| Literature DB >> 16793264 |
Huiyong Hu1, Aleksandr Kolesnikov, Jennifer R Riggs, Kieron E Wesson, Robin Stephens, Ellen M Leahy, William D Shrader, Paul A Sprengeler, Michael J Green, Ellen Sanford, Margaret Nguyen, Erik Gjerstad, Ronnel Cabuslay, Wendy B Young.
Abstract
The 4-amino-5-azaindole as an amidino-benzimidazole replacement is described. A series of potent and selective analogs were discovered and showed desirable ex vivo efficacy as measured by PT.Entities:
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Year: 2006 PMID: 16793264 DOI: 10.1016/j.bmcl.2006.06.016
Source DB: PubMed Journal: Bioorg Med Chem Lett ISSN: 0960-894X Impact factor: 2.823