Literature DB >> 16774255

4,7-Dimethoxy-1,10-phenanthroline: an excellent ligand for the Cu-catalyzed N-arylation of imidazoles.

Ryan A Altman1, Stephen L Buchwald.   

Abstract

[reaction: see text] 4,7-Dimethoxy-1,10-phenanthroline (L) was found to be an efficient ligand for the copper-catalyzed N-arylation of imidazole with aryl iodides and bromides under mild conditions. A variety of hindered and functionalized imidazoles and aryl halides were transformed in good to excellent yields.

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Year:  2006        PMID： 16774255     DOI： 10.1021/ol0608505

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  9 in total

1.  Copper-Catalyzed Aerobic C-H Trifluoromethylation of Phenanthrolines.

Authors:  Cheng-Liang Zhu; Yong-Qiang Zhang; Yong-An Yuan; Hao Xu
Journal:  Synlett       Date:  2015       Impact factor: 2.454

2.  Structure-activity relationship studies and biological characterization of human NAD(+)-dependent 15-hydroxyprostaglandin dehydrogenase inhibitors.

Authors:  Damien Y Duveau; Adam Yasgar; Yuhong Wang; Xin Hu; Jennifer Kouznetsova; Kyle R Brimacombe; Ajit Jadhav; Anton Simeonov; Craig J Thomas; David J Maloney
Journal:  Bioorg Med Chem Lett       Date:  2013-12-04       Impact factor: 2.823

3.  Effect of Ligand Structure on the Electron Density and Activity of Iridium Catalysts for the Borylation of Alkanes.

Authors:  Matthew A Larsen; Raphael J Oeschger; John F Hartwig
Journal:  ACS Catal       Date:  2020-02-11       Impact factor: 13.084

4.  PIII /PV =O Catalyzed Cascade Synthesis of N-Functionalized Azaheterocycles.

Authors:  Trevor V Nykaza; Gen Li; Junyu Yang; Michael R Luzung; Alexander T Radosevich
Journal:  Angew Chem Int Ed Engl       Date:  2020-01-29       Impact factor: 15.336

5.  Synthesis and biological evaluation of analogues of the kinase inhibitor nilotinib as Abl and Kit inhibitors.

Authors:  Damien Y Duveau; Xin Hu; Martin J Walsh; Suneet Shukla; Amanda P Skoumbourdis; Matthew B Boxer; Suresh V Ambudkar; Min Shen; Craig J Thomas
Journal:  Bioorg Med Chem Lett       Date:  2012-12-10       Impact factor: 2.823

6.  Completely N1-selective palladium-catalyzed arylation of unsymmetric imidazoles: application to the synthesis of nilotinib.

Authors:  Satoshi Ueda; Mingjuan Su; Stephen L Buchwald
Journal:  J Am Chem Soc       Date:  2011-12-14       Impact factor: 15.419

7.  catena-Poly[[[bis-(nitrato-κO)copper(II)]-bis-[μ-1,3-bis-(imidazol-1-yl)-5-methyl-benzene-κ(2)N(3):N(3')]] dihydrate].

Authors:  Guang-Xiang Liu
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2012-05-31

8.  Silver Benzoate Facilitates the Copper-Catalyzed C-N Coupling of Iodoazoles with Aromatic Nitrogen Heterocycles.

Authors:  Cedric Lozano; Cristian Ramirez; Ny Sin; Hélène M-F Viart; Stanley B Prusiner; Nick A Paras; Jay Conrad
Journal:  ACS Omega       Date:  2021-03-31

Review 9.  Key Developments in Ionic Liquid Crystals.

Authors:  Alexandra Alvarez Fernandez; Paul H J Kouwer
Journal:  Int J Mol Sci       Date:  2016-05-16       Impact factor: 5.923
  9 in total

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