Literature DB >> 16086097

Pre-irradiation 9-amino [20s] camptothecin (9-AC) in patients with newly diagnosed glioblastoma multiforme.

Daniel Farray1, Manmeet S Ahluwalia, Josette Snyder, Gene H Barnett, Bruce H Cohen, John H Suh, David M Peereboom.   

Abstract

PURPOSE: To evaluate the efficacy of 9-amino [20s] camptothecin (9-AC) given before radiation therapy to patients with newly diagnosed glioblastoma multiforme (GBM).
METHODS: Eligible patients had newly diagnosed GBM who had residual measurable contrast-enhancing tumor. The trial was a phase 2 trial of 9-AC at 1100 microg/m2 /24 h infused over 72 h every two weeks for up to six cycles in patients with newly diagnosed GBM before radiation therapy.
RESULTS: Fourteen patients entered the study and all were evaluable. All of the patients had progressive disease by imaging criteria after at least two cycles of 9-AC (1 month). The median overall survival was 7.5 months (range 1.5-18 months). The most common adverse event was transient lymphopenia (grade 3-4). One patient developed grade 4 neutropenic fever that resolved after three days of diagnosis.
CONCLUSIONS: 9-AC lacks activity against glioblastoma multiforme (GBM). Further studies looking at the efficacy of 9-AC in GBM may be futile.

Entities:  

Mesh:

Substances:

Year:  2006        PMID: 16086097     DOI: 10.1007/s10637-005-2464-5

Source DB:  PubMed          Journal:  Invest New Drugs        ISSN: 0167-6997            Impact factor:   3.651


  19 in total

Review 1.  DNA topoisomerases.

Authors:  J C Wang
Journal:  Annu Rev Biochem       Date:  1985       Impact factor: 23.643

2.  Cancer statistics, 2000.

Authors:  R T Greenlee; T Murray; S Bolden; P A Wingo
Journal:  CA Cancer J Clin       Date:  2000 Jan-Feb       Impact factor: 508.702

3.  Topotecan treatment of adults with primary malignant glioma. The Brain Tumor Center at Duke.

Authors:  H S Friedman; T Kerby; S Fields; J E Zilisch; D Graden; R E McLendon; P J Houghton; S Arbuck; I Cokgor; A H Friedman
Journal:  Cancer       Date:  1999-03-01       Impact factor: 6.860

4.  Irinotecan therapy in adults with recurrent or progressive malignant glioma.

Authors:  H S Friedman; W P Petros; A H Friedman; L J Schaaf; T Kerby; J Lawyer; M Parry; P J Houghton; S Lovell; K Rasheed; T Cloughsey; E S Stewart; O M Colvin; J M Provenzale; R E McLendon; D D Bigner; I Cokgor; M Haglund; J Rich; D Ashley; J Malczyn; G L Elfring; L L Miller
Journal:  J Clin Oncol       Date:  1999-05       Impact factor: 44.544

5.  A North Central Cancer Treatment Group phase II trial of topotecan in relapsed gliomas.

Authors:  P A Burch; A M Bernath; T L Cascino; B W Scheithauer; P Novotny; S Nair; J C Buckner; D M Pfeifle; J W Kugler; L K Tschetter
Journal:  Invest New Drugs       Date:  2000-08       Impact factor: 3.850

6.  Phase I and pharmacologic study of 9-aminocamptothecin given by 72-hour infusion in adult cancer patients.

Authors:  W Dahut; N Harold; C Takimoto; C Allegra; A Chen; J M Hamilton; S Arbuck; M Sorensen; F Grollman; H Nakashima; R Lieberman; M Liang; W Corse; J Grem
Journal:  J Clin Oncol       Date:  1996-04       Impact factor: 44.544

7.  Temozolomide in combination with irinotecan for treatment of recurrent malignant glioma.

Authors:  Michael L Gruber; Ward P Buster
Journal:  Am J Clin Oncol       Date:  2004-02       Impact factor: 2.339

8.  Altered irinotecan pharmacokinetics in pediatric high-grade glioma patients receiving enzyme-inducing anticonvulsant therapy.

Authors:  Kristine R Crews; Clinton F Stewart; Dana Jones-Wallace; Stephen J Thompson; Peter J Houghton; Richard L Heideman; Maryam Fouladi; Daniel C Bowers; Murali M Chintagumpala; Amar Gajjar
Journal:  Clin Cancer Res       Date:  2002-07       Impact factor: 12.531

9.  A phase I and pharmacokinetic study of a new camptothecin derivative, 9-aminocamptothecin.

Authors:  E Rubin; V Wood; A Bharti; D Trites; C Lynch; S Hurwitz; S Bartel; S Levy; A Rosowsky; D Toppmeyer
Journal:  Clin Cancer Res       Date:  1995-03       Impact factor: 12.531

Review 10.  Current perspectives on camptothecins in cancer treatment.

Authors:  J Dancey; E A Eisenhauer
Journal:  Br J Cancer       Date:  1996-08       Impact factor: 7.640

View more
  1 in total

Review 1.  Camptothecin (CPT) and its derivatives are known to target topoisomerase I (Top1) as their mechanism of action: did we miss something in CPT analogue molecular targets for treating human disease such as cancer?

Authors:  Fengzhi Li; Tao Jiang; Qingyong Li; Xiang Ling
Journal:  Am J Cancer Res       Date:  2017-12-01       Impact factor: 6.166

  1 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.