Literature DB >> 17148967

Effects of metformin and rosiglitazone in HIV-infected patients with hyperinsulinemia and elevated waist/hip ratio.

Kathleen Mulligan1, Yang Yang, David A Wininger, Susan L Koletar, Robert A Parker, Beverly L Alston-Smith, Jeffrey T Schouten, Roger A Fielding, Michael T Basar, Steven Grinspoon.   

Abstract

OBJECTIVE: To evaluate the effects of metformin and rosiglitazone, alone or in combination, on fat distribution, insulin sensitivity, and lipids in HIV-infected patients with insulin resistance and changes in fat distribution.
METHODS: A total of 105 subjects were randomly assigned to receive metformin (500 mg twice a day increasing to 1000 mg twice a day after 2 weeks) with rosiglitazone placebo (Met/P, N = 26); rosiglitazone (4 mg/day) with metformin placebo (Rosi/P, N = 27); rosiglitazone (4 mg/day) plus metformin (500 mg twice a day increasing to 1000 mg twice a day after 2 weeks; Met/Rosi, N = 25); or dual placebo (P/P, N = 27) for 16 weeks. Efficacy assessments included oral glucose tolerance testing, abdominal computed tomography, whole-body dual-energy X-ray absorptiometry, and the measurement of fasting lipids and other biochemical indices. Safety was monitored throughout. Intent-to-treat analyses were performed using non-parametric methods.
RESULTS: The median insulin area under the curve (AUC) decreased significantly compared with baseline in both groups randomly assigned to rosiglitazone (Rosi/P -25.7 microIU/ml, P = 0.012; Met/Rosi -17.7 microIU/ml, P = 0.002); and tended to decrease in the Met/P group (-11.1 microIU/ml, P = 0.058). The change in AUC with combination therapy was significant compared with placebo (P = 0.032). No treatment was associated with significant changes in visceral or subcutaneous abdominal fat. Leg fat increased in subjects on Rosi/P compared with placebo (+4.8 versus -8.3%, P = 0.034). Rosiglitazone, but not metformin, increased adiponectin but also increased LDL-cholesterol and decreased HDL-cholesterol. Gastrointestinal effects occurred frequently in subjects on metformin.
CONCLUSION: Both treatments improved insulin sensitivity, but neither reduced visceral fat. Rosiglitazone may increase subcutaneous fat in some individuals.

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Year:  2007        PMID: 17148967     DOI: 10.1097/QAD.0b013e328011220e

Source DB:  PubMed          Journal:  AIDS        ISSN: 0269-9370            Impact factor:   4.177


  27 in total

1.  Rosiglitazone improves lipoatrophy in patients receiving thymidine-sparing regimens.

Authors:  Marisa Tungsiripat; Dalia El Bejjani; Nesrine Rizk; Mary Ann O'riordan; Allison C Ross; Corrilynn Hileman; Norma Storer; Danielle Harrill; Grace A McComsey
Journal:  AIDS       Date:  2010-06-01       Impact factor: 4.177

Review 2.  Management of the metabolic effects of HIV and HIV drugs.

Authors:  Todd T Brown; Marshall J Glesby
Journal:  Nat Rev Endocrinol       Date:  2011-09-20       Impact factor: 43.330

3.  Pioglitazone therapy for HIV/HAART-associated lipodystrophy syndrome could increase subcutaneous fat mass in non-lipoatrophic but not in lipoatrophic regions.

Authors:  Sadanori Okada; Mitsuru Konishi; Hitoshi Ishii
Journal:  BMJ Case Rep       Date:  2016-02-25

4.  Designer adiponectin receptor agonist stabilizes metabolic function and prevents brain injury caused by HIV protease inhibitors.

Authors:  Jennifer K Pepping; Laszlo Otvos; Eva Surmacz; Sunita Gupta; Jeffrey N Keller; Annadora J Bruce-Keller
Journal:  J Neuroimmune Pharmacol       Date:  2014-02-23       Impact factor: 4.147

Review 5.  Pathogenesis and treatment of HIV lipohypertrophy.

Authors:  Vivien L Leung; Marshall J Glesby
Journal:  Curr Opin Infect Dis       Date:  2011-02       Impact factor: 4.915

6.  The effects of recombinant human leptin on visceral fat, dyslipidemia, and insulin resistance in patients with human immunodeficiency virus-associated lipoatrophy and hypoleptinemia.

Authors:  Kathleen Mulligan; Hootan Khatami; Jean-Marc Schwarz; Giorgos K Sakkas; Alex M DePaoli; Viva W Tai; Michael J Wen; Grace A Lee; Carl Grunfeld; Morris Schambelan
Journal:  J Clin Endocrinol Metab       Date:  2009-01-27       Impact factor: 5.958

7.  Changes in Inflammation, Oxidative Stress, Mitochondrial DNA Content after Rosiglitazone in HIV Lipoatrophy.

Authors:  Marisa Tungsiripat; Dalia El-Bejjani; Nesrine Rizk; Bo Hu; Allison C Ross; Ulrich A Walker; Dirk Lebrecht; Ginger Milne; Norma Storer; Grace A McComsey
Journal:  J AIDS Clin Res       Date:  2012-10-15

8.  The efficacy and safety of insulin-sensitizing drugs in HIV-associated lipodystrophy syndrome: a meta-analysis of randomized trials.

Authors:  Siddharth H Sheth; Robin J Larson
Journal:  BMC Infect Dis       Date:  2010-06-23       Impact factor: 3.090

9.  Rosiglitazone increases small dense low-density lipoprotein concentration and decreases high-density lipoprotein particle size in HIV-infected patients.

Authors:  Colleen Hadigan; Sasha Mazza; Dana Crum; Steven Grinspoon
Journal:  AIDS       Date:  2007-11-30       Impact factor: 4.177

Review 10.  Approach to the human immunodeficiency virus-infected patient with lipodystrophy.

Authors:  Todd T Brown
Journal:  J Clin Endocrinol Metab       Date:  2008-08       Impact factor: 5.958

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