Literature DB >> 15863316

Structure-activity relationships of arylbenzofuran H3 receptor antagonists.

Gregory A Gfesser1, Ramin Faghih, Youssef L Bennani, Michael P Curtis, Timothy A Esbenshade, Arthur A Hancock, Marlon D Cowart.   

Abstract

An SAR study of histamine H3 receptor antagonists based on substituted (R)-2-methyl-1-[2-(5-phenyl-benzofuran-2-yl)-ethyl]-pyrrolidines is presented.

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Year:  2005        PMID： 15863316     DOI： 10.1016/j.bmcl.2005.03.047

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  7 in total

1.  A new approach to fused furan ring systems and benzofurans: Intramolecular cyclization reactions of unsaturated acyloxy sulfone derivatives.

Authors:  Yuan Liu; Hollie K Jacobs; Aravamudan S Gopalan
Journal:  Tetrahedron Lett       Date:  2011-06-08       Impact factor: 2.415

2.  Parallel synthesis of a multi-substituted benzo[b]furan library.

Authors:  Chul-Hee Cho; Benjamin Neuenswander; Gerald H Lushington; Richard C Larock
Journal:  J Comb Chem       Date:  2008-10-21

3.  Synthesis of multi-functionalized benzofurans through the condensation of ninhydrin and phenols using SSA as a recyclable heterogeneous acid catalyst.

Authors:  Ashis Kundu; Animesh Pramanik
Journal:  Mol Divers       Date:  2016-02-01       Impact factor: 2.943

4.  Comparison of Different 2D and 3D-QSAR Methods on Activity Prediction of Histamine H3 Receptor Antagonists.

Authors:  Siavoush Dastmalchi; Maryam Hamzeh-Mivehroud; Karim Asadpour-Zeynali
Journal:  Iran J Pharm Res       Date:  2012       Impact factor: 1.696

5.  Rapid regio- and multi-coupling reactivity of 2,3-dibromobenzofurans with atom-economic triarylbismuths under palladium catalysis.

Authors:  Maddali L N Rao; Jalindar B Talode; Venneti N Murty
Journal:  Beilstein J Org Chem       Date:  2016-09-22       Impact factor: 2.883

Review 6.  QSAR Modeling of Histamine H3R Antagonists/inverse Agonists as Future Drugs for Neurodegenerative Diseases.

Authors:  Michelle Fidelis Correa; Joao Paulo Dos Santos Fernandes
Journal:  Curr Neuropharmacol       Date:  2018       Impact factor: 7.363

7.  Palladium-catalyzed Tsuji-Trost-type reaction of benzofuran-2-ylmethyl acetates with nucleophiles.

Authors:  Antonio Arcadi; Giancarlo Fabrizi; Andrea Fochetti; Francesca Ghirga; Antonella Goggiamani; Antonia Iazzetti; Federico Marrone; Giulia Mazzoccanti; Andrea Serraiocco
Journal:  RSC Adv       Date:  2021-01-04       Impact factor: 3.361
  7 in total

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