Literature DB >> 16986202

2-Anilinobenzamides as SIRT inhibitors.

Takayoshi Suzuki1, Keiko Imai, Hidehiko Nakagawa, Naoki Miyata.   

Abstract

Entities:  

Mesh:

Substances:

Year:  2006        PMID: 16986202     DOI: 10.1002/cmdc.200600162

Source DB:  PubMed          Journal:  ChemMedChem        ISSN: 1860-7179            Impact factor:   3.466


× No keyword cloud information.
  6 in total

Review 1.  Nicotinamide is an inhibitor of SIRT1 in vitro, but can be a stimulator in cells.

Authors:  Eun Seong Hwang; Seon Beom Song
Journal:  Cell Mol Life Sci       Date:  2017-04-17       Impact factor: 9.261

Review 2.  Rejuvenating sirtuins: the rise of a new family of cancer drug targets.

Authors:  Santina Bruzzone; Marco Daniele Parenti; Alessia Grozio; Alberto Ballestrero; Inga Bauer; Alberto Del Rio; Alessio Nencioni
Journal:  Curr Pharm Des       Date:  2013       Impact factor: 3.116

3.  Identification of a novel polyprenylated acylphloroglucinol‑derived SIRT1 inhibitor with cancer‑specific anti-proliferative and invasion-suppressing activities.

Authors:  Lijia Zhu; Ji Qi; Christine Ya-Chi Chiao; Qiang Zhang; John A Porco; Douglas V Faller; Yan Dai
Journal:  Int J Oncol       Date:  2014-09-03       Impact factor: 5.650

4.  The Discovery of Novel 10,11-Dihydro-5H-dibenz[b,f]azepine SIRT2 Inhibitors.

Authors:  Paolo Di Fruscia; Ka-Kei Ho; Sasiwan Laohasinnarong; Mattaka Khongkow; Sebastian H B Kroll; Suhail A Islam; Michael J E Sternberg; Karin Schmidtkunz; Manfred Jung; Eric W-F Lam; Matthew J Fuchter
Journal:  Medchemcomm       Date:  2012-03-01       Impact factor: 3.597

5.  Ligand-based virtual screening and inductive learning for identification of SIRT1 inhibitors in natural products.

Authors:  Yunan Sun; Hui Zhou; Hongmei Zhu; Siu-wai Leung
Journal:  Sci Rep       Date:  2016-01-25       Impact factor: 4.379

6.  Potent mechanism-based sirtuin-2-selective inhibition by an in situ-generated occupant of the substrate-binding site, "selectivity pocket" and NAD+-binding site.

Authors:  Paolo Mellini; Yukihiro Itoh; Hiroki Tsumoto; Ying Li; Miki Suzuki; Natsuko Tokuda; Taeko Kakizawa; Yuri Miura; Jun Takeuchi; Maija Lahtela-Kakkonen; Takayoshi Suzuki
Journal:  Chem Sci       Date:  2017-07-21       Impact factor: 9.825

  6 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.