Literature DB >> 16183277

Synthesis and HIV-1 integrase inhibitory activities of caffeic acid dimers derived from Salvia officinalis.

Fabrice Bailly1, Clémence Queffelec, Gladys Mbemba, Jean-François Mouscadet, Philippe Cotelle.   

Abstract

The synthesis of two caffeoyl-coumarin conjugates, derived from sagecoumarin, has been accomplished, starting from ferulic acid, isoferulic acid and sesamol. Both compounds exhibited potent inhibitory activities at micromolar concentrations against HIV-1 integrase in 3'-end processing reaction but were less effective against HIV-1 replication in a single-round infection assay of HeLa-beta-gal-CD4+ cells.

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Year:  2005        PMID： 16183277     DOI： 10.1016/j.bmcl.2005.07.091

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  5 in total

Review 1.  HIV-1 IN inhibitors: 2010 update and perspectives.

Authors:  Christophe Marchand; Kasthuraiah Maddali; Mathieu Métifiot; Yves Pommier
Journal:  Curr Top Med Chem       Date:  2009       Impact factor: 3.295

2.  6-Hy-droxy-2H-1,3-benzodioxole-5-carbaldehyde.

Authors:  Mehbub I K Momin; Neil Koorbanally; Deresh Ramjugernath; Muhammad D Bala
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2011-09-17

3.  Comparative Analysis of Phenolic Compound Characterization and Their Biosynthesis Genes between Two Diverse Bread Wheat (Triticum aestivum) Varieties Differing for Chapatti (Unleavened Flat Bread) Quality.

Authors:  Monica Sharma; Rajat Sandhir; Anuradha Singh; Pankaj Kumar; Ankita Mishra; Sanjay Jachak; Sukhvinder P Singh; Jagdeep Singh; Joy Roy
Journal:  Front Plant Sci       Date:  2016-12-15       Impact factor: 5.753

Review 4.  Potential of selected Lamiaceae plants in anti(retro)viral therapy.

Authors:  Maja Bekut; Snežana Brkić; Nebojša Kladar; Gordana Dragović; Neda Gavarić; Biljana Božin
Journal:  Pharmacol Res       Date:  2017-12-16       Impact factor: 7.658

Review 5.  Medicinal Plants Used in the Treatment of Human Immunodeficiency Virus.

Authors:  Bahare Salehi; Nanjangud V Anil Kumar; Bilge Şener; Mehdi Sharifi-Rad; Mehtap Kılıç; Gail B Mahady; Sanja Vlaisavljevic; Marcello Iriti; Farzad Kobarfard; William N Setzer; Seyed Abdulmajid Ayatollahi; Athar Ata; Javad Sharifi-Rad
Journal:  Int J Mol Sci       Date:  2018-05-14       Impact factor: 5.923
  5 in total

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