Literature DB >> 16144892

Comparison of rosiglitazone and metformin for treating HIV lipodystrophy: a randomized trial.

Jeroen P H van Wijk1, Eelco J P de Koning, Manuel Castro Cabezas, Jos op't Roodt, Jorge Joven, Ton J Rabelink, Andy I Hoepelman.   

Abstract

BACKGROUND: The use of antiretroviral combination therapy in HIV has been associated with lipodystrophy and cardiovascular risk factors.
OBJECTIVE: To compare the effects of the peroxisome proliferator-activated receptor-gamma agonist rosiglitazone and metformin for treating HIV lipodystrophy.
DESIGN: An open, randomized, 6-month clinical trial.
SETTING: University Medical Center, Utrecht, the Netherlands. PATIENTS: 39 HIV-infected men with lipodystrophy. INTERVENTION: Rosiglitazone, 8 g/d, or metformin, 2 g/d [DOSAGE ERROR CORRECTED] MEASUREMENTS: Insulin sensitivity estimated by the oral glucose tolerance test, subcutaneous and visceral abdominal fat measured by single-slice computed tomography, endothelial function measured by flow-mediated vasodilation, and fasting plasma measurements. Two patients in the metformin group withdrew from the study. Complete case analysis was performed.
RESULTS: Compared with metformin, rosiglitazone increased subcutaneous abdominal fat (between-treatment change from baseline, 27 cm2 [95% CI, 7 cm2 to 46 cm2]) and visceral abdominal fat (between-treatment change from baseline, 24 cm2 [CI, 6 cm2 to 51 cm2]). The area under the curve for insulin after the oral glucose tolerance test decreased similarly with both agents, but only rosiglitazone increased adiponectin levels. Metformin showed greater benefits on fasting lipid profile than rosiglitazone. Flow-mediated vasodilation statistically significantly increased with metformin (mean change, 1.5% [CI, 0.4% to 3.3%]) and not with rosiglitazone (mean change, 0.7% [CI, -1.1% to 2.7%]). The metformin versus rosiglitazone increases did not statistically differ. Rosiglitazone and metformin did not change C-reactive protein levels. LIMITATIONS: This small trial was not blinded or placebo-controlled and did not measure clinical outcomes.
CONCLUSIONS: The findings emphasize the importance of individualized care in HIV-infected patients. Although rosiglitazone may partly correct lipoatrophy, metformin improves visceral fat accumulation, fasting lipid profile, and endothelial function.

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Year:  2005        PMID: 16144892     DOI: 10.7326/0003-4819-143-5-200509060-00009

Source DB:  PubMed          Journal:  Ann Intern Med        ISSN: 0003-4819            Impact factor:   25.391


  34 in total

1.  Rosiglitazone improves lipoatrophy in patients receiving thymidine-sparing regimens.

Authors:  Marisa Tungsiripat; Dalia El Bejjani; Nesrine Rizk; Mary Ann O'riordan; Allison C Ross; Corrilynn Hileman; Norma Storer; Danielle Harrill; Grace A McComsey
Journal:  AIDS       Date:  2010-06-01       Impact factor: 4.177

Review 2.  Lipodystrophy: pathophysiology and advances in treatment.

Authors:  Christina G Fiorenza; Sharon H Chou; Christos S Mantzoros
Journal:  Nat Rev Endocrinol       Date:  2010-11-16       Impact factor: 43.330

Review 3.  Exploration and Development of PPAR Modulators in Health and Disease: An Update of Clinical Evidence.

Authors:  Hong Sheng Cheng; Wei Ren Tan; Zun Siong Low; Charlie Marvalim; Justin Yin Hao Lee; Nguan Soon Tan
Journal:  Int J Mol Sci       Date:  2019-10-11       Impact factor: 5.923

Review 4.  Aging and HIV infection.

Authors:  Rakhi Kohli; Robert S Klein; Ellie E Schoenbaum; Kathryn Anastos; Howard Minkoff; Henry S Sacks
Journal:  J Urban Health       Date:  2006-01       Impact factor: 3.671

Review 5.  Impact of antiretroviral therapy on growth, body composition and metabolism in pediatric HIV patients.

Authors:  Roy J Kim; Richard M Rutstein
Journal:  Paediatr Drugs       Date:  2010-06       Impact factor: 3.022

6.  Metabolic abnormalities in HIV-infected patients: an update.

Authors:  Todd T Brown; Joseph Cofrancesco
Journal:  Curr Infect Dis Rep       Date:  2006-11       Impact factor: 3.725

7.  The effects of recombinant human leptin on visceral fat, dyslipidemia, and insulin resistance in patients with human immunodeficiency virus-associated lipoatrophy and hypoleptinemia.

Authors:  Kathleen Mulligan; Hootan Khatami; Jean-Marc Schwarz; Giorgos K Sakkas; Alex M DePaoli; Viva W Tai; Michael J Wen; Grace A Lee; Carl Grunfeld; Morris Schambelan
Journal:  J Clin Endocrinol Metab       Date:  2009-01-27       Impact factor: 5.958

8.  Changes in Inflammation, Oxidative Stress, Mitochondrial DNA Content after Rosiglitazone in HIV Lipoatrophy.

Authors:  Marisa Tungsiripat; Dalia El-Bejjani; Nesrine Rizk; Bo Hu; Allison C Ross; Ulrich A Walker; Dirk Lebrecht; Ginger Milne; Norma Storer; Grace A McComsey
Journal:  J AIDS Clin Res       Date:  2012-10-15

9.  PPARalpha and PPARgamma attenuate HIV-induced dysregulation of tight junction proteins by modulations of matrix metalloproteinase and proteasome activities.

Authors:  Wen Huang; Sung Yong Eum; Ibolya E András; Bernhard Hennig; Michal Toborek
Journal:  FASEB J       Date:  2009-01-13       Impact factor: 5.191

10.  The efficacy and safety of insulin-sensitizing drugs in HIV-associated lipodystrophy syndrome: a meta-analysis of randomized trials.

Authors:  Siddharth H Sheth; Robin J Larson
Journal:  BMC Infect Dis       Date:  2010-06-23       Impact factor: 3.090

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