Literature DB >> 17308968

Levodopa slows progression of Parkinson's disease: external validation by clinical trial simulation.

Phylinda L S Chan1, John G Nutt, Nicholas H G Holford.   

Abstract

PURPOSE: To externally validate the model predictions of a DATATOP cohort analysis through application of clinical trial simulation with the study design of the ELLDOPA trial.
METHODS: The stochastic pharmacokinetic-pharmacodynamic and disease progress model was developed from the large DATATOP cohort of patients followed for 8 years. ELLDOPA was designed to detect a difference between placebo and levodopa treated arms in the total Unified Parkinson's Disease Rating Scale (UPDRS) taken at baseline and following 2 weeks levodopa washout after 40 weeks of treatment. The total UPDRS response was simulated with different assumptions on levodopa effect (symptomatic with/without disease modifying capability) and washout speed of symptomatic effect.
RESULTS: The observed results of ELLDOPA were similar to the model predictions assuming levodopa slows disease progression and has a slow washout of symptomatic effect.
CONCLUSIONS: This simulation work confirmed the conclusion of the DATATOP analysis finding that levodopa slows disease progression. The simulation results also showed that a dose-related increased rate of progression in Parkinson's disease, obscured by symptomatic benefit, is very unlikely. Finally, the simulation results also shown that 2 weeks washout period was not adequate to completely eliminate the symptomatic benefits of levodopa.

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Year:  2007        PMID: 17308968     DOI: 10.1007/s11095-006-9202-3

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


  27 in total

1.  Chronic levodopa is not toxic for remaining dopamine neurons, but instead promotes their recovery, in rats with moderate nigrostriatal lesions.

Authors:  M G Murer; G Dziewczapolski; L B Menalled; M C García; Y Agid; O Gershanik; R Raisman-Vozari
Journal:  Ann Neurol       Date:  1998-05       Impact factor: 10.422

2.  A size standard for pharmacokinetics.

Authors:  N H Holford
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Review 3.  Understanding the dose-effect relationship: clinical application of pharmacokinetic-pharmacodynamic models.

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4.  DATATOP: a multicenter controlled clinical trial in early Parkinson's disease. Parkinson Study Group.

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Journal:  Arch Neurol       Date:  1989-10

5.  Non-linearity of Parkinson's disease progression: implications for sample size calculations in clinical trials.

Authors:  Paulo Guimaraes; Karl Kieburtz; Christopher G Goetz; Jordan J Elm; Yuko Y Palesch; Peng Huang; Bernard Ravina; Caroline M Tanner; Barbara C Tilley
Journal:  Clin Trials       Date:  2005       Impact factor: 2.486

Review 6.  Parkinson disease, the effect of levodopa, and the ELLDOPA trial. Earlier vs Later L-DOPA.

Authors:  S Fahn
Journal:  Arch Neurol       Date:  1999-05

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Authors:  S G Diamond; C H Markham; M M Hoehn; F H McDowell; M D Muenter
Journal:  Ann Neurol       Date:  1987-07       Impact factor: 10.422

8.  Quantitative description of loss of clinical benefit following withdrawal of levodopa-carbidopa and bromocriptine in early Parkinson's disease.

Authors:  Robert A Hauser; Nicholas H G Holford
Journal:  Mov Disord       Date:  2002-09       Impact factor: 10.338

9.  Toxic and protective effects of L-dopa on mesencephalic cell cultures.

Authors:  C Mytilineou; S K Han; G Cohen
Journal:  J Neurochem       Date:  1993-10       Impact factor: 5.372

10.  L-dopa increases nigral production of hydroxyl radicals in vivo: potential L-dopa toxicity?

Authors:  T S Smith; W D Parker; J P Bennett
Journal:  Neuroreport       Date:  1994-04-14       Impact factor: 1.837

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  17 in total

1.  Progression of motor and nonmotor features of Parkinson's disease and their response to treatment.

Authors:  Thuy C Vu; John G Nutt; Nicholas H G Holford
Journal:  Br J Clin Pharmacol       Date:  2012-08       Impact factor: 4.335

2.  Disease progression, drug action and Parkinson's disease: why time cannot be ignored.

Authors:  Nick Holford; John G Nutt
Journal:  Eur J Clin Pharmacol       Date:  2007-12-19       Impact factor: 2.953

Review 3.  Disease progression and neuroscience.

Authors:  Nick Holford
Journal:  J Pharmacokinet Pharmacodyn       Date:  2013-04-17       Impact factor: 2.745

Review 4.  Early versus delayed initiation of pharmacotherapy in Parkinson's disease.

Authors:  Matthias Löhle; Carl-Johan Ramberg; Heinz Reichmann; Anthony H V Schapira
Journal:  Drugs       Date:  2014-04       Impact factor: 9.546

Review 5.  A review of disease progression models of Parkinson's disease and applications in clinical trials.

Authors:  Charles S Venuto; Nicholas B Potter; E Ray Dorsey; Karl Kieburtz
Journal:  Mov Disord       Date:  2016-05-26       Impact factor: 10.338

Review 6.  Protection against Parkinson's disease progression: clinical experience.

Authors:  Peter A LeWitt; Danette C Taylor
Journal:  Neurotherapeutics       Date:  2008-04       Impact factor: 7.620

7.  Progression of MDS-UPDRS Scores Over Five Years in De Novo Parkinson Disease from the Parkinson's Progression Markers Initiative Cohort.

Authors:  Samantha K Holden; Taylor Finseth; Stefan H Sillau; Brian D Berman
Journal:  Mov Disord Clin Pract       Date:  2017-09-22

8.  Modeling and simulation to optimize the design and analysis of confirmatory trials, characterize risk-benefit, and support label claims.

Authors:  S F Marshall; R Hemmings; F Josephson; M O Karlsson; M Posch; J-L Steimer
Journal:  CPT Pharmacometrics Syst Pharmacol       Date:  2013-02-27

9.  Imaging mass spectrometry reveals elevated nigral levels of dynorphin neuropeptides in L-DOPA-induced dyskinesia in rat model of Parkinson's disease.

Authors:  Anna Ljungdahl; Jörg Hanrieder; Maria Fälth; Jonas Bergquist; Malin Andersson
Journal:  PLoS One       Date:  2011-09-30       Impact factor: 3.240

10.  Targeting the progression of Parkinson's disease.

Authors:  J L George; S Mok; D Moses; S Wilkins; A I Bush; R A Cherny; D I Finkelstein
Journal:  Curr Neuropharmacol       Date:  2009-03       Impact factor: 7.363

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