Literature DB >> 16375751

A2B adenosine receptor antagonists: recent developments.

Barbara Cacciari1, Giorgia Pastorin, Chiara Bolcato, Giampiero Spalluto, Magdalena Bacilieri, Stefano Moro.   

Abstract

There are pharmacological evidences that A(2B) receptors are involved in inflammatory processes, such as asthma. For this reason, many efforts has been made for identifying selective A(2B) antagonists as anti-asthmatic agents. The updated material related to this field has been rationalised and arranged in order to offer an overview of the topic.

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Year:  2005        PMID: 16375751     DOI: 10.2174/138955705774933374

Source DB:  PubMed          Journal:  Mini Rev Med Chem        ISSN: 1389-5575            Impact factor:   3.862


  9 in total

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Review 5.  The Role of Adenosine Signaling in Headache: A Review.

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Review 8.  Allosteric Modulation of Adenosine A2A Receptors as a New Therapeutic Avenue.

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9.  Progress in the discovery of selective, high affinity A(2B) adenosine receptor antagonists as clinical candidates.

Authors:  Rao V Kalla; Jeff Zablocki
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  9 in total

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