Literature DB >> 15753761

Analysis of the brain bioavailability of peripherally administered magnesium sulfate: A study in humans with acute brain injury undergoing prolonged induced hypermagnesemia.

J Andrew McKee1, Randall P Brewer, Gary E Macy, Barbara Phillips-Bute, Kurt A Campbell, Cecil O Borel, James D Reynolds, David S Warner.   

Abstract

OBJECTIVE: Based on preclinical investigations, magnesium sulfate (MgSO4) has gained interest as a neuroprotective agent. However, the ability of peripherally administered MgSO4 to penetrate the blood-brain barrier is limited in normal brain. The current study measured the passage of intravenously administered Mg into cerebrospinal fluid in patients with brain injury requiring ventricular drainage.
DESIGN: A prospective evaluation of the cerebrospinal fluid total and ionized magnesium concentration, [Mg], during sustained hypermagnesemia was performed.
SETTING: Neurosciences intensive care unit at a major teaching institution. PATIENTS: Thirty patients with acute brain injury secondary to subarachnoid hemorrhage, traumatic brain injury, primary intracerebral hemorrhage, subdural hematoma, brain tumor, central nervous system infection, or ischemic stroke were studied.
INTERVENTIONS: Patients underwent 24 hrs of induced hypermagnesemia during which total and ionized cerebrospinal fluid [Mg] was measured. Serum [Mg] was adjusted to 2.1-2.5 mmol/L. Cerebrospinal fluid [Mg] was measured at baseline, at 12 and 24 hrs after onset of infusion, and at 12 hrs following infusion termination.
MEASUREMENTS AND MAIN RESULTS: At baseline, total (1.25 +/- 0.14 mmol/L) and ionized (0.80 +/- 0.10 mmol/L) cerebrospinal fluid [Mg] was greater than serum total (0.92 +/- 0.18 mmol/L) and ionized (0.63 +/- 0.07 mmol/L) [Mg] (p < .05). Total (1.43 +/- 0.13 mmol/L) and ionized (0.89 +/- 0.12 mmol/L) cerebrospinal fluid [Mg] was maximally increased by 15% and 11% relative to baseline, respectively, during induced hypermagnesemia (p < .05).
CONCLUSIONS: Hypermagnesemia produced only marginal increases in total and ionized cerebrospinal fluid [Mg]. Regulation of cerebrospinal fluid [Mg] is largely maintained following acute brain injury and limits the brain bioavailability of MgSO4.

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Year:  2005        PMID: 15753761     DOI: 10.1097/01.ccm.0000156293.35868.b2

Source DB:  PubMed          Journal:  Crit Care Med        ISSN: 0090-3493            Impact factor:   7.598


  17 in total

Review 1.  Magnesium neuroprotection is limited in humans with acute brain injury.

Authors:  J Andrew McKee; Randall P Brewer; Gary E Macy; Cecil O Borel; James D Reynolds; David S Warner
Journal:  Neurocrit Care       Date:  2005       Impact factor: 3.210

Review 2.  Multifunctional drugs for head injury.

Authors:  Robert Vink; Alan J Nimmo
Journal:  Neurotherapeutics       Date:  2009-01       Impact factor: 7.620

3.  Incidence, hemodynamic, and electrical characteristics of spreading depolarization in a swine model are affected by local but not by intravenous application of magnesium.

Authors:  Edgar Santos; Fiorella León; Humberto Silos; Renan Sanchez-Porras; C William Shuttleworth; Andreas Unterberg; Oliver W Sakowitz
Journal:  J Cereb Blood Flow Metab       Date:  2016-09-28       Impact factor: 6.200

4.  Long-term enhancement of synaptic transmission between antennal lobe and mushroom body in cultured Drosophila brain.

Authors:  Kohei Ueno; Shintaro Naganos; Yukinori Hirano; Junjiro Horiuchi; Minoru Saitoe
Journal:  J Physiol       Date:  2012-10-01       Impact factor: 5.182

5.  Mg(2+) block of Drosophila NMDA receptors is required for long-term memory formation and CREB-dependent gene expression.

Authors:  Tomoyuki Miyashita; Yoshiaki Oda; Junjiro Horiuchi; Jerry C P Yin; Takako Morimoto; Minoru Saitoe
Journal:  Neuron       Date:  2012-06-07       Impact factor: 17.173

6.  High dose magnesium infusions are not associated with increased pressor requirements after carotid endarterectomy.

Authors:  Camay Chiu; Eric J Heyer; Anita D Rampersad; Joseph Zurica; Eugene Ornstein; Daniel H Sahlein; Robert R Sciacca; E Sander Connolly
Journal:  Neurosurgery       Date:  2006-01       Impact factor: 4.654

Review 7.  Use of magnesium in traumatic brain injury.

Authors:  Ananda P Sen; Anil Gulati
Journal:  Neurotherapeutics       Date:  2010-01       Impact factor: 7.620

8.  Chronic dietary magnesium-L-threonate speeds extinction and reduces spontaneous recovery of a conditioned taste aversion.

Authors:  G Andrew Mickley; Nita Hoxha; Joseph L Luchsinger; Morgan M Rogers; Nathanael R Wiles
Journal:  Pharmacol Biochem Behav       Date:  2013-03-06       Impact factor: 3.533

9.  Intraoperative magnesium administration does not improve neurocognitive function after cardiac surgery.

Authors:  Joseph P Mathew; William D White; David B Schinderle; Mihai V Podgoreanu; Miles Berger; Carmelo A Milano; Daniel T Laskowitz; Mark Stafford-Smith; James A Blumenthal; Mark F Newman
Journal:  Stroke       Date:  2013-10-08       Impact factor: 7.914

10.  Update in the treatment of traumatic brain injury.

Authors:  Scott E Bell; Roman Hlatky
Journal:  Curr Treat Options Neurol       Date:  2006-03       Impact factor: 3.972

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