Literature DB >> 16516352

Synthesis and antimicrobial activity of new (E)-4-[piperidino (4'-methylpiperidino-, morpholino-) N-alkoxy]stilbenes.

Elzbieta Wyrzykiewicz1, Monika Wendzonka, Bogdan Kedzia.   

Abstract

The synthesis of twenty-one new (E)-4-[piperidino-(4;-methylpiperidino-, morpholino-)N-alkoxy] stilbenes is reported. The compounds were tested for antimicrobial activities against Gram-negative, Gram-positive bacteria, and fungi. In particular, compounds 3b, 3c, 3f, 3g, 3h, 3k, 3l showed good antibacterial activity against Staphylococcus aureus and 3h, 3k, 3m, 3n also against Bacillus subtilis, as well as 3h, 3n also against Streptococcus faecalis.

Entities:  

Mesh:

Substances:

Year:  2006        PMID: 16516352     DOI: 10.1016/j.ejmech.2005.11.010

Source DB:  PubMed          Journal:  Eur J Med Chem        ISSN: 0223-5234            Impact factor:   6.514


  5 in total

1.  Activity and synergistic interactions of stilbenes and antibiotic combinations against bacteria in vitro.

Authors:  S Nishanth Kumar; J V Siji; Bala Nambisan; C Mohandas
Journal:  World J Microbiol Biotechnol       Date:  2012-07-11       Impact factor: 3.312

2.  From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human α9α10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue.

Authors:  Francesco Bavo; Marco Pallavicini; Susanna Pucci; Rebecca Appiani; Alessandro Giraudo; Brek Eaton; Linda Lucero; Cecilia Gotti; Milena Moretti; Paul Whiteaker; Cristiano Bolchi
Journal:  J Med Chem       Date:  2022-07-14       Impact factor: 8.039

3.  Antimicrobial and antiurease activities of newly synthesized morpholine derivatives containing an azole nucleus.

Authors:  Hakan Bektaş; Sule Ceylan; Neslihan Demirbaş; Sengül Alpay-Karaoğlu; Bahar Bilgin Sökmen
Journal:  Med Chem Res       Date:  2012-11-29       Impact factor: 1.965

Review 4.  Synthetic approaches toward stilbenes and their related structures.

Authors:  Zulfiqar Ali Khan; Ahsan Iqbal; Sohail Anjum Shahzad
Journal:  Mol Divers       Date:  2017-04-21       Impact factor: 2.943

5.  Microwave-Assisted Synthesis, Structural Characterization and Assessment of the Antibacterial Activity of Some New Aminopyridine, Pyrrolidine, Piperidine and Morpholine Acetamides.

Authors:  Abdulmajeed S H Alsamarrai; Saba S Abdulghani
Journal:  Molecules       Date:  2021-01-20       Impact factor: 4.411

  5 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.