogen receptor-positive breast cancer cells.

Authors:  Eric A Ariazi; Eugen Brailoiu; Smitha Yerrum; Heather A Shupp; Michael J Slifker; Heather E Cunliffe; Michael A Black; Anne L Donato; Jeffrey B Arterburn; Tudor I Oprea; Eric R Prossnitz; Nae J Dun; V Craig Jordan
Journal:  Cancer Res       Date:  2010-01-19       Impact factor: 12.701

Review 8.  Signaling, physiological functions and clinical relevance of the G protein-coupled estrogen receptor GPER.

Authors:  Eric R Prossnitz; Matthias Barton
Journal:  Prostaglandins Other Lipid Mediat       Date:  2009-05-13       Impact factor: 3.072

9.  Role of GPER1, EGFR and CXCR1 in differentiating between malignant follicular thyroid carcinoma and benign follicular thyroid adenoma.

Authors:  Le Zhao; Xiao-Yun Zhu; Rong Jiang; Man Xu; Ni Wang; George G Chen; Zhi-Min Liu
Journal:  Int J Clin Exp Pathol       Date:  2015-09-01

Review 10.  Macromolecular Modelling and Docking Simulations for the Discovery of Selective GPER Ligands.

Authors:  Camillo Rosano; Marco Ponassi; Maria Francesca Santolla; Assunta Pisano; Lamberto Felli; Adele Vivacqua; Marcello Maggiolini; Rosamaria Lappano
Journal:  AAPS J       Date:  2015-11-16       Impact factor: 4.009

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