Literature DB >> 17027257

A feasibility study of the efficacy and tolerability of the combination of Exemestane with the COX-2 inhibitor Celecoxib in post-menopausal patients with advanced breast cancer.

P A Canney1, M A Machin, J Curto.   

Abstract

BACKGROUND: This was a feasibility study of the combination of Exemestane and the cyclooxygenase-2 (COX-2) inhibitor Celecoxib in advanced breast cancer. PATIENTS AND METHODS: Post-menopausal women with histologically proven, hormone receptor positive, advanced breast cancer who had progressive disease, normal blood counts, liver and renal function were eligible. Exemestane was given at a dose of 25 mg daily and Celecoxib at a dose of 400 mg bd. Responses were assessed according to RECIST criteria and toxicity was accessed according to CTC. The primary end-point was the percentage of patients who had neither discontinued therapy nor progressed at 6 months ('treatment successes').
RESULTS: Fifty-three eligible patients were enrolled. Of 30 patients with target lesions, 4 (13%) had a complete response (CR), 12 (40%) a partial response (PR) and 5 (17%) stable disease (SD). The best response in 18 of the 23 patients with no target lesions at baseline was stable disease. The clinical benefit (CR, PR+SD) for the whole group was therefore 39/53 (74%). The 'treatment success' rate was 60%. There were two non-malignant deaths which may have been associated with treatment.
CONCLUSION: The combination of Exemestane and Celecoxib shows promising activity and tolerability and these results support the use of this combination in phase III clinical trials of short duration treatments.

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Year:  2006        PMID: 17027257     DOI: 10.1016/j.ejca.2006.08.014

Source DB:  PubMed          Journal:  Eur J Cancer        ISSN: 0959-8049            Impact factor:   9.162


  10 in total

1.  Phase II trial of neoadjuvant exemestane in combination with celecoxib in postmenopausal women who have breast cancer.

Authors:  Maryam B Lustberg; Stephen P Povoski; Weiqiang Zhao; Rebecca M Ziegler; Yasuro Sugimoto; Amy S Ruppert; Amy M Lehman; Donna R Shiels; Ewa Mrozek; Bhuvaneswari Ramaswamy; Rachel M Layman; Robert W Brueggemeier; Charles L Shapiro
Journal:  Clin Breast Cancer       Date:  2011-05-19       Impact factor: 3.225

2.  Synergistic effect between celecoxib and luteolin is dependent on estrogen receptor in human breast cancer cells.

Authors:  Ye Won Jeon; Young Ee Ahn; Won Sang Chung; Hyun Joo Choi; Young Jin Suh
Journal:  Tumour Biol       Date:  2015-04-08

3.  Aspirin potentiates celecoxib-induced growth inhibition and apoptosis in human non-small cell lung cancer by targeting GRP78 activity.

Authors:  Xiangyu Zhang; Jia Chen; Cheng Cheng; Ping Li; Fangfang Cai; Huangru Xu; Yanyan Lu; Nini Cao; Jia Liu; Jigang Wang; Zi-Chun Hua; Hongqin Zhuang
Journal:  Ther Adv Med Oncol       Date:  2020-09-17       Impact factor: 8.168

4.  COX2 expression in high-grade breast cancer: evidence for prognostic significance in the subset of triple-negative breast cancer patients.

Authors:  Bar Chikman; Sergey Vasyanovich; Ron Lavy; Liliana Habler; Gleb Tolstov; Andronik Kapiev; Ariel Halevy; Judith Sandbank
Journal:  Med Oncol       Date:  2014-05-10       Impact factor: 3.064

5.  Aldo-keto reductase 1C3 expression in MCF-7 cells reveals roles in steroid hormone and prostaglandin metabolism that may explain its over-expression in breast cancer.

Authors:  Michael C Byrns; Ling Duan; Seon Hwa Lee; Ian A Blair; Trevor M Penning
Journal:  J Steroid Biochem Mol Biol       Date:  2009-12-28       Impact factor: 4.292

6.  COX-2 activation is associated with Akt phosphorylation and poor survival in ER-negative, HER2-positive breast cancer.

Authors:  Sharon A Glynn; Robyn L Prueitt; Lisa A Ridnour; Brenda J Boersma; Tiffany M Dorsey; David A Wink; Julie E Goodman; Harris G Yfantis; Dong H Lee; Stefan Ambs
Journal:  BMC Cancer       Date:  2010-11-15       Impact factor: 4.430

7.  Effects of celecoxib and ly117018 combination on human breast cancer cells in vitro.

Authors:  Klaus H Baumann; Elmar Klusmeier; Isabel Eggemann; Silke Reinartz; Achim Almeroth; Mathias Kalder; Uwe Wagner
Journal:  Breast Cancer (Auckl)       Date:  2009-04-07

8.  Celecoxib and acetylbritannilactone interact synergistically to suppress breast cancer cell growth via COX-2-dependent and -independent mechanisms.

Authors:  B Liu; J K Wen; B H Li; X M Fang; J J Wang; Y P Zhang; C J Shi; D Q Zhang; M Han
Journal:  Cell Death Dis       Date:  2011-07-28       Impact factor: 8.469

Review 9.  Celecoxib in breast cancer prevention and therapy.

Authors:  Jieqing Li; Qiongyu Hao; Wei Cao; Jaydutt V Vadgama; Yong Wu
Journal:  Cancer Manag Res       Date:  2018-10-26       Impact factor: 3.989

10.  Curcumol potentiates celecoxib-induced growth inhibition and apoptosis in human non-small cell lung cancer.

Authors:  Fangfang Cai; Minghui Chen; Daolong Zha; Peng Zhang; Xiangyu Zhang; Nini Cao; Jishuang Wang; Yan He; Xinxin Fan; Wenjing Zhang; Zhongping Fu; Yueyang Lai; Zi-Chun Hua; Hongqin Zhuang
Journal:  Oncotarget       Date:  2017-12-14
  10 in total

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