Literature DB >> 15978659

A phase II evaluation of flavopiridol as second-line chemotherapy of endometrial carcinoma: a Gynecologic Oncology Group study.

Edward C Grendys1, John A Blessing, Robert Burger, James Hoffman.   

Abstract

OBJECTIVE: A phase II study was conducted to determine the efficacy of single agent flavopiridol therapy in patients with recurrent or persistent endometrial adenocarcinoma refractory to established treatments.
METHODS: Eligible patients with measurable disease who failed primary therapy including one cytotoxic regimen were eligible for the trial. They were treated with single agent flavopiridol (50 mg/m(2)/day, IV bolus days 1, 2, 3). Treatment was repeated every 21 days with dose adjustments made for toxicity. Patients were treated until progression of disease or adverse side effects precluded further therapy.
RESULTS: A total of 26 patients were enrolled in the study of whom, 23 patients were eligible. There were no objective responses. Five patients had stable disease (22%), 15 (65%) had increasing disease, and response could not be assessed in 3 (13%). The most frequent side effects included anemia, neutropenia, and diarrhea, all of which appeared manageable.
CONCLUSION: Flavopiridol as a single agent in the above dosing schedule appears to have minimal activity as second-line chemotherapy of endometrial adenocarcinoma.

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Year:  2005        PMID: 15978659     DOI: 10.1016/j.ygyno.2005.05.017

Source DB:  PubMed          Journal:  Gynecol Oncol        ISSN: 0090-8258            Impact factor:   5.482


  13 in total

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Authors:  Kathleen N Moore; Michael W Sill; Meaghan E Tenney; Christopher J Darus; David Griffin; Theresa L Werner; Peter G Rose; Robert Behrens
Journal:  Gynecol Oncol       Date:  2015-07-11       Impact factor: 5.482

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9.  The flavonoid glycosides, myricitrin, gossypin and naringin exert anxiolytic action in mice.

Authors:  Sebastian P Fernandez; Michael Nguyen; Tin Thing Yow; Cindy Chu; Graham A R Johnston; Jane R Hanrahan; Mary Chebib
Journal:  Neurochem Res       Date:  2009-04-23       Impact factor: 3.996

10.  A phase 1 study of SNS-032 (formerly BMS-387032), a potent inhibitor of cyclin-dependent kinases 2, 7 and 9 administered as a single oral dose and weekly infusion in patients with metastatic refractory solid tumors.

Authors:  Elisabeth I Heath; Keith Bible; Robert E Martell; Daniel C Adelman; Patricia M Lorusso
Journal:  Invest New Drugs       Date:  2007-10-16       Impact factor: 3.850

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