Literature DB >> 1671420

Dual antagonists of platelet activating factor and histamine. Identification of structural requirements for dual activity of N-Acyl-4-(5,6-dihydro-11H-benzo [5,6]cyclohepta-[1,2-b]pyridin-11-ylidene)piperidines.

J J Piwinski1, J K Wong, M J Green, A K Ganguly, M M Billah, R E West, W Kreutner.   

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Year:  1991        PMID： 1671420     DOI： 10.1021/jm00105a069

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  9 in total

Review 1.  Classification of scaffold-hopping approaches.

Authors:  Hongmao Sun; Gregory Tawa; Anders Wallqvist
Journal:  Drug Discov Today       Date:  2011-10-26       Impact factor: 7.851

2.  Safety of rupatadine administered over a period of 1 year in the treatment of persistent allergic rhinitis: a multicentre, open-label study in Spain.

Authors:  Antonio Valero; Fernando de la Torre; José Antonio Castillo; Pilar Rivas; Alfonso del Cuvillo; Ignacio Antépara; Javier Borja; Esther Donado; Oriol Molà; Iñaki Izquierdo
Journal:  Drug Saf       Date:  2009       Impact factor: 5.606

3.  Cyclizations of phenylethyl-substituted pyridinecarboxaldehydes.

Authors:  Rajasekhar Reddy Naredla; Douglas A Klumpp
Journal:  Tetrahedron       Date:  2013-03-04       Impact factor: 2.457

Review 4.  Role of histamine and platelet-activating factor in allergic rhinitis.

Authors:  V Alfaro
Journal:  J Physiol Biochem       Date:  2004-06       Impact factor: 5.080

Review 5.  An overview of the synthetic routes to the best selling drugs containing 6-membered heterocycles.

Authors:  Marcus Baumann; Ian R Baxendale
Journal:  Beilstein J Org Chem       Date:  2013-10-30       Impact factor: 2.883

6.  Route to Prolonged Residence Time at the Histamine H1 Receptor: Growing from Desloratadine to Rupatadine.

Authors:  Reggie Bosma; Zhiyong Wang; Albert J Kooistra; Nick Bushby; Sebastiaan Kuhne; Jelle van den Bor; Michael J Waring; Chris de Graaf; Iwan J de Esch; Henry F Vischer; Robert J Sheppard; Maikel Wijtmans; Rob Leurs
Journal:  J Med Chem       Date:  2019-07-05       Impact factor: 7.446

7.  High pressure assisted synthetic approach for novel 6,7-dihydro-5H-benzo[6,7]cyclohepta[1,2-b]pyridine and 5,6-dihydrobenzo[h]quinoline derivatives and their assessment as anticancer agents.

Authors:  Haider Behbehani; Fatemah A Aryan; Kamal M Dawood; Hamada Mohamed Ibrahim
Journal:  Sci Rep       Date:  2020-12-10       Impact factor: 4.379

Review 8.  Prescribed drugs containing nitrogen heterocycles: an overview.

Authors:  Majid M Heravi; Vahideh Zadsirjan
Journal:  RSC Adv       Date:  2020-12-15       Impact factor: 4.036

9.  A direct comparison of efficacy between desloratadine and rupatadine in seasonal allergic rhinoconjunctivitis: a randomized, double-blind, placebo-controlled study.

Authors:  Kf Lukat; P Rivas; A Roger; Ml Kowalski; U Botzen; F Wessel; F Sanquer; I Agache; I Izquierdo
Journal:  J Asthma Allergy       Date:  2013-02-22
  9 in total

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