| Literature DB >> 15771435 |
Jan Heeres1, Marc R de Jonge, Lucien M H Koymans, Frits F D Daeyaert, Maarten Vinkers, Koen J A Van Aken, Eddy Arnold, Kalyan Das, Amuri Kilonda, Georges J Hoornaert, Frans Compernolle, Marek Cegla, Rasha A Azzam, Koen Andries, Marie-Pierre de Béthune, Hilde Azijn, Rudi Pauwels, Paul J Lewi, Paul A J Janssen.
Abstract
A series of novel pyrazinones designed as non-nucleoside reverse transcriptase inhibitors (NNRTIs) was synthesized and their anti-HIV structure-activity relationship (SAR) was studied.Entities:
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Year: 2005 PMID: 15771435 DOI: 10.1021/jm040829e
Source DB: PubMed Journal: J Med Chem ISSN: 0022-2623 Impact factor: 7.446