Literature DB >> 17311506

Novel molecular defect in the platelet ADP receptor P2Y12 of a patient with haemorrhagic diathesis.

Jasper A Remijn1, Martin J W IJsseldijk, Annuska L M Strunk, Andre P Abbes, Henk Engel, Bert Dikkeschei, Ellen C Dompeling, Philip G de Groot, Robbert J Slingerland.   

Abstract

BACKGROUND: The platelet adenosine 5'-diphosphate (ADP) receptor P2Y(12) plays a crucial role in haemostasis. Only a few patients with haemorrhagic diathesis due to molecular defects in the P2Y(12) receptor have been described so far. We report a novel molecular defect in the gene coding for P2Y(12) in a patient with a history of epistaxis, easy bruising and excessive posttraumatic blood loss.
METHODS: Platelet aggregation studies, perfusion studies, in which patient blood was perfused over collagen surfaces at arterial shear rates, and PCR and sequencing were used.
RESULTS: Platelet aggregation studies showed impaired ADP and collagen-induced aggregation for patient G.S. Perfusion of patient blood over collagen surfaces showed small thrombi consisting of spread platelets overlayered with non-spread platelets. These thrombi were identical to control thrombi formed in the presence of a P2Y(12) antagonist. DNA analysis of the P2Y(12) gene revealed a novel heterozygous base pair C-->A substitution in exon 3, changing codon 258 from proline to threonine in the third extracellular loop of the P2Y(12) receptor.
CONCLUSIONS: We conclude that perfusion studies with patient blood are of added value in the diagnostic process, which resulted in identification of a novel molecular defect in the P2Y(12) gene of a patient with haemorrhagic diathesis.

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Year:  2007        PMID: 17311506     DOI: 10.1515/CCLM.2007.036

Source DB:  PubMed          Journal:  Clin Chem Lab Med        ISSN: 1434-6621            Impact factor:   3.694


  12 in total

Review 1.  P2Y(12) receptors in platelets and other hematopoietic and non-hematopoietic cells.

Authors:  Christian Gachet
Journal:  Purinergic Signal       Date:  2012-04-11       Impact factor: 3.765

2.  Molecular defects of the platelet P2 receptors.

Authors:  Marco Cattaneo
Journal:  Purinergic Signal       Date:  2011-01-29       Impact factor: 3.765

Review 3.  Inherited dysfunctional platelet P2Y12 receptor mutations associated with bleeding disorders.

Authors:  Anna Lecchi; Eti A Femia; Silvia Paoletta; Arnaud Dupuis; Philippe Ohlmann; Christian Gachet; Kenneth A Jacobson; Katharina Machura; Gian M Podda; Barbara Zieger; Marco Cattaneo
Journal:  Hamostaseologie       Date:  2016-08-04       Impact factor: 1.778

4.  Identification of a new dysfunctional platelet P2Y12 receptor variant associated with bleeding diathesis.

Authors:  Anna Lecchi; Cristina Razzari; Silvia Paoletta; Arnaud Dupuis; Lea Nakamura; Philippe Ohlmann; Christian Gachet; Kenneth A Jacobson; Barbara Zieger; Marco Cattaneo
Journal:  Blood       Date:  2014-11-26       Impact factor: 22.113

5.  Identification of determinants required for agonistic and inverse agonistic ligand properties at the ADP receptor P2Y12.

Authors:  Philipp Schmidt; Lars Ritscher; Elizabeth N Dong; Thomas Hermsdorf; Maxi Cöster; Doreen Wittkopf; Jens Meiler; Torsten Schöneberg
Journal:  Mol Pharmacol       Date:  2012-10-23       Impact factor: 4.436

Review 6.  Inherited platelet disorders: thrombocytopenias and thrombocytopathies.

Authors:  Giovanna D'Andrea; Massimiliano Chetta; Maurizio Margaglione
Journal:  Blood Transfus       Date:  2009-10       Impact factor: 3.443

7.  An intact PDZ motif is essential for correct P2Y12 purinoceptor traffic in human platelets.

Authors:  Shaista Nisar; Martina E Daly; Augusto B Federici; Andrea Artoni; Andrew D Mumford; Stephen P Watson; Stuart J Mundell
Journal:  Blood       Date:  2011-09-21       Impact factor: 22.113

Review 8.  Rare platelet GPCR variants: what can we learn?

Authors:  S P Nisar; M L Jones; M R Cunningham; A D Mumford; S J Mundell
Journal:  Br J Pharmacol       Date:  2014-11-24       Impact factor: 8.739

9.  Structural and functional evolution of the P2Y(12)-like receptor group.

Authors:  Torsten Schöneberg; Thomas Hermsdorf; Eva Engemaier; Kathrin Engel; Ines Liebscher; Doreen Thor; Klaas Zierau; Holger Römpler; Angela Schulz
Journal:  Purinergic Signal       Date:  2007-09-06       Impact factor: 3.765

10.  The P2Y 13 Met-158-Thr polymorphism, which is in linkage disequilibrium with the P2Y 12 locus, is not associated with acute myocardial infarction.

Authors:  Stefan Amisten; Oscar O Braun; Lovisa Johansson; Martin Ridderstråle; Olle Melander; David Erlinge
Journal:  PLoS One       Date:  2008-01-23       Impact factor: 3.240

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