Literature DB >> 17253880

Safety profile of rosuvastatin: results of a prescription-event monitoring study of 11,680 patients.

Rachna Kasliwal1, Lynda V Wilton, Victoria Cornelius, Beate Aurich-Barrera, Saad A W Shakir.   

Abstract

BACKGROUND AND
OBJECTIVE: Rosuvastatin is a lipid-lowering drug, the newest of a class of drugs called HMG-CoA reductase inhibitors, or 'statins', launched in the UK in March 2003. Our objective was to monitor the post-marketing safety of this drug, prescribed in primary care in England, using prescription-event monitoring.
METHODS: An observational cohort study in which patients were identified from dispensed prescriptions issued by primary care physicians/general practitioners (GPs) between August and December 2003. Demographic and clinical-event data were collected from questionnaires posted to GPs at least 6 months after the date of first prescription for each patient. Stratified analysis of specific events by starting dose of rosuvastatin was conducted. Follow-up and causality assessment of medically significant events was undertaken.
RESULTS: The cohort comprised 11,680 patients (median age 64 years); 50.3% were males (5880 of 11,680). The median period of treatment was 9.8 months. Of these patients, 72.7% (n = 8494) were started on rosuvastatin 10 mg/day. A total of 17.5% (n = 2047) of the patients were reported to have stopped treatment with rosuvastatin. Myalgia was the most frequent reason for stopping rosuvastatin and the most frequently reported clinical event. A 2.5-fold increase in the rate of abnormal liver-function tests (LFTs) was observed for patients started on rosuvastatin 40 mg/day compared with those started on 10 mg/day (2.71; 95% CI 1.53, 4.53). No case of rhabdomyolysis was reported in this cohort.
CONCLUSION: Rosuvastatin was considered to be a reasonably well tolerated drug. In the majority of patients, rosuvastatin was prescribed in line with recommendations. Abnormality of LFTs was found to be more frequent with the 40 mg/day dosage of rosuvastatin. Results from this study should be taken into account together with those of other clinical and pharmacoepidemiological studies of rosuvastatin.

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Year:  2007        PMID: 17253880     DOI: 10.2165/00002018-200730020-00005

Source DB:  PubMed          Journal:  Drug Saf        ISSN: 0114-5916            Impact factor:   5.606


  19 in total

1.  Statins and myopathy.

Authors:  Iain P Hargreaves; Simon Heales
Journal:  Lancet       Date:  2002-02-23       Impact factor: 79.321

2.  Rosuvastatin-warfarin drug interaction.

Authors:  Michael Barry
Journal:  Lancet       Date:  2004-01-24       Impact factor: 79.321

Review 3.  High density lipoproteins (HDLs) and atherosclerosis; the unanswered questions.

Authors:  Philip Barter; John Kastelein; Alistair Nunn; Richard Hobbs
Journal:  Atherosclerosis       Date:  2003-06       Impact factor: 5.162

4.  Should rosuvastatin be withdrawn from the market?

Authors:  John J P Kastelein
Journal:  Lancet       Date:  2004 Oct 30-Nov 5       Impact factor: 79.321

Review 5.  Hydrophilicity/lipophilicity: relevance for the pharmacology and clinical effects of HMG-CoA reductase inhibitors.

Authors:  B A Hamelin; J Turgeon
Journal:  Trends Pharmacol Sci       Date:  1998-01       Impact factor: 14.819

Review 6.  HMG-CoA reductase inhibitors and myotoxicity.

Authors:  M Ucar; T Mjörndal; R Dahlqvist
Journal:  Drug Saf       Date:  2000-06       Impact factor: 5.606

Review 7.  Rosuvastatin safety: lessons from the FDA review and post-approval surveillance.

Authors:  Michael H Davidson
Journal:  Expert Opin Drug Saf       Date:  2004-11       Impact factor: 4.250

8.  Incidence of hospitalized rhabdomyolysis in patients treated with lipid-lowering drugs.

Authors:  David J Graham; Judy A Staffa; Deborah Shatin; Susan E Andrade; Stephanie D Schech; Lois La Grenade; Jerry H Gurwitz; K Arnold Chan; Michael J Goodman; Richard Platt
Journal:  JAMA       Date:  2004-11-22       Impact factor: 56.272

9.  Autoimmune hepatitis revealed by atorvastatin.

Authors:  Nicoletta Pelli; Maurizio Setti; Paola Ceppa; Carlo Toncini; Francesco Indiveri
Journal:  Eur J Gastroenterol Hepatol       Date:  2003-08       Impact factor: 2.566

10.  Safety of rosuvastatin.

Authors:  James Shepherd; Donald B Hunninghake; Evan A Stein; John J P Kastelein; Susan Harris; John Pears; Howard G Hutchinson
Journal:  Am J Cardiol       Date:  2004-10-01       Impact factor: 2.778

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  6 in total

1.  Erythromelalgia accompanying rosuvastatin-associated myopathy.

Authors:  Nevio Cimolai; Tomas Cimolai
Journal:  J Dermatol Case Rep       Date:  2009-04-05

2.  Clinical importance of the drug interaction between statins and CYP3A4 inhibitors: a retrospective cohort study in The Health Improvement Network.

Authors:  Christopher G Rowan; Steven M Brunelli; Jeffrey Munson; James Flory; Peter P Reese; Sean Hennessy; James Lewis; Daniel Mines; Jeffrey S Barrett; Warren Bilker; Brian L Strom
Journal:  Pharmacoepidemiol Drug Saf       Date:  2012-03-16       Impact factor: 2.890

3.  Statin-induced liver injury in an area endemic for hepatitis B virus infection: risk factors and outcome analysis.

Authors:  Li Yueh Wang; Yi-Shin Huang; Chin-Lin Perng; Bryan Huang; Han-Chieh Lin
Journal:  Br J Clin Pharmacol       Date:  2016-06-17       Impact factor: 4.335

4.  Long-term use of rosuvastatin: a critical risk benefit appraisal and comparison with other antihyperlipidemics.

Authors:  Leonardo Calza
Journal:  Drug Healthc Patient Saf       Date:  2009-08-28

5.  SLCO1B1 Polymorphisms and Statin-Induced Myopathy.

Authors:  Alison Stewart
Journal:  PLoS Curr       Date:  2013-12-04

6.  Statin-induced myopathy in a usual care setting-a prospective observational study of gender differences.

Authors:  Ilona Skilving; Mats Eriksson; Anders Rane; Marie-Louise Ovesjö
Journal:  Eur J Clin Pharmacol       Date:  2016-08-02       Impact factor: 2.953

  6 in total

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