Literature DB >> 16106299

A straightforward approach towards thiazoles and endothiopeptides via Ugi reaction.

Uli Kazmaier1, Stefanie Ackermann.   

Abstract

Endothiopeptides can easily be obtained via Ugi reaction using thio acids as acid components. If isonitriles with an acetal group are applied, the endothiopeptides can directly be converted into thiazoles using TMSCl-NaI under microwave irradiation.

Entities:  

Mesh：

Substances：

Year:  2005        PMID： 16106299     DOI： 10.1039/b507028g

Source DB:  PubMed          Journal:  Org Biomol Chem        ISSN： 1477-0520            Impact factor:   3.876


  8 in total

1.  Construction of functionalized tricyclic dihydropyrazino-quinazolinedione chemotypes via an Ugi/N-acyliminium ion cyclization cascade.

Authors:  Steven Gunawan; Christopher Hulme
Journal:  Tetrahedron Lett       Date:  2013-08-14       Impact factor: 2.415

Review 2.  Controlled microwave heating in modern organic synthesis: highlights from the 2004-2008 literature.

Authors:  C Oliver Kappe; Doris Dallinger
Journal:  Mol Divers       Date:  2009-04-21       Impact factor: 2.943

3.  A straightforward approach towards combined α-amino and α-hydroxy acids based on Passerini reactions.

Authors:  Ameer F Zahoor; Sarah Thies; Uli Kazmaier
Journal:  Beilstein J Org Chem       Date:  2011-09-19       Impact factor: 2.883

4.  Thiazole formation through a modified Gewald reaction.

Authors:  Carl J Mallia; Lukas Englert; Gary C Walter; Ian R Baxendale
Journal:  Beilstein J Org Chem       Date:  2015-05-26       Impact factor: 2.883

5.  A universal isocyanide for diverse heterocycle syntheses.

Authors:  Pravin Patil; Kareem Khoury; Eberhardt Herdtweck; Alexander Dömling
Journal:  Org Lett       Date:  2014-10-29       Impact factor: 6.005

6.  Cysteine Isocyanide in Multicomponent Reaction: Synthesis of Peptido-Mimetic 1,3-Azoles.

Authors:  Thimmalapura M Vishwanatha; Katarzyna Kurpiewska; Justyna Kalinowska-Tłuścik; Alexander Dömling
Journal:  J Org Chem       Date:  2017-08-25       Impact factor: 4.354

7.  Chemo- and Stereoselective Synthesis of Substituted Thiazoles from tert-Alcohols Bearing Alkene and Alkyne Groups with Alkaline Earth Catalysts.

Authors:  Srinivasarao Yaragorla; Dandugula Sneha Latha
Journal:  ACS Omega       Date:  2022-09-15

8.  Synthetic studies towards bottromycin.

Authors:  Stefanie Ackermann; Hans-Georg Lerchen; Dieter Häbich; Angelika Ullrich; Uli Kazmaier
Journal:  Beilstein J Org Chem       Date:  2012-10-01       Impact factor: 2.883
  8 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.