Literature DB >> 1613758

(E)-1,3-dialkyl-7-methyl-8-(3,4,5-trimethoxystyryl)xanthines: potent and selective adenosine A2 antagonists.

J Shimada1, F Suzuki, H Nonaka, A Ishii, S Ichikawa.   

Abstract

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Year:  1992        PMID： 1613758     DOI： 10.1021/jm00090a027

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  23 in total

1.  The utilization of a unified pharmacophore query in the discovery of new antagonists of the adenosine receptor family.

Authors:  T R Webb; N Melman; D Lvovskiy; X D Ji; K A Jacobson
Journal:  Bioorg Med Chem Lett       Date:  2000-01-03       Impact factor: 2.823

Review 2.  Xanthines as adenosine receptor antagonists.

Authors:  Christa E Müller; Kenneth A Jacobson
Journal:  Handb Exp Pharmacol       Date:  2011

3.  Evidence for high-affinity binding sites for the adenosine A2A receptor agonist [3H] CGS 21680 in the rat hippocampus and cerebral cortex that are different from striatal A2A receptors.

Authors:  R A Cunha; B Johansson; M D Constantino; A M Sebastião; B B Fredholm
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1996-02       Impact factor: 3.000

4.  Adenosine A2A receptors mediate the inhibitory effect of adenosine on formyl-Met-Leu-Phe-stimulated respiratory burst in neutrophil leucocytes.

Authors:  B B Fredholm; Y Zhang; I van der Ploeg
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1996 Aug-Sep       Impact factor: 3.000

5.  Molecular modeling of adenosine receptors. The ligand binding site on the rat adenosine A2A receptor.

Authors:  A P IJzerman; E M van der Wenden; P J van Galen; K A Jacobson
Journal:  Eur J Pharmacol       Date:  1994-06-15       Impact factor: 4.432

Review 6.  Nomenclature and classification of purinoceptors.

Authors:  B B Fredholm; M P Abbracchio; G Burnstock; J W Daly; T K Harden; K A Jacobson; P Leff; M Williams
Journal:  Pharmacol Rev       Date:  1994-06       Impact factor: 25.468

7.  Structure-activity relationships of 8-styrylxanthines as A2-selective adenosine antagonists.

Authors:  K A Jacobson; C Gallo-Rodriguez; N Melman; B Fischer; M Maillard; A van Bergen; P J van Galen; Y Karton
Journal:  J Med Chem       Date:  1993-05-14       Impact factor: 7.446

8.  Covalent binding of a selective agonist irreversibly activates guinea pig coronary artery A2 adenosine receptors.

Authors:  K Niiya; K A Jacobson; S K Silvia; R A Olsson
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1993-05       Impact factor: 3.000

9.  Evidence for P2-purinoceptor-mediated inhibition of noradrenaline release in rat brain cortex.

Authors:  I von Kügelgen; L Späth; K Starke
Journal:  Br J Pharmacol       Date:  1994-11       Impact factor: 8.739

10.  In vitro pharmacological profile of the A2A receptor antagonist istradefylline.

Authors:  Mayumi Saki; Koji Yamada; Etsuko Koshimura; Katsutoshi Sasaki; Tomoyuki Kanda
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  2013-06-29       Impact factor: 3.000
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