Literature DB >> 16446832

Lithocholic acid analogues, new and potent alpha-2,3-sialyltransferase inhibitors.

Kai-Hsuan Chang1, Lenselot Lee, Jessica Chen, Wen-Shan Li.   

Abstract

A new type of noncompetitive alpha-2,3-sialyltransferase inhibitor has been synthesized; we report the discovery, preparation and inhibitory activity of sixteen lithocholic acid analogues.

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Year:  2006        PMID： 16446832     DOI： 10.1039/b514915k

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  9 in total

1.  Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor.

Authors:  Matteo Incerti; Massimiliano Tognolini; Simonetta Russo; Daniele Pala; Carmine Giorgio; Iftiin Hassan-Mohamed; Roberta Noberini; Elena B Pasquale; Paola Vicini; Silvia Piersanti; Silvia Rivara; Elisabetta Barocelli; Marco Mor; Alessio Lodola
Journal:  J Med Chem       Date:  2013-03-22       Impact factor: 7.446

2.  Identification of non-substrate-like glycosyltransferase inhibitors from library screening: pitfalls & hits.

Authors:  Masaki Ema; Yong Xu; Sebastian Gehrke; Gerd K Wagner
Journal:  Medchemcomm       Date:  2017-11-29       Impact factor: 3.597

Review 3.  Biosynthetic Machinery Involved in Aberrant Glycosylation: Promising Targets for Developing of Drugs Against Cancer.

Authors:  Andréia Vasconcelos-Dos-Santos; Isadora A Oliveira; Miguel Clodomiro Lucena; Natalia Rodrigues Mantuano; Stephen A Whelan; Wagner Barbosa Dias; Adriane Regina Todeschini
Journal:  Front Oncol       Date:  2015-06-25       Impact factor: 6.244

Review 4.  Selectins-The Two Dr. Jekyll and Mr. Hyde Faces of Adhesion Molecules-A Review.

Authors:  Igor Tvaroška; Chandrabose Selvaraj; Jaroslav Koča
Journal:  Molecules       Date:  2020-06-19       Impact factor: 4.411

5.  Semi-synthesis of β-keto-1,2,3-triazole derivatives from ethinylestradiol and evaluation of the cytotoxic activity.

Authors:  Thayane M Queiroz; Erika V M Orozco; Valdenizia R Silva; Luciano S Santos; Milena B P Soares; Daniel P Bezerra; André L M Porto
Journal:  Heliyon       Date:  2019-09-06

6.  LINEAGE: Label-free identification of endogenous informative single-cell mitochondrial RNA mutation for lineage analysis.

Authors:  Li Lin; Yufeng Zhang; Weizhou Qian; Yao Liu; Yingkun Zhang; Fanghe Lin; Cenxi Liu; Guangxing Lu; Di Sun; Xiaoxu Guo; YanLing Song; Jia Song; Chaoyong Yang; Jin Li
Journal:  Proc Natl Acad Sci U S A       Date:  2022-02-01       Impact factor: 12.779

Review 7.  Aberrant Sialylation in Cancer: Therapeutic Opportunities.

Authors:  Jennifer Munkley
Journal:  Cancers (Basel)       Date:  2022-08-31       Impact factor: 6.575

8.  Establishment of In Vitro and In Vivo Anticolorectal Cancer Efficacy of Lithocholic Acid-Based Imidazolium Salts.

Authors:  Diana Sawicka; Agnieszka Hryniewicka; Sylwia Gohal; Anna Sadowska; Anna Pryczynicz; Katarzyna Guzińska-Ustymowicz; Emilia Sokołowska; Jacek W Morzycki; Halina Car
Journal:  Int J Mol Sci       Date:  2022-06-24       Impact factor: 6.208

9.  HCV poly U/UC sequence-induced inflammation leads to metabolic disorders in vulvar lichen sclerosis.

Authors:  Qing Cong; Xiao Guo; Shengwei Zhang; Jinhui Wang; Yi Zhu; Lili Wang; Guangxing Lu; Yufeng Zhang; Wei Fu; Liying Zhou; Shuaikang Wang; Cenxi Liu; Jia Song; Chaoyong Yang; Chi Luo; Ting Ni; Long Sui; He Huang; Jin Li
Journal:  Life Sci Alliance       Date:  2021-06-18
  9 in total

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