| Literature DB >> 16134929 |
Mark Wittman1, Joan Carboni, Ricardo Attar, Balu Balasubramanian, Praveen Balimane, Patrick Brassil, Francis Beaulieu, Chiehying Chang, Wendy Clarke, Janet Dell, Jeffrey Eummer, David Frennesson, Marco Gottardis, Ann Greer, Steven Hansel, Warren Hurlburt, Bruce Jacobson, Subramaniam Krishnananthan, Francis Y Lee, Aixin Li, Tai-An Lin, Peiying Liu, Carl Ouellet, Xiaopeng Sang, Mark G Saulnier, Karen Stoffan, Yax Sun, Upender Velaparthi, Henry Wong, Zheng Yang, Kurt Zimmermann, Mary Zoeckler, Dolatrai Vyas.
Abstract
Compound 3 (BMS-536924), a novel small-molecule inhibitor of the insulin-like growth factor receptor kinase with equal potency against the insulin receptor is described. The in vitro and in vivo biological activity of this interesting compound is also reported.Entities:
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Year: 2005 PMID: 16134929 DOI: 10.1021/jm050392q
Source DB: PubMed Journal: J Med Chem ISSN: 0022-2623 Impact factor: 7.446