Literature DB >> 16277306

Benzotriazole-assisted thioacylation.

Alan R Katritzky1, Rachel M Witek, Valerie Rodriguez-Garcia, Prabhu P Mohapatra, James W Rogers, Janet Cusido, Ashraf A A Abdel-Fattah, Peter J Steel.   

Abstract

[Chemical reaction: See text] Benzotriazole reagents for thioacylation (RCSBt), thiocarbamoylation (RR'NCSBt), aryl/alkoxythioacylation (ROCSBt), and aryl/alkylthiothioacylation (RSCSBt) are synthesized, and their utility is assessed by syntheses of representative heteroaryl thioureas 3a-g, thioamides 15a-s, thionoesters 16a-h, thiocarbamates 17a-e, dithiocarbamates 18a-d, thiocarbonates 19a-c, and dithiocarbonates 20a-c.

Entities:  

Year:  2005        PMID： 16277306     DOI： 10.1021/jo050670t

Source DB:  PubMed          Journal:  J Org Chem        ISSN： 0022-3263            Impact factor:   4.354


  11 in total

1.  Halogenated benzimidazole carboxamides target integrin alpha4beta1 on T-cell and B-cell lymphomas.

Authors:  Richard D Carpenter; Arutselvan Natarajan; Edmond Y Lau; Mirela Andrei; Danielle M Solano; Felice C Lightstone; Sally J Denardo; Kit S Lam; Mark J Kurth
Journal:  Cancer Res       Date:  2010-06-08       Impact factor: 12.701

2.  Thiorhodamines containing amide and thioamide functionality as inhibitors of the ATP-binding cassette drug transporter P-glycoprotein (ABCB1).

Authors:  Alexandra Orchard; Gregory A Schamerhorn; Brandon D Calitree; Geri A Sawada; Tip W Loo; M Claire Bartlett; David M Clarke; Michael R Detty
Journal:  Bioorg Med Chem       Date:  2012-06-07       Impact factor: 3.641

3.  Thioamides in the collagen triple helix.

Authors:  Robert W Newberry; Brett VanVeller; Ronald T Raines
Journal:  Chem Commun (Camb)       Date:  2015-06-14       Impact factor: 6.222

4.  Rhodamine inhibitors of P-glycoprotein: an amide/thioamide "switch" for ATPase activity.

Authors:  Michael K Gannon; Jason J Holt; Stephanie M Bennett; Bryan R Wetzel; Tip W Loo; M Claire Bartlett; David M Clarke; Geri A Sawada; J William Higgins; Gregory Tombline; Thomas J Raub; Michael R Detty
Journal:  J Med Chem       Date:  2009-05-28       Impact factor: 7.446

5.  Selenorhodamine photosensitizers for photodynamic therapy of P-glycoprotein-expressing cancer cells.

Authors:  Jacqueline E Hill; Michelle K Linder; Kellie S Davies; Geri A Sawada; Janet Morgan; Tymish Y Ohulchanskyy; Michael R Detty
Journal:  J Med Chem       Date:  2014-10-01       Impact factor: 7.446

Review 6.  Mechanochemistry: A Force of Synthesis.

Authors:  Jean-Louis Do; Tomislav Friščić
Journal:  ACS Cent Sci       Date:  2016-12-29       Impact factor: 14.553

Review 7.  Mechanochemistry as an emerging tool for molecular synthesis: what can it offer?

Authors:  Joseph L Howard; Qun Cao; Duncan L Browne
Journal:  Chem Sci       Date:  2018-03-07       Impact factor: 9.825

Review 8.  Main group mechanochemistry.

Authors:  Agota A Gečiauskaitė; Felipe García
Journal:  Beilstein J Org Chem       Date:  2017-10-05       Impact factor: 2.883

Review 9.  Mechanochemical synthesis of thioureas, ureas and guanidines.

Authors:  Vjekoslav Štrukil
Journal:  Beilstein J Org Chem       Date:  2017-09-01       Impact factor: 2.883

10.  Modulating multi-functional ERK complexes by covalent targeting of a recruitment site in vivo.

Authors:  Tamer S Kaoud; William H Johnson; Nancy D Ebelt; Andrea Piserchio; Diana Zamora-Olivares; Sabrina X Van Ravenstein; Jacey R Pridgen; Ramakrishna Edupuganti; Rachel Sammons; Micael Cano; Mangalika Warthaka; Matthew Harger; Clint D J Tavares; Jihyun Park; Mohamed F Radwan; Pengyu Ren; Eric V Anslyn; Kenneth Y Tsai; Ranajeet Ghose; Kevin N Dalby
Journal:  Nat Commun       Date:  2019-11-19       Impact factor: 14.919
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