Literature DB >> 16641825

Vaginal and rectal topical microbicide development: safety and efficacy of 1.0% Savvy (C31G) in the pigtailed macaque.

Dorothy L Patton1, Yvonne T Cosgrove Sweeney, Jennifer E Balkus, Sharon L Hillier.   

Abstract

BACKGROUND: A 1.0% gel formulation of C31G, a surfactant, has been shown to have in vitro antiviral and antibacterial activity. GOAL: The goal of this study was to evaluate the safety and efficacy of vaginal and rectal applications of 1.0% Savvy (C31G) in the nonhuman primate model. STUDY
DESIGN: The safety of repeated 1.0% C31G application was evaluated by microflora, pH, vaginal biopsy, colposcopy, and rectal lavage. Efficacy in preventing chlamydial infection was documented by culture, nucleic acid amplification tests, and serology.
RESULTS: Repeated applications of Savvy (1.0% C31G) were not associated with significant changes in pH, microflora, or inflammatory infiltrates on tissues. No significant differences in epithelial desquamation were noted after rectal product use compared with placebo. Four of 6 animals were protected from chlamydial infection after pretreatment with Savvy. C31G was shown to be safe to both vaginal and rectal mucosal tissues and to the microflora with repeated daily use.
CONCLUSION: Savvy has an acceptable safety profile after repeated vaginal and rectal use. A single intravaginal application of 1.0% C31G provided partial protection from acquiring cervical chlamydial infection.

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Year:  2006        PMID: 16641825     DOI: 10.1097/01.olq.0000216022.18321.d3

Source DB:  PubMed          Journal:  Sex Transm Dis        ISSN: 0148-5717            Impact factor:   2.830


  13 in total

1.  A guide for standardizing colposcopic observations for the evaluation of topical microbicide products in the pigtailed macaque model.

Authors:  Dorothy L Patton
Journal:  J Med Primatol       Date:  2011-10-24       Impact factor: 0.667

Review 2.  Animal models for microbicide studies.

Authors:  Ronald S Veazey; Robin J Shattock; Per Johan Klasse; John P Moore
Journal:  Curr HIV Res       Date:  2012-01-01       Impact factor: 1.581

3.  Identification of rhesus macaque genital microbiota by 16S pyrosequencing shows similarities to human bacterial vaginosis: implications for use as an animal model for HIV vaginal infection.

Authors:  Gregory T Spear; Douglas Gilbert; Masoumeh Sikaroodi; Lara Doyle; Linda Green; Patrick M Gillevet; Alan L Landay; Ronald S Veazey
Journal:  AIDS Res Hum Retroviruses       Date:  2010-02       Impact factor: 2.205

4.  A comparison of lower genital tract glycogen and lactic acid levels in women and macaques: implications for HIV and SIV susceptibility.

Authors:  Paria Mirmonsef; Douglas Gilbert; Ronald S Veazey; Jing Wang; Sabrina R Kendrick; Gregory T Spear
Journal:  AIDS Res Hum Retroviruses       Date:  2011-06-28       Impact factor: 2.205

5.  High resolution imaging of epithelial injury in the sheep cervicovaginal tract: a promising model for testing safety of candidate microbicides.

Authors:  Kathleen L Vincent; Nigel Bourne; Brent A Bell; Gracie Vargas; Alai Tan; Daniel Cowan; Lawrence R Stanberry; Susan L Rosenthal; Massoud Motamedi
Journal:  Sex Transm Dis       Date:  2009-05       Impact factor: 2.830

Review 6.  Rectal microbicide development.

Authors:  Ian McGowan; Charlene Dezzutti
Journal:  Curr Top Microbiol Immunol       Date:  2014       Impact factor: 4.291

7.  The antimicrobial agent C31G is effective for therapy for HSV-1 ocular keratitis in the rabbit eye model.

Authors:  James M Hill; Ethan M Stern; Partha S Bhattacharjee; Daniel Malamud; Christian Clement; Paulo Rodriguez; Walter J Lukiw; Augusto C Ochoa; Timothy P Foster; Cruz Velasco; Harris E McFerrin
Journal:  Antiviral Res       Date:  2013-07-13       Impact factor: 5.970

8.  Microbicide safety/efficacy studies in animals: macaques and small animal models.

Authors:  Ronald S Veazey
Journal:  Curr Opin HIV AIDS       Date:  2008-09       Impact factor: 4.283

Review 9.  Rectal pre-exposure prophylaxis (PrEP).

Authors:  Lisa C Rohan; Haitao Yang; Lin Wang
Journal:  Antiviral Res       Date:  2013-11-01       Impact factor: 5.970

10.  A summary of preclinical topical microbicide rectal safety and efficacy evaluations in a pigtailed macaque model.

Authors:  Dorothy L Patton; Yvonne T Cosgrove Sweeney; Kathleen J Paul
Journal:  Sex Transm Dis       Date:  2009-06       Impact factor: 2.830

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