P Ward1, G B Ewan, C C Jordan, S J Ireland, R M Hagan, J R Brown. Show Affiliations » 1. Department of Medicinal Chemistry, Glaxo Group Research Ltd., Greenford, Middlesex, U.K.
Abstract
Mesh: See more » Amino Acid SequenceAnimalsGuinea PigsIn Vitro TechniquesIntestinal Mucosa/metabolismIntestines/drug effectsIntestines/physiologyMolecular Sequence DataMolecular StructureMuscle Contraction/drug effectsMuscle, Smooth/drug effectsMuscle, Smooth/metabolismMuscle, Smooth/physiologyNeurokinin A/analogs & derivativesNeurokinin A/antagonists & inhibitorsNeurokinin A/chemical synthesisNeurokinin A/pharmacologyNeurokinin B/analogs & derivativesNeurokinin B/antagonists & inhibitorsNeurokinin B/chemical synthesisNeurokinin B/pharmacologyProtein ConformationRatsReceptors, Neurokinin-1Receptors, Neurokinin-2Receptors, Neurokinin-3Receptors, Neurotransmitter/drug effectsReceptors, Neurotransmitter/metabolismStructure-Activity RelationshipSubstance P/analogs & derivativesSubstance P/antagonists & inhibitorsSubstance P/chemical synthesisSubstance P/pharmacology
Substances: See more » Receptors, Neurokinin-1Receptors, Neurokinin-2Receptors, Neurokinin-3Receptors, NeurotransmitterSubstance PNeurokinin ANeurokinin B
Year: 1990 PMID: 1694545 DOI: 10.1021/jm00169a003
Source DB: PubMed Journal: J Med Chem ISSN: 0022-2623 Impact factor: 7.446