Literature DB >> 15979309

Glycosidase inhibition by 1-glycosyl-4-phenyl triazoles.

Lauren L Rossi1, Amit Basu.   

Abstract

1-Glycosyl-4-phenyl triazoles have been prepared via a copper-mediated [3+2] cycloaddition of glycosyl azides with phenylacetylene. These triazoles have been evaluated for their ability to inhibit the enzymatic activity of glycosidases.

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Year:  2005        PMID： 15979309     DOI： 10.1016/j.bmcl.2005.05.081

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  7 in total

1.  Anti-bacterial glycosyl triazoles - Identification of an N-acetylglucosamine derivative with bacteriostatic activity against Bacillus.

Authors:  Helene Kuhn; Danielle Gutelius; Eimear Black; Christina Nadolny; Amit Basu; Christopher Reid
Journal:  Medchemcomm       Date:  2014-08       Impact factor: 3.597

2.  C(1)-/C(2)-aromatic-imino-glyco-conjugates: experimental and computational studies of binding, inhibition and docking aspects towards glycosidases isolated from soybean and jack bean.

Authors:  Amit Kumar; Nitin K Singhal; Balaji Ramanujam; Atanu Mitra; Nagender R Rameshwaram; Siva K Nadimpalli; Chebrolu P Rao
Journal:  Glycoconj J       Date:  2008-10-25       Impact factor: 2.916

3.  Mechanistic insights into the inhibition of endo-β 1,4 xyloglucan hydrolase by a classical aspartic protease inhibitor.

Authors:  Vishnu Menon; Mala Rao
Journal:  J Fluoresc       Date:  2012-12-05       Impact factor: 2.217

4.  'Click chemistry' synthesis of 1-(α-D-mannopyranosyl)-1,2,3-triazoles for inhibition of α-mannosidases.

Authors:  Monika Poláková; Rhiannon Stanton; Iain B H Wilson; Ivana Holková; Sergej Šesták; Eva Machová; Zuzana Jandová; Juraj Kóňa
Journal:  Carbohydr Res       Date:  2015-01-19       Impact factor: 2.104

Review 5.  Advancements in the mechanistic understanding of the copper-catalyzed azide-alkyne cycloaddition.

Authors:  Regina Berg; Bernd F Straub
Journal:  Beilstein J Org Chem       Date:  2013-12-02       Impact factor: 2.883

6.  Gram scale production of 1-azido-β-d-glucose via enzyme catalysis for the synthesis of 1,2,3-triazole-glucosides.

Authors:  Jaggaiah N Gorantla; Salila Pengthaisong; Sunaree Choknud; Teadkait Kaewpuang; Tanaporn Manyum; Vinich Promarak; James R Ketudat Cairns
Journal:  RSC Adv       Date:  2019-02-20       Impact factor: 3.361

7.  Carbohydrate-Functionalized Triazolylidene Iridium Complexes: Hydrogenation Catalysis in Water with Asymmetric Induction.

Authors:  Joseph P Byrne; Lidia Delgado; Francesca Paradisi; Martin Albrecht
Journal:  ChemCatChem       Date:  2022-03-11       Impact factor: 5.497
  7 in total

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