Literature DB >> 16437685

Cyclosporine A, FK-506, 40-0-[2-hydroxyethyl]rapamycin and mycophenolate mofetil inhibit proliferation of human intrahepatic biliary epithelial cells in vitro.

Chao Liu1, Thomas Schreiter, Andrea Frilling, Uta Dahmen, Christoph E Broelsch, Guido Gerken, Ulrich Treichel.   

Abstract

AIM: To investigate the effect of cyclosporine A (CsA), FK-506, and mycophenolate mofetil (MMF) and 40-0-[2-hydroxyethyl]rapamycin (RAD) on proliferation of human intrahepatic biliary epithelial cells (BECs) in vitro.
METHODS: BECs were isolated from six human liver tissuespecimens with the immunomagnetic separation method and treated with different concentrations of CsA, FK-506, RAD, and MMF in vitro. Proliferation of the cells was measured by MTT assay at 24 and 48 h after treatment, respectively. One-way analysis of variance was used to analyze the results. Expression of CK 19 in BECs was monitored by flow cytometry and Western blot.
RESULTS: Six lines of BECs were established. They survived for 4-18 wk in vitro. Flow cytometry analysis showed that these cells always expressed CK19. CsA, FK-506, RAD, and MMF inhibited proliferation of BECs in a dose-dependent manner. The lowest concentration of CsA, FK-506, RAD, and MMF to inhibit proliferation of BECs (P<0.05) was 500, 100, 0.25, and 100 mug/L, respectively. However, the expression of CK19 by BECs was not changed.
CONCLUSION: CsA, FK-506, RAD, and MMF have an antiproliferative effect on human intrahepatic BECs in vitro, while RAD has the strongest growth-inhibitory effect. Their possible effects on liver regeneration and bile duct injury in transplant patients should be further investigated.

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Year:  2005        PMID: 16437685      PMCID: PMC4727236          DOI: 10.3748/wjg.v11.i48.7602

Source DB:  PubMed          Journal:  World J Gastroenterol        ISSN: 1007-9327            Impact factor:   5.742


  18 in total

1.  The effect of mycophenolate mofetil on liver regeneration.

Authors:  P Motale; A Mall; C W Spearman; Z Lotz; M Tyler; E Shepherd; D Kahn
Journal:  Transplant Proc       Date:  2001 Feb-Mar       Impact factor: 1.066

2.  Hepatotrophic effect of cyclosporine and FK 506 is not mimicked by rapamycin.

Authors:  R Chávez; N Jamieson; S Takamori; S Nivatvongs; G Pino; A Metcalfe; C Watson; D Romero; S Metcalfe
Journal:  Transplant Proc       Date:  1999-09       Impact factor: 1.066

3.  Biliary epithelial cells from the liver of patients with primary biliary cirrhosis: isolation, characterization, and short-term culture.

Authors:  R Joplin; A J Strain; J M Neuberger
Journal:  J Pathol       Date:  1990-11       Impact factor: 7.996

4.  Hepatotrophic effects of FK506 in dogs.

Authors:  T E Starzl; K A Porter; V Mazzaferro; S Todo; J Fung; A Francavilla
Journal:  Transplantation       Date:  1991-01       Impact factor: 4.939

Review 5.  Isolated hepatocytes: use in experimental and clinical hepatology.

Authors:  A J Strain
Journal:  Gut       Date:  1994-04       Impact factor: 23.059

6.  Augmentation of rat liver regeneration by FK 506 compared with cyclosporin.

Authors:  A Francavilla; M Barone; S Todo; Q Zeng; K A Porter; T E Starzl
Journal:  Lancet       Date:  1989-11-25       Impact factor: 79.321

7.  The hepatotropic influence of cyclosporine.

Authors:  V Mazzaferro; K A Porter; C L Scotti-Foglieni; R Venkataramanan; L Makowka; L Rossaro; A Francavilla; S Todo; D H Van Thiel; T E Starzl
Journal:  Surgery       Date:  1990-05       Impact factor: 3.982

8.  Effect of cyclosporine on liver regeneration after orthotopic reduced-size hepatic transplantation in the rat.

Authors:  N Kikuchi; Y Yamaguchi; K Mori; N Takata; M Goto; Y Makino; H Hamaguchi; N Hisama; M Ogawa
Journal:  Dig Dis Sci       Date:  1993-08       Impact factor: 3.199

9.  Azathioprine and the liver. Evidence favoring idiosyncratic, mixed cholestatic-hepatocellular injury in humans.

Authors:  R A DePinho; C S Goldberg; J H Lefkowitch
Journal:  Gastroenterology       Date:  1984-01       Impact factor: 22.682

10.  Cyclosporine augments hepatic regenerative response in rats.

Authors:  D Kahn; L Makowka; H Lai; P K Eagon; V Dindzans; T E Starzl; D H Van Thiel
Journal:  Dig Dis Sci       Date:  1990-03       Impact factor: 3.199

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  3 in total

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Authors:  Yan-Kui Chu; Yi Liu; Ji-Kai Yin; Nan Wang; Liang Cai; Jian-Guo Lu
Journal:  World J Hepatol       Date:  2010-08-27

2.  Effects of mycophenolate mofetil on proliferation and mucin-5AC expression in human conjunctival goblet cells in vitro.

Authors:  Hong He; Hui Ding; Aiping Liao; Qiong Liu; Jun Yang; Xingwu Zhong
Journal:  Mol Vis       Date:  2010-10-01       Impact factor: 2.367

Review 3.  Adverse effects of immunosuppressant drugs upon airway epithelial cell and mucociliary clearance: implications for lung transplant recipients.

Authors:  Rogerio Pazetti; Paulo Manuel Pêgo-Fernandes; Fabio Biscegli Jatene
Journal:  Drugs       Date:  2013-07       Impact factor: 9.546

  3 in total

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