Literature DB >> 15739093

The effect of citalopram hydrobromide on 5-HT2A receptors in the impulsive-aggressive dog, as measured with 123I-5-I-R91150 SPECT.

K Peremans1, K Audenaert, Y Hoybergs, A Otte, I Goethals, I Gielen, P Blankaert, M Vervaet, C van Heeringen, R Dierckx.   

Abstract

PURPOSE: Involvement of the serotonergic system in impulsive aggression has been demonstrated in both human and animal studies. The purpose of the present study was to investigate the effect of citalopram hydrobromide (a selective serotonin re-uptake inhibitor) on the 5-HT(2A) receptor and brain perfusion in impulsive-aggressive dogs by means of single-photon emission computed tomography.
METHODS: The binding index of the radioligand (123)I-5-I-R91150 was measured before and after treatment with citalopram hydrobromide in nine impulsive-aggressive dogs. Regional perfusion was measured with (99m)Tc-ethyl cysteinate dimer (ECD). Behaviour was assessed before treatment and again after 6 weeks of treatment.
RESULTS: A correlation was found between decreased binding and behavioural improvement in eight out of nine dogs. The 5-HT(2A) receptor binding index was significantly reduced after citalopram hydrobromide treatment in all cortical regions but not in the subcortical area. None of the dogs displayed alterations in perfusion on the post-treatment scans.
CONCLUSION: This study supports previous findings regarding the involvement of the serotonergic system in impulsive aggression in dogs in general. More specifically, the effect of treatment on the 5-HT(2A) receptor binding index could be demonstrated and the decreased binding index correlated with behavioural improvement.

Entities:  

Mesh:

Substances:

Year:  2005        PMID: 15739093     DOI: 10.1007/s00259-005-1772-5

Source DB:  PubMed          Journal:  Eur J Nucl Med Mol Imaging        ISSN: 1619-7070            Impact factor:   9.236


  51 in total

Review 1.  Assessment, management, and prognosis of canine dominance-related aggression.

Authors:  I R Reisner
Journal:  Vet Clin North Am Small Anim Pract       Date:  1997-05       Impact factor: 2.093

2.  The effects of single dose nefazodone and paroxetine upon 5-HT2A binding potential in humans using [18F]-setoperone PET.

Authors:  J H Meyer; R Cho; S Kennedy; S Kapur
Journal:  Psychopharmacology (Berl)       Date:  1999-06       Impact factor: 4.530

3.  Serotonergic blunting to meta-chlorophenylpiperazine (m-CPP) highly correlates with sustained childhood abuse in impulsive and autoaggressive female borderline patients.

Authors:  T Rinne; H G Westenberg; J A den Boer; W van den Brink
Journal:  Biol Psychiatry       Date:  2000-03-15       Impact factor: 13.382

4.  Reduction by paroxetine of suicidal behavior in patients with repeated suicide attempts but not major depression.

Authors:  R J Verkes; R C Van der Mast; M W Hengeveld; J P Tuyl; A H Zwinderman; G M Van Kempen
Journal:  Am J Psychiatry       Date:  1998-04       Impact factor: 18.112

5.  Effects of chronic paroxetine administration on measures of aggressive and impulsive responses of adult males with a history of conduct disorder.

Authors:  Don R Cherek; Scott D Lane; Cynthia J Pietras; Joel L Steinberg
Journal:  Psychopharmacology (Berl)       Date:  2001-10-12       Impact factor: 4.530

6.  Activation of 5-HT2A receptors impairs response control of rats in a five-choice serial reaction time task.

Authors:  T Koskinen; S Ruotsalainen; T Puumala; R Lappalainen; E Koivisto; P T Männistö; J Sirviö
Journal:  Neuropharmacology       Date:  2000-01-28       Impact factor: 5.250

7.  Increase in extracellular serotonin produced by uptake inhibitors is enhanced after chronic treatment with fluoxetine.

Authors:  J J Rutter; C Gundlah; S B Auerbach
Journal:  Neurosci Lett       Date:  1994-04-25       Impact factor: 3.046

8.  Fenfluramine challenge, self-injurious behavior, and aggression in rhesus monkeys.

Authors:  Stefan Tiefenbacher; Matthew D Davenport; Melinda A Novak; Amber L Pouliot; Jerrold S Meyer
Journal:  Physiol Behav       Date:  2003-11

9.  5-HT(2A) receptor binding is reduced in drug-naive and unchanged in SSRI-responder depressed patients compared to healthy controls: a PET study.

Authors:  Cristina Messa; Cristina Colombo; Rosa Maria Moresco; Clara Gobbo; Laura Galli; Giovanni Lucignani; Maria Carla Gilardi; Giovanna Rizzo; Enrico Smeraldi; Raffaella Zanardi; Francesc Artigas; Ferruccio Fazio
Journal:  Psychopharmacology (Berl)       Date:  2003-03-11       Impact factor: 4.530

10.  Excessive mortality in young free-ranging male nonhuman primates with low cerebrospinal fluid 5-hydroxyindoleacetic acid concentrations.

Authors:  J D Higley; P T Mehlman; S B Higley; B Fernald; J Vickers; S G Lindell; D M Taub; S J Suomi; M Linnoila
Journal:  Arch Gen Psychiatry       Date:  1996-06
View more
  6 in total

1.  Variation in the gene encoding the serotonin 2A receptor is associated with outcome of antidepressant treatment.

Authors:  Francis J McMahon; Silvia Buervenich; Dennis Charney; Robert Lipsky; A John Rush; Alexander F Wilson; Alexa J M Sorant; George J Papanicolaou; Gonzalo Laje; Maurizio Fava; Madhukar H Trivedi; Stephen R Wisniewski; Husseini Manji
Journal:  Am J Hum Genet       Date:  2006-03-20       Impact factor: 11.025

Review 2.  Measuring serotonin synthesis: from conventional methods to PET tracers and their (pre)clinical implications.

Authors:  Anniek K D Visser; Aren van Waarde; Antoon T M Willemsen; Fokko J Bosker; Paul G M Luiten; Johan A den Boer; Ido P Kema; Rudi A J O Dierckx
Journal:  Eur J Nucl Med Mol Imaging       Date:  2010-11-27       Impact factor: 9.236

3.  Long-term citalopram maintenance in mice: selective reduction of alcohol-heightened aggression.

Authors:  Elizabeth E Caldwell; Klaus A Miczek
Journal:  Psychopharmacology (Berl)       Date:  2007-10-20       Impact factor: 4.530

Review 4.  The effect of increased serotonergic neurotransmission on aggression: a critical meta-analytical review of preclinical studies.

Authors:  Maria Carrillo; Lesley A Ricci; Glen A Coppersmith; Richard H Melloni
Journal:  Psychopharmacology (Berl)       Date:  2009-04-30       Impact factor: 4.530

5.  Similar striatal gene expression profiles in the striatum of the YAC128 and HdhQ150 mouse models of Huntington's disease are not reflected in mutant Huntingtin inclusion prevalence.

Authors:  Zubeyde Bayram-Weston; Timothy C Stone; Peter Giles; Linda Elliston; Nari Janghra; Gemma V Higgs; Peter A Holmans; Stephen B Dunnett; Simon P Brooks; Lesley Jones
Journal:  BMC Genomics       Date:  2015-12-21       Impact factor: 3.969

6.  Hostility in medication-resistant major depression and comorbid generalized anxiety disorder is related to increased hippocampal-amygdala 5-HT2A receptor density.

Authors:  Chris Baeken; Yanfeng Xu; Guo-Rong Wu; Robrecht Dockx; Kathelijne Peremans; Rudi De Raedt
Journal:  Eur Arch Psychiatry Clin Neurosci       Date:  2021-04-27       Impact factor: 5.270

  6 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.