Literature DB >> 17228132

Acute drug induced hepatitis due to erlotinib.

Jeyanthi Ramanarayanan1, Sarah L Scarpace.   

Abstract

CONTEXT: Acute drug induced hepatitis has not been commonly associated with epidermal growth factor receptor (EGFR) inhibitors. Hepatotoxicity seen with erlotinib, a small molecule tyrosine kinase inhibitor to EGFR, is usually transient with mild elevation of transaminases. CASE REPORT: We report a case of acute severe hepatitis resulting from erlotinib monotherapy in a patient with locally advanced pancreatic cancer. Hepatotoxicity resolved once erlotinib was discontinued and serum transaminases returned to baseline normal values.
CONCLUSIONS: Acute severe hepatitis though rare is occasionally observed with EGFR inhibitors gefitinib or erlotinib. As EGFR inhibitors are now incorporated with chemotherapy in advanced pancreatic cancers, clinicians should be aware of this potential complication.

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Year:  2007        PMID: 17228132

Source DB:  PubMed          Journal:  JOP        ISSN: 1590-8577


  7 in total

1.  The escalating role of epidermal growth factor receptor inhibitors in cancer management: clinical considerations for the health system pharmacist.

Authors:  Dwight D Kloth; Lew Iacovelli; Rebecca Arbuckle; Angela C McIntosh
Journal:  P T       Date:  2010-04

2.  Cytochrome P450-mediated bioactivation of the epidermal growth factor receptor inhibitor erlotinib to a reactive electrophile.

Authors:  Xiaohai Li; Theodore M Kamenecka; Michael D Cameron
Journal:  Drug Metab Dispos       Date:  2010-04-09       Impact factor: 3.922

Review 3.  Metabolism considerations for kinase inhibitors in cancer treatment.

Authors:  Derek R Duckett; Michael D Cameron
Journal:  Expert Opin Drug Metab Toxicol       Date:  2010-10       Impact factor: 4.481

4.  Reactivation of hepatitis B virus after withdrawal of erlotinib.

Authors:  N Bui; I Wong-Sefidan
Journal:  Curr Oncol       Date:  2015-12       Impact factor: 3.677

5.  Autoimmune-like hepatitis during masitinib therapy in an amyotrophic lateral sclerosis patient.

Authors:  Maria Salvado; Victor Vargas; Marta Vidal; Macarena Simon-Talero; Jessica Camacho; Josep Gamez
Journal:  World J Gastroenterol       Date:  2015-09-28       Impact factor: 5.742

6.  Acute Fatal Liver Toxicity under Erlotinib.

Authors:  Sabina Schacher-Kaufmann; Miklos Pless
Journal:  Case Rep Oncol       Date:  2010-06-08

7.  Disposition of Erlotinib and Its Metabolite OSI420 in a Patient with High Bilirubin Levels.

Authors:  M Czejka; A Sahmanovic; P Buchner; T Steininger; C Dittrich
Journal:  Case Rep Oncol       Date:  2013-12-12
  7 in total

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