Literature DB >> 16757524

Long-term progestin-only contraceptives result in reduced endometrial blood flow and oxidative stress.

M Hickey1, G Krikun, P Kodaman, Frederick Schatz, C Carati, C J Lockwood.   

Abstract

CONTEXT: Because of their safety and efficacy, long-term progestin-only contraceptives (LTPOCs) are well-suited for women with restricted access to health care. However, abnormal uterine bleeding (AUB) causes half of all users to discontinue therapy within 12 months. Endometria of LTPOC-treated patients display aberrant angiogenesis with abnormally enlarged, thin-walled, fragile blood vessels, inflammation, and focal hemorrhage. In this study, similar effects were observed with a new third-generation implantable LTPOC.
OBJECTIVE: We hypothesized that LTPOC reduces uterine and endometrial blood flow, leading to hypoxia/reperfusion, which triggers the generation of reactive oxygen species. The latter induce aberrant angiogenesis, causing AUB.
DESIGN: Endometrial perfusion was measured by laser-Doppler fluxmetry in women requesting LTPOCs. Endometrial biopsies were obtained for in vivo and in vitro experiments.
SETTING: The study was conducted in the Yale University School of Medicine and Family-Planning Center in Western Australia. PATIENTS: Seven women 18 yr or older requesting implantable LTPOCs were recruited in Western Australia. INTERVENTION: Women received etonorgestrel implants. MAIN OUTCOME: LTPOC treatment resulted in reduced endometrial perfusion and increased endometrial oxidative damage.
CONCLUSIONS: We propose that LTPOCs result in hypoxia reperfusion, which leads to aberrant angiogenesis resulting in AUB.

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Year:  2006        PMID: 16757524     DOI: 10.1210/jc.2006-0724

Source DB:  PubMed          Journal:  J Clin Endocrinol Metab        ISSN: 0021-972X            Impact factor:   5.958


  11 in total

Review 1.  Mechanisms of normal and abnormal endometrial bleeding.

Authors:  Charles J Lockwood
Journal:  Menopause       Date:  2011-04       Impact factor: 2.953

Review 2.  The role of decidual cells in uterine hemostasis, menstruation, inflammation, adverse pregnancy outcomes and abnormal uterine bleeding.

Authors:  Frederick Schatz; Ozlem Guzeloglu-Kayisli; Sefa Arlier; Umit A Kayisli; Charles J Lockwood
Journal:  Hum Reprod Update       Date:  2016-02-23       Impact factor: 15.610

3.  Long-acting progestin-only contraceptives enhance human endometrial stromal cell expressed neuronal pentraxin-1 and reactive oxygen species to promote endothelial cell apoptosis.

Authors:  O Guzeloglu-Kayisli; M Basar; J P Shapiro; N Semerci; J S Huang; F Schatz; C J Lockwood; U A Kayisli
Journal:  J Clin Endocrinol Metab       Date:  2014-07-16       Impact factor: 5.958

4.  Long-acting progestin-only contraceptives impair endometrial vasculature by inhibiting uterine vascular smooth muscle cell survival.

Authors:  Umit A Kayisli; Murat Basar; Ozlem Guzeloglu-Kayisli; Nihan Semerci; Helen C Atkinson; John Shapiro; Taryn Summerfield; S Joseph Huang; Katja Prelle; Frederick Schatz; Charles J Lockwood
Journal:  Proc Natl Acad Sci U S A       Date:  2015-04-06       Impact factor: 11.205

5.  Effects of etonogestrel treatment in the reproductive organs and uterine arteries of nonoophorectomized guinea pigs.

Authors:  Graciela Krikun; C J Booth; L Buchwalder; F Schatz; G Osol; Maurizio Mandala; C J Lockwood
Journal:  Reprod Sci       Date:  2012-01-19       Impact factor: 3.060

6.  Mass spectrometry identification of potential mediators of progestin-only contraceptive-induced abnormal uterine bleeding in human endometrial stromal cells.

Authors:  John P Shapiro; Murat Basar; Umit A Kayisli; Ozlem Guzeloglu-Kayisli; S Joseph Huang; Adrian A Suarez; Hatice Gulcin Ozer; Frederick Schatz; Charles J Lockwood
Journal:  Contraception       Date:  2014-11-21       Impact factor: 3.375

7.  Long-term progestin contraceptives (LTPOC) induce aberrant angiogenesis, oxidative stress and apoptosis in the guinea pig uterus: A model for abnormal uterine bleeding in humans.

Authors:  Graciela Krikun; Irina A Buhimschi; Martha Hickey; Frederick Schatz; Lynn Buchwalder; Charles J Lockwood
Journal:  J Angiogenes Res       Date:  2010-04-27

Review 8.  Decidualized human endometrial stromal cells mediate hemostasis, angiogenesis, and abnormal uterine bleeding.

Authors:  Charles J Lockwood; Graciela Krikun; Martha Hickey; S Joseph Huang; Frederick Schatz
Journal:  Reprod Sci       Date:  2009-02       Impact factor: 3.060

9.  Progestins Upregulate FKBP51 Expression in Human Endometrial Stromal Cells to Induce Functional Progesterone and Glucocorticoid Withdrawal: Implications for Contraceptive- Associated Abnormal Uterine Bleeding.

Authors:  Ozlem Guzeloglu Kayisli; Umit A Kayisli; Murat Basar; Nihan Semerci; Frederick Schatz; Charles J Lockwood
Journal:  PLoS One       Date:  2015-10-05       Impact factor: 3.240

Review 10.  Solving the Puzzle: What Is the Role of Progestogens in Neovascularization?

Authors:  Zhi Xia; Jian Xiao; Qiong Chen
Journal:  Biomolecules       Date:  2021-11-12
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