Literature DB >> 16899619

Valproic Acid prolongs survival time of severe combined immunodeficient mice bearing intracerebellar orthotopic medulloblastoma xenografts.

Qin Shu1, Barbara Antalffy, Jack Meng Feng Su, Adekunle Adesina, Ching-Nan Ou, Torsten Pietsch, Susan M Blaney, Ching C Lau, Xiao-Nan Li.   

Abstract

PURPOSE: To develop novel orthotopic xenograft models of medulloblastoma in severe combined immunodeficient mice and to evaluate the in vivo antitumor efficacy of valproic acid. EXPERIMENTAL
DESIGN: Orthotopic xenografts were developed by injecting 10(3) to 10(5) tumor cells from four medulloblastoma cell lines (D283-MED, DAOY, MHH-MED-1, and MEB-MED-8A) into the right cerebellum of severe combined immunodeficient mice. Animals were then examined for reproducibility of tumorigenicity, cell number-survival time relationship, and histopathologic features. Tumor growth was monitored in vivo by serially sectioning the xenograft brains at 2, 4, 6, and 8 weeks postinjection. Valproic acid treatment, administered at 600 microg/h for 2 weeks via s.c. osmotic minipumps, was initiated 2 weeks after injection of 10(5) medulloblastoma cells, and treated and untreated animals were monitored for differences in survival. Changes in histone acetylation, proliferation, apoptosis, differentiation, and angiogenesis in xenografts were also evaluated.
RESULTS: Tumorigenicity was maintained at 100% in D283-MED, DAOY, and MHH-MED-1 cell lines. These cerebellar xenografts displayed histologic features and immunohistochemical profiles (microtubule-associated protein 2, glial fibrillary acidic protein, and vimentin) similar to human medulloblastomas. Animal survival time was inversely correlated with injected tumor cell number. Treatment with valproic acid prolonged survival time in two (D283-MED and MHH-MED-1) of the three models and was associated with induction of histone hyperacetylation, inhibition of proliferation and angiogenesis, and enhancement of apoptosis and differentiation.
CONCLUSION: We have developed intracerebellar orthotopic models that closely recapitulated the biological features of human medulloblastomas and characterized their in vivo growth characteristics. Valproic acid treatment of these xenografts showed potent in vivo anti-medulloblastoma activity. These xenograft models should facilitate the understanding of medulloblastoma pathogenesis and future preclinical evaluation of new therapies against medulloblastoma.

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Year:  2006        PMID: 16899619     DOI: 10.1158/1078-0432.CCR-05-2849

Source DB:  PubMed          Journal:  Clin Cancer Res        ISSN: 1078-0432            Impact factor:   12.531


  31 in total

1.  Association of Valproic Acid Use, a Potent Histone Deacetylase Inhibitor, and Melanoma Risk.

Authors:  Afton Chavez; Charles P Quesenberry; Jeanne Darbinian; Maryam M Asgari
Journal:  J Invest Dermatol       Date:  2020-04-28       Impact factor: 8.551

2.  Concurrent Inhibition of Neurosphere and Monolayer Cells of Pediatric Glioblastoma by Aurora A Inhibitor MLN8237 Predicted Survival Extension in PDOX Models.

Authors:  Mari Kogiso; Lin Qi; Frank K Braun; Sarah G Injac; Linna Zhang; Yuchen Du; Huiyuan Zhang; Frank Y Lin; Sibo Zhao; Holly Lindsay; Jack M Su; Patricia A Baxter; Adekunle M Adesina; Debra Liao; Mark G Qian; Stacey Berg; Jodi A Muscal; Xiao-Nan Li
Journal:  Clin Cancer Res       Date:  2018-02-20       Impact factor: 12.531

3.  Efficacy of novel histone deacetylase inhibitor, AR42, in a mouse model of, human T-lymphotropic virus type 1 adult T cell lymphoma.

Authors:  Bevin Zimmerman; Aaron Sargeant; Kristina Landes; Soledad A Fernandez; Ching-Shih Chen; Michael D Lairmore
Journal:  Leuk Res       Date:  2011-07-29       Impact factor: 3.156

4.  Global gene expression profiling confirms the molecular fidelity of primary tumor-based orthotopic xenograft mouse models of medulloblastoma.

Authors:  Xiumei Zhao; Zhigang Liu; Litian Yu; Yujing Zhang; Patricia Baxter; Horatiu Voicu; Sivashankarappa Gurusiddappa; Joseph Luan; Jack M Su; Hon-chiu Eastwood Leung; Xiao-Nan Li
Journal:  Neuro Oncol       Date:  2012-03-29       Impact factor: 12.300

5.  Phase 1 study of valproic acid in pediatric patients with refractory solid or CNS tumors: a children's oncology group report.

Authors:  Jack M Su; Xiao-Nan Li; Patrick Thompson; Ching-Nan Ou; Ashish M Ingle; Heidi Russell; Ching C Lau; Peter C Adamson; Susan M Blaney
Journal:  Clin Cancer Res       Date:  2010-11-29       Impact factor: 12.531

6.  Valproic acid treatment response in vitro is determined by TP53 status in medulloblastoma.

Authors:  Bruna Mascaro-Cordeiro; Indhira Dias Oliveira; Francine Tesser-Gamba; Lorena Favaro Pavon; Nasjla Saba-Silva; Sergio Cavalheiro; Patrícia Dastoli; Silvia Regina Caminada Toledo
Journal:  Childs Nerv Syst       Date:  2018-05-22       Impact factor: 1.475

7.  Valproic acid reduces the tolerability of temsirolimus in children and adolescents with solid tumors.

Authors:  Don W Coulter; Christine Walko; Jai Patel; Billie M Moats-Staats; Andrew McFadden; Scott V Smith; Wasiuddin A Khan; Arlene S Bridges; Allison M Deal; Javier Oesterheld; Ian J Davis; Julie Blatt
Journal:  Anticancer Drugs       Date:  2013-04       Impact factor: 2.248

8.  Reactivation of death receptor 4 (DR4) expression sensitizes medulloblastoma cell lines to TRAIL.

Authors:  Dolly G Aguilera; Chandra M Das; Neeta D Sinnappah-Kang; Celine Joyce; Pete H Taylor; Sijin Wen; Martin Hasselblatt; Werner Paulus; Greg Fuller; Johannes E Wolff; Vidya Gopalakrishnan
Journal:  J Neurooncol       Date:  2009-01-16       Impact factor: 4.130

9.  HDAC and PI3K Antagonists Cooperate to Inhibit Growth of MYC-Driven Medulloblastoma.

Authors:  Yanxin Pei; Kun-Wei Liu; Jun Wang; Alexandra Garancher; Ran Tao; Lourdes A Esparza; Donna L Maier; Yoko T Udaka; Najiba Murad; Sorana Morrissy; Huriye Seker-Cin; Sebastian Brabetz; Lin Qi; Mari Kogiso; Simone Schubert; James M Olson; Yoon-Jae Cho; Xiao-Nan Li; John R Crawford; Michael L Levy; Marcel Kool; Stefan M Pfister; Michael D Taylor; Robert J Wechsler-Reya
Journal:  Cancer Cell       Date:  2016-03-14       Impact factor: 31.743

Review 10.  The molecular genetics of medulloblastoma: an assessment of new therapeutic targets.

Authors:  Carlos G Carlotti; Christian Smith; James T Rutka
Journal:  Neurosurg Rev       Date:  2008-06-12       Impact factor: 3.042

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