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12 in total

1. Diastereoselective addition of monoorganocuprates to a chiral fumarate: reaction development and synthesis of (-)-dihydroprotolichesterinic acid.

Authors: J Caleb Hethcox; Charles S Shanahan; Stephen F Martin
Journal: Tetrahedron Date: 2015-09-16 Impact factor: 2.457

2. Structurally simple, potent, Plasmodium selective farnesyltransferase inhibitors that arrest the growth of malaria parasites.

Authors: Matthew P Glenn; Sung-Youn Chang; Carrie Hornéy; Kasey Rivas; Kohei Yokoyama; Erin E Pusateri; Steven Fletcher; Christopher G Cummings; Frederick S Buckner; Prakash R Pendyala; Debopam Chakrabarti; Saïd M Sebti; Michael Gelb; Wesley C Van Voorhis; Andrew D Hamilton
Journal: J Med Chem Date: 2006-09-21 Impact factor: 7.446

3. Structures of Cryptococcus neoformans protein farnesyltransferase reveal strategies for developing inhibitors that target fungal pathogens.

Authors: Michael A Hast; Connie B Nichols; Stephanie M Armstrong; Shannon M Kelly; Homme W Hellinga; J Andrew Alspaugh; Lorena S Beese
Journal: J Biol Chem Date: 2011-08-04 Impact factor: 5.157

4. Manumycin A Is a Potent Inhibitor of Mammalian Thioredoxin Reductase-1 (TrxR-1).

Authors: Anupama Tuladhar; Kathleen S Rein
Journal: ACS Med Chem Lett Date: 2018-03-05 Impact factor: 4.345

5. Structure-based design and synthesis of potent, ethylenediamine-based, mammalian farnesyltransferase inhibitors as anticancer agents.

Authors: Steven Fletcher; Erin Pusateri Keaney; Christopher G Cummings; Michelle A Blaskovich; Michael A Hast; Matthew P Glenn; Sung-Youn Chang; Cynthia J Bucher; Ryan J Floyd; William P Katt; Michael H Gelb; Wesley C Van Voorhis; Lorena S Beese; Said M Sebti; Andrew D Hamilton
Journal: J Med Chem Date: 2010-10-14 Impact factor: 7.446

6. Isoprenoid biosynthesis inhibition disrupts Rab5 localization and food vacuolar integrity in Plasmodium falciparum.

Authors: Ruth Howe; Megan Kelly; John Jimah; Dana Hodge; Audrey R Odom
Journal: Eukaryot Cell Date: 2012-12-07

7. Potent, Plasmodium-selective farnesyltransferase inhibitors that arrest the growth of malaria parasites: structure-activity relationships of ethylenediamine-analogue scaffolds and homology model validation.

Authors: Steven Fletcher; Christopher G Cummings; Kasey Rivas; William P Katt; Carrie Hornéy; Frederick S Buckner; Debopam Chakrabarti; Saïd M Sebti; Michael H Gelb; Wesley C Van Voorhis; Andrew D Hamilton
Journal: J Med Chem Date: 2008-08-08 Impact factor: 7.446

8. Imidazole-containing farnesyltransferase inhibitors: 3D quantitative structure-activity relationships and molecular docking.

Authors: Aihua Xie; Srinivas Odde; Sivaprakasam Prasanna; Robert J Doerksen
Journal: J Comput Aided Mol Des Date: 2009-05-29 Impact factor: 3.686

9. Structural basis for binding and selectivity of antimalarial and anticancer ethylenediamine inhibitors to protein farnesyltransferase.

Authors: Michael A Hast; Steven Fletcher; Christopher G Cummings; Erin E Pusateri; Michelle A Blaskovich; Kasey Rivas; Michael H Gelb; Wesley C Van Voorhis; Said M Sebti; Andrew D Hamilton; Lorena S Beese
Journal: Chem Biol Date: 2009-02-27

10. Protein Prenylation and Hsp40 in Thermotolerance of Plasmodium falciparum Malaria Parasites.

Authors: Emily S Mathews; Andrew J Jezewski; Audrey R Odom John
Journal: mBio Date: 2021-06-29 Impact factor: 7.867