| Literature DB >> 16219463 |
Richard Chesworth1, Matthew D Wessel, Lisa Heyden, F Michael Mangano, Michael Zawistoski, Laura Gegnas, David Galluzzo, Bruce Lefker, Kimberly O Cameron, Jeanne Tickner, Bihong Lu, Tessa A Castleberry, Donna N Petersen, Amy Brault, Pia Perry, Oicheng Ng, Thomas A Owen, Lydia Pan, Hua-Zhu Ke, Thomas A Brown, David D Thompson, Paul DaSilva-Jardine.
Abstract
A series of ligands with varying heterocyclic cores and substituents that display a range of selectivity's (up to >100x) for ER-beta over ER-alpha are reported.Entities:
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Year: 2005 PMID: 16219463 DOI: 10.1016/j.bmcl.2005.08.010
Source DB: PubMed Journal: Bioorg Med Chem Lett ISSN: 0960-894X Impact factor: 2.823