Literature DB >> 16543288

Crucial role of the melanocortin receptor MC1R in experimental colitis.

C Maaser1, K Kannengiesser, C Specht, A Lügering, T Brzoska, T A Luger, W Domschke, T Kucharzik.   

Abstract

BACKGROUND AND AIMS: alpha-Melanocyte stimulating hormone (alpha MSH) is known to exert anti-inflammatory effects, for example in murine DSS (dextran sodium sulphate induced) colitis. The anti-inflammatory functions of alpha MSH are mediated by the melanocortin1-receptor (MC1R) in an autoregulatory loop. The aim of this study was therefore to determine whether a breakdown of the alpha MSH-MC1R pathway leads to worsening of disease.
METHODS: Experimental colitis was induced in mice with a frameshift mutation in the MC1R gene (MC1Re/e), C57BL/6 wild type mice, and MC1Re/e-C57BL/6 bone marrow chimeras. The course of inflammation was monitored by weight loss, histological changes in the colon, and myeloperoxidase activity. In addition, MC1R expression was analysed in intestinal epithelial cells.
RESULTS: While the colon of untreated MC1Re/e appeared normal, the course of DSS-colitis in MC1Re/e mice was dramatically aggravated, with a significantly higher weight loss and marked histological changes compared to C57BL/6WT. The inflammation eventually led to death in all MC1Re/e, while all C57BL/6WT survived. Similar observations were detected in a transmissible murine colitis model induced by Citrobacter rodentium. Infected MC1Re/e showed delayed clearance of infection. To determine whether missing haematopoietic cell expressed MC1R was responsible, DSS colitis was induced in MC1Re/e-C57BL/6 bone marrow chimeras. MC1Re/e mice receiving MC1R+ bone marrow showed a similar course of inflammation to non-transplanted MC1Re/e. Likewise, transplantation of MC1R bone marrow into C57BL/6WT mice did not lead to any worsening of disease.
CONCLUSIONS: This is the first study to show a functional role of MC1R in intestinal inflammation. The data suggest a pivotal role of non-haematopoietic cell expressed MC1R in the host's response to pathogenic stimuli.

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Year:  2006        PMID: 16543288      PMCID: PMC1856418          DOI: 10.1136/gut.2005.083634

Source DB:  PubMed          Journal:  Gut        ISSN: 0017-5749            Impact factor:   23.059


  49 in total

1.  New highly specific agonistic peptides for human melanocortin MC(1) receptor.

Authors:  M Szardenings; R Muceniece; I Mutule; F Mutulis; J E Wikberg
Journal:  Peptides       Date:  2000-02       Impact factor: 3.750

2.  Developmentally regulated expression of alpha-MSH and MC-1 receptor in C57BL/6 mouse skin suggests functions beyond pigmentation.

Authors:  V A Botchkarev; N V Botchkareva; A Slominski; B Roloff; T Luger; R Paus
Journal:  Ann N Y Acad Sci       Date:  1999-10-20       Impact factor: 5.691

3.  Melanocortin-1 receptor polymorphisms and risk of melanoma: is the association explained solely by pigmentation phenotype?

Authors:  J S Palmer; D L Duffy; N F Box; J F Aitken; L E O'Gorman; A C Green; N K Hayward; N G Martin; R A Sturm
Journal:  Am J Hum Genet       Date:  2000-01       Impact factor: 11.025

4.  Melanocortin-1-receptor gene and sun sensitivity in individuals without red hair.

Authors:  E Healy; N Flannagan; A Ray; C Todd; I J Jackson; J N Matthews; M A Birch-Machin; J L Rees
Journal:  Lancet       Date:  2000-03-25       Impact factor: 79.321

Review 5.  Corticotropin releasing hormone and proopiomelanocortin involvement in the cutaneous response to stress.

Authors:  A Slominski; J Wortsman; T Luger; R Paus; S Solomon
Journal:  Physiol Rev       Date:  2000-07       Impact factor: 37.312

Review 6.  Mechanisms of antiinflammatory action of alpha-MSH peptides. In vivo and in vitro evidence.

Authors:  J M Lipton; H Zhao; T Ichiyama; G S Barsh; A Catania
Journal:  Ann N Y Acad Sci       Date:  1999-10-20       Impact factor: 5.691

7.  Human peripheral blood-derived dendritic cells express functional melanocortin receptor MC-1R.

Authors:  E Becher; K Mahnke; T Brzoska; D H Kalden; S Grabbe; T A Luger
Journal:  Ann N Y Acad Sci       Date:  1999-10-20       Impact factor: 5.691

8.  Mechanisms of the antiinflammatory effects of alpha-MSH. Role of transcription factor NF-kappa B and adhesion molecule expression.

Authors:  D H Kalden; T Scholzen; T Brzoska; T A Luger
Journal:  Ann N Y Acad Sci       Date:  1999-10-20       Impact factor: 5.691

9.  Molecular basis of the alpha-MSH/IL-1 antagonism.

Authors:  T Brzoska; D H Kalden; T Scholzen; T A Luger
Journal:  Ann N Y Acad Sci       Date:  1999-10-20       Impact factor: 5.691

10.  Preservation of eumelanin hair pigmentation in proopiomelanocortin-deficient mice on a nonagouti (a/a) genetic background.

Authors:  Andrzej Slominski; Przemyslaw M Plonka; Alexander Pisarchik; James L Smart; Virginie Tolle; Jacobo Wortsman; Malcolm J Low
Journal:  Endocrinology       Date:  2004-11-24       Impact factor: 4.736

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  30 in total

Review 1.  MC1R, eumelanin and pheomelanin: their role in determining the susceptibility to skin cancer.

Authors:  Tahseen H Nasti; Laura Timares
Journal:  Photochem Photobiol       Date:  2014-11-07       Impact factor: 3.421

Review 2.  Leveraging melanocortin pathways to treat glomerular diseases.

Authors:  Rujun Gong
Journal:  Adv Chronic Kidney Dis       Date:  2014-03       Impact factor: 3.620

3.  The melanocortin agonist AP214 exerts anti-inflammatory and proresolving properties.

Authors:  Trinidad Montero-Melendez; Hetal B Patel; Michael Seed; Søren Nielsen; Thomas E N Jonassen; Mauro Perretti
Journal:  Am J Pathol       Date:  2011-05-10       Impact factor: 4.307

4.  The tripeptide KdPT protects from intestinal inflammation and maintains intestinal barrier function.

Authors:  Dominik Bettenworth; Marion Buyse; Markus Böhm; Rudolf Mennigen; Isabel Czorniak; Klaus Kannengiesser; Thomas Brzoska; Thomas A Luger; Torsten Kucharzik; Wolfram Domschke; Christian Maaser; Andreas Lügering
Journal:  Am J Pathol       Date:  2011-07-08       Impact factor: 4.307

5.  The melanocortin MC(1) receptor agonist BMS-470539 inhibits leucocyte trafficking in the inflamed vasculature.

Authors:  G Leoni; M-B Voisin; K Carlson; Sj Getting; S Nourshargh; M Perretti
Journal:  Br J Pharmacol       Date:  2010-03-19       Impact factor: 8.739

6.  Inflammation-induced functional connectivity of melanin-concentrating hormone and IL-10.

Authors:  Dimitrios C Ziogas; Apostolos K A Karagiannis; Brenda M Geiger; Beatriz Gras-Miralles; Robert Najarian; Ofer Reizes; Leo R Fitzpatrick; Efi Kokkotou
Journal:  Peptides       Date:  2014-02-18       Impact factor: 3.750

7.  The neuropeptide alpha-melanocyte-stimulating hormone is critically involved in the development of cytotoxic CD8+ T cells in mice and humans.

Authors:  Karin Loser; Thomas Brzoska; Vinzenz Oji; Matteo Auriemma; Maik Voskort; Verena Kupas; Lars Klenner; Cornelius Mensing; Axel Hauschild; Stefan Beissert; Thomas A Luger
Journal:  PLoS One       Date:  2010-02-01       Impact factor: 3.240

8.  Gram-positive pathogenic bacteria induce a common early response in human monocytes.

Authors:  Svetlin Tchatalbachev; Rohit Ghai; Hamid Hossain; Trinad Chakraborty
Journal:  BMC Microbiol       Date:  2010-11-02       Impact factor: 3.605

9.  Functional melanocortin 1 receptor Mc1r is not necessary for an inflammatory response to UV radiation in adult mouse skin.

Authors:  Agnieszka Wolnicka-Glubisz; Edward De Fabo; Frances Noonan
Journal:  Exp Dermatol       Date:  2013-03       Impact factor: 3.960

10.  Inflamed phenotype of the mesenteric microcirculation of melanocortin type 3 receptor-null mice after ischemia-reperfusion.

Authors:  Giovanna Leoni; Hetal B Patel; André L F Sampaio; Felicity N E Gavins; Joanne F Murray; Paolo Grieco; Stephen J Getting; Mauro Perretti
Journal:  FASEB J       Date:  2008-08-29       Impact factor: 5.191

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